JP2008044952A5 - - Google Patents
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- Publication number
- JP2008044952A5 JP2008044952A5 JP2007241012A JP2007241012A JP2008044952A5 JP 2008044952 A5 JP2008044952 A5 JP 2008044952A5 JP 2007241012 A JP2007241012 A JP 2007241012A JP 2007241012 A JP2007241012 A JP 2007241012A JP 2008044952 A5 JP2008044952 A5 JP 2008044952A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- mono
- substituted
- halogen atom
- lower alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 125000003545 alkoxy group Chemical group 0.000 claims 6
- 125000000217 alkyl group Chemical group 0.000 claims 6
- 125000003277 amino group Chemical group 0.000 claims 4
- 125000005843 halogen group Chemical group 0.000 claims 4
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 4
- 125000004453 alkoxycarbonyl group Chemical group 0.000 claims 3
- 125000004390 alkyl sulfonyl group Chemical group 0.000 claims 3
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 claims 3
- 125000005236 alkanoylamino group Chemical group 0.000 claims 2
- 125000005153 alkyl sulfamoyl group Chemical group 0.000 claims 2
- 125000004644 alkyl sulfinyl group Chemical group 0.000 claims 2
- 125000004414 alkyl thio group Chemical group 0.000 claims 2
- 125000004397 aminosulfonyl group Chemical group NS(=O)(=O)* 0.000 claims 2
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 2
- 125000004093 cyano group Chemical group *C#N 0.000 claims 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 2
- 150000003839 salts Chemical class 0.000 claims 2
- 125000003282 alkyl amino group Chemical group 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- 125000002057 carboxymethyl group Chemical group [H]OC(=O)C([H])([H])[*] 0.000 claims 1
- 125000002485 formyl group Chemical group [H]C(*)=O 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- -1 nitrogen-containing 5-membered heterocyclic compound Chemical class 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 229910052717 sulfur Inorganic materials 0.000 claims 1
- 125000001544 thienyl group Chemical group 0.000 claims 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2007241012A JP2008044952A (ja) | 2001-04-16 | 2007-09-18 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2001116436 | 2001-04-16 | ||
| JP2001249671 | 2001-08-20 | ||
| JP2007241012A JP2008044952A (ja) | 2001-04-16 | 2007-09-18 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002580915A Division JP4073786B2 (ja) | 2001-04-16 | 2002-04-15 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008044952A JP2008044952A (ja) | 2008-02-28 |
| JP2008044952A5 true JP2008044952A5 (enExample) | 2008-06-26 |
Family
ID=26613619
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002580915A Expired - Fee Related JP4073786B2 (ja) | 2001-04-16 | 2002-04-15 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
| JP2007241012A Pending JP2008044952A (ja) | 2001-04-16 | 2007-09-18 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002580915A Expired - Fee Related JP4073786B2 (ja) | 2001-04-16 | 2002-04-15 | 高コンダクタンス型カルシウム感受性ｋチャネル開口薬 |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US7759373B2 (enExample) |
| EP (1) | EP1432690A2 (enExample) |
| JP (2) | JP4073786B2 (enExample) |
| KR (1) | KR100863659B1 (enExample) |
| CN (2) | CN100540538C (enExample) |
| AR (1) | AR035828A1 (enExample) |
| AU (1) | AU2002246397B2 (enExample) |
| BR (1) | BR0208956A (enExample) |
| CA (1) | CA2444596A1 (enExample) |
| CZ (1) | CZ20032829A3 (enExample) |
| HU (1) | HUP0303829A3 (enExample) |
| IL (1) | IL158168A0 (enExample) |
| MX (1) | MXPA03009440A (enExample) |
| NZ (1) | NZ529043A (enExample) |
| PL (1) | PL367325A1 (enExample) |
| TW (2) | TWI322686B (enExample) |
| WO (1) | WO2002083111A2 (enExample) |
Families Citing this family (94)
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| EP1554269A1 (en) * | 2002-07-09 | 2005-07-20 | Vertex Pharmaceuticals Incorporated | Imidazoles, oxazoles and thiazoles with protein kinase inhibiting activities |
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| DK2010528T3 (en) | 2006-04-19 | 2018-01-15 | Novartis Ag | 6-O-Substituted Benzoxazole and Benzothiazole Compounds and Methods for Inhibiting CSF-1R Signaling |
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| JPS5936614A (ja) * | 1982-08-25 | 1984-02-28 | Tanabe Seiyaku Co Ltd | 抗脂血剤 |
| JPS59152382A (ja) * | 1983-02-18 | 1984-08-31 | Tanabe Seiyaku Co Ltd | フリルオキサゾリル酢酸誘導体 |
| JPS59172488A (ja) * | 1983-03-18 | 1984-09-29 | Tanabe Seiyaku Co Ltd | 抗脂血剤 |
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| JPS60202820A (ja) * | 1984-03-27 | 1985-10-14 | Tanabe Seiyaku Co Ltd | 抗脂血剤 |
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| US5340826A (en) * | 1993-02-04 | 1994-08-23 | Pfizer Inc. | Pharmaceutical agents for treatment of urinary incontinence |
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| EP0891340B1 (en) * | 1996-04-03 | 2002-11-13 | Takeda Chemical Industries, Ltd. | Oxazole derivatives, their production and use |
| TW467902B (en) | 1996-07-31 | 2001-12-11 | Bristol Myers Squibb Co | Diphenyl heterocycles as potassium channel modulators |
| US6121260A (en) | 1997-07-03 | 2000-09-19 | Neurogen Corporation | Method of treating conditions susceptible to modulation of NPY receptors with diarylimidazole derivatives |
| GB9726989D0 (en) | 1997-12-22 | 1998-02-18 | Ciba Geigy Ag | Organic compounds |
| AU735704B2 (en) | 1998-01-29 | 2001-07-12 | Bristol-Myers Squibb Company | Derivatives of 1,3,4-oxadiazolone |
| CZ296507B6 (cs) | 1998-03-30 | 2006-03-15 | Japan Tobacco Inc. | Zpusob výroby oxazolylethanolových derivátu |
-
2002
- 2002-04-15 CN CNB028083709A patent/CN100540538C/zh not_active Expired - Fee Related
- 2002-04-15 CA CA002444596A patent/CA2444596A1/en not_active Abandoned
- 2002-04-15 EP EP02714577A patent/EP1432690A2/en not_active Withdrawn
- 2002-04-15 WO PCT/JP2002/003723 patent/WO2002083111A2/en not_active Ceased
- 2002-04-15 BR BR0208956-4A patent/BR0208956A/pt not_active IP Right Cessation
- 2002-04-15 CZ CZ20032829A patent/CZ20032829A3/cs unknown
- 2002-04-15 IL IL15816802A patent/IL158168A0/xx unknown
- 2002-04-15 HU HU0303829A patent/HUP0303829A3/hu unknown
- 2002-04-15 JP JP2002580915A patent/JP4073786B2/ja not_active Expired - Fee Related
- 2002-04-15 NZ NZ529043A patent/NZ529043A/en unknown
- 2002-04-15 KR KR1020037013493A patent/KR100863659B1/ko not_active Expired - Fee Related
- 2002-04-15 AU AU2002246397A patent/AU2002246397B2/en not_active Ceased
- 2002-04-15 PL PL02367325A patent/PL367325A1/xx unknown
- 2002-04-15 CN CNA200910004656XA patent/CN101519386A/zh active Pending
- 2002-04-15 US US10/474,850 patent/US7759373B2/en not_active Expired - Fee Related
- 2002-04-16 TW TW091107687A patent/TWI322686B/zh not_active IP Right Cessation
- 2002-04-16 TW TW098138199A patent/TW201006831A/zh unknown
- 2002-04-16 AR ARP020101381A patent/AR035828A1/es unknown
-
2003
- 2003-10-15 MX MXPA03009440A patent/MXPA03009440A/es active IP Right Grant
-
2007
- 2007-09-18 JP JP2007241012A patent/JP2008044952A/ja active Pending
-
2010
- 2010-06-07 US US12/795,323 patent/US20100256165A1/en not_active Abandoned
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