ATE240325T1 - Verfahren zur herstellung von biphenylderivaten - Google Patents

Verfahren zur herstellung von biphenylderivaten

Info

Publication number
ATE240325T1
ATE240325T1 AT96918189T AT96918189T ATE240325T1 AT E240325 T1 ATE240325 T1 AT E240325T1 AT 96918189 T AT96918189 T AT 96918189T AT 96918189 T AT96918189 T AT 96918189T AT E240325 T1 ATE240325 T1 AT E240325T1
Authority
AT
Austria
Prior art keywords
tert
butyl
tetrazol
pyrido
pyrimidin
Prior art date
Application number
AT96918189T
Other languages
English (en)
Inventor
Pierre Giguere
Silvio Iera
Michel Bernatchez
Giuseppe Barreca
Graziano Castaldi
Vincenzo Cannata
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/657,490 external-priority patent/US5760220A/en
Application filed by Wyeth Corp filed Critical Wyeth Corp
Application granted granted Critical
Publication of ATE240325T1 publication Critical patent/ATE240325T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT96918189T 1995-06-07 1996-06-06 Verfahren zur herstellung von biphenylderivaten ATE240325T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US47859295A 1995-06-07 1995-06-07
US08/657,490 US5760220A (en) 1995-06-07 1996-06-04 Process for preparation of biphenyl derivatives
PCT/US1996/009117 WO1996040684A1 (en) 1995-06-07 1996-06-06 Process for preparation of biphenyl derivatives

Publications (1)

Publication Number Publication Date
ATE240325T1 true ATE240325T1 (de) 2003-05-15

Family

ID=27045956

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96918189T ATE240325T1 (de) 1995-06-07 1996-06-06 Verfahren zur herstellung von biphenylderivaten

Country Status (15)

Country Link
US (1) US5977372A (de)
EP (1) EP0846117B1 (de)
JP (1) JPH11507625A (de)
CN (1) CN1073110C (de)
AT (1) ATE240325T1 (de)
AU (1) AU718553B2 (de)
BR (1) BR9609403A (de)
CA (1) CA2223783A1 (de)
CZ (1) CZ390097A3 (de)
DE (1) DE69628175D1 (de)
EA (1) EA000622B1 (de)
HU (1) HUP9900871A3 (de)
IL (1) IL122220A (de)
NZ (1) NZ310164A (de)
WO (1) WO1996040684A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1291356B1 (it) * 1997-05-13 1999-01-07 Zambon Spa Processo per la rimozione di metalli pesanti
IT1292437B1 (it) * 1997-06-30 1999-02-08 Zambon Spa Processo di orto-metallazione utile per la sintesi di 1 - tetrazol- 5-il) benzeni 2-sostituiti
JP4524072B2 (ja) 2000-10-23 2010-08-11 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー 新規化合物
GB0222056D0 (en) * 2002-09-23 2002-10-30 Novartis Ag Process for the manufacture of organic compounds
DE102004060699A1 (de) * 2004-12-16 2006-06-22 Ratiopharm Gmbh Verfahren zur Herstellung von Candesartan
AR053346A1 (es) * 2005-03-25 2007-05-02 Glaxo Group Ltd Compuesto derivado de 8h -pirido (2,3-d) pirimidin -7 ona 2,4,8- trisustituida composicion farmaceutica y uso para preparar una composicion para tratamiento y profilxis de una enfermedad mediada por la quinasa csbp/ rk/p38
WO2008134890A1 (en) * 2007-05-07 2008-11-13 Valorisation-Recherche, Societe En Commandite Methods for preparing diorganozinc compounds
JP2022550451A (ja) * 2019-10-02 2022-12-01 ブループリント メディシンズ コーポレイション アクチビン受容体様キナーゼ阻害剤を調製するためのプロセス

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5039814A (en) * 1990-05-02 1991-08-13 Merck & Co., Inc. Ortho-lithiation process for the synthesis of 2-substituted 1-(tetrazol-5-yl)benzenes
US5290780A (en) * 1991-01-30 1994-03-01 American Cyanamid Co. Angiotensin II receptor blocking 2,3,6 substituted quinazolinones
US5149699A (en) * 1991-10-24 1992-09-22 American Home Products Corporation Substituted pyridopyrimidines useful as antgiotensin II antagonists
EP0550313A1 (de) * 1991-12-30 1993-07-07 Synthelabo 2-(Tetranol-5-yl)-(1,1'-Biphenyl)derivate, ihre Herstellung und Anwendung als Zwischenverbindungen
US5466692A (en) * 1993-03-24 1995-11-14 American Home Products Corporation Substituted pyridopyrimidines and antihypertensives

Also Published As

Publication number Publication date
JPH11507625A (ja) 1999-07-06
CN1073110C (zh) 2001-10-17
HUP9900871A2 (hu) 1999-07-28
HUP9900871A3 (en) 2000-07-28
IL122220A0 (en) 1996-06-06
US5977372A (en) 1999-11-02
EP0846117B1 (de) 2003-05-14
EA199800035A1 (ru) 1998-08-27
CA2223783A1 (en) 1996-12-19
IL122220A (en) 2001-08-08
EP0846117A1 (de) 1998-06-10
AU718553B2 (en) 2000-04-13
NZ310164A (en) 2000-01-28
BR9609403A (pt) 1999-05-11
EA000622B1 (ru) 1999-12-29
DE69628175D1 (de) 2003-06-18
CZ390097A3 (cs) 1998-06-17
AU6090296A (en) 1996-12-30
WO1996040684A1 (en) 1996-12-19
CN1192214A (zh) 1998-09-02

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