JP2008534513A5 - - Google Patents

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Publication number
JP2008534513A5
JP2008534513A5 JP2008503238A JP2008503238A JP2008534513A5 JP 2008534513 A5 JP2008534513 A5 JP 2008534513A5 JP 2008503238 A JP2008503238 A JP 2008503238A JP 2008503238 A JP2008503238 A JP 2008503238A JP 2008534513 A5 JP2008534513 A5 JP 2008534513A5
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JP
Japan
Prior art keywords
santillietal
methylmercaptopyrimidine
heterocycl
ocl
dihydroxy
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JP2008503238A
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JP2008534513A (ja
JP5037487B2 (ja
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Priority claimed from PCT/US2006/010855 external-priority patent/WO2006104915A2/en
Publication of JP2008534513A publication Critical patent/JP2008534513A/ja
Publication of JP2008534513A5 publication Critical patent/JP2008534513A5/ja
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Publication of JP5037487B2 publication Critical patent/JP5037487B2/ja
Expired - Fee Related legal-status Critical Current
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Description

出発物質１−スキーム７は、市販されている４，６−ジヒドロキシ−２−メチルメルカプトピリミジンから、文献で公知の方法、例えば、ＯＣｌ３およびＤＭＦを用いる、Santillietal., J. Heterocycl. Chem. (1971), 445-53に記載の方法を用いて得ることができる。

JP2008503238A 2005-03-25 2006-03-24 新規化合物 Expired - Fee Related JP5037487B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US66531505P 2005-03-25 2005-03-25
US60/665,315 2005-03-25
PCT/US2006/010855 WO2006104915A2 (en) 2005-03-25 2006-03-24 8-PHENYL-7,8-DIHYDROPYRIDO[2,3-d]PYRIMIDIN-7-ONES AND THEIR USE AS PHARMACEUTICALS

Publications (3)

Publication Number Publication Date
JP2008534513A JP2008534513A (ja) 2008-08-28
JP2008534513A5 true JP2008534513A5 (ja) 2010-01-14
JP5037487B2 JP5037487B2 (ja) 2012-09-26

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ID=37053943

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JP2008503238A Expired - Fee Related JP5037487B2 (ja) 2005-03-25 2006-03-24 新規化合物

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US (3) US8207176B2 (ja)
EP (3) EP1868611B1 (ja)
JP (1) JP5037487B2 (ja)
KR (1) KR101235497B1 (ja)
CN (4) CN102746300A (ja)
AR (1) AR053346A1 (ja)
AU (1) AU2006229993B2 (ja)
BR (1) BRPI0609437A2 (ja)
CA (1) CA2602553C (ja)
EA (1) EA012875B1 (ja)
ES (2) ES2426251T3 (ja)
HK (1) HK1111422A1 (ja)
IL (1) IL185870A (ja)
MA (1) MA29341B1 (ja)
MX (1) MX2007011856A (ja)
MY (2) MY145343A (ja)
NO (1) NO20075275L (ja)
NZ (1) NZ561237A (ja)
PE (2) PE20100737A1 (ja)
SG (1) SG166771A1 (ja)
TW (1) TWI389690B (ja)
UA (1) UA95444C2 (ja)
UY (1) UY29440A1 (ja)
WO (1) WO2006104915A2 (ja)
ZA (1) ZA200707564B (ja)

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