JP2008539267A - ベンズイソオキサゾールピペリジン化合物及びその使用方法 - Google Patents

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Publication number

JP2008539267A

JP2008539267A JP2008509128A JP2008509128A JP2008539267A JP 2008539267 A JP2008539267 A JP 2008539267A JP 2008509128 A JP2008509128 A JP 2008509128A JP 2008509128 A JP2008509128 A JP 2008509128A JP 2008539267 A JP2008539267 A JP 2008539267A

Authority

JP

Japan

Prior art keywords

conhs

sleep

alkyl

compound

compound according

Prior art date

2005-04-26

Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)

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• 238000000034 method Methods 0.000 title abstract description 27
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• 230000007958 sleep Effects 0.000 claims abstract description 145
• 150000001875 compounds Chemical class 0.000 claims description 302
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• 125000000217 alkyl group Chemical group 0.000 claims description 97
• 229910052739 hydrogen Inorganic materials 0.000 claims description 71
• 150000003839 salts Chemical class 0.000 claims description 68
• 208000019116 sleep disease Diseases 0.000 claims description 67
• 238000011282 treatment Methods 0.000 claims description 62
• OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims description 58
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• 229910052794 bromium Inorganic materials 0.000 claims description 30
• 229910052801 chlorine Inorganic materials 0.000 claims description 30
• 229910052731 fluorine Inorganic materials 0.000 claims description 30
• 229910052717 sulfur Inorganic materials 0.000 claims description 29
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• 239000000651 prodrug Substances 0.000 claims description 26
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