JP2008019261A5 - - Google Patents
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- JP2008019261A5 JP2008019261A5 JP2007201372A JP2007201372A JP2008019261A5 JP 2008019261 A5 JP2008019261 A5 JP 2008019261A5 JP 2007201372 A JP2007201372 A JP 2007201372A JP 2007201372 A JP2007201372 A JP 2007201372A JP 2008019261 A5 JP2008019261 A5 JP 2008019261A5
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- JP
- Japan
- Prior art keywords
- group
- independently
- substituted
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- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51956603P | 2003-11-12 | 2003-11-12 | |
| US55701104P | 2004-03-25 | 2004-03-25 | |
| US59297204P | 2004-07-30 | 2004-07-30 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006539906A Division JP5435841B2 (ja) | 2003-11-12 | 2004-11-12 | 複素環式ボロン酸化合物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2008019261A JP2008019261A (ja) | 2008-01-31 |
| JP2008019261A5 true JP2008019261A5 (https=) | 2008-09-18 |
Family
ID=34595944
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006539906A Expired - Fee Related JP5435841B2 (ja) | 2003-11-12 | 2004-11-12 | 複素環式ボロン酸化合物 |
| JP2007201372A Withdrawn JP2008019261A (ja) | 2003-11-12 | 2007-08-01 | 複素環式ボロン酸化合物 |
| JP2008220344A Expired - Fee Related JP5398199B2 (ja) | 2003-11-12 | 2008-08-28 | 複素環式ボロン酸化合物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006539906A Expired - Fee Related JP5435841B2 (ja) | 2003-11-12 | 2004-11-12 | 複素環式ボロン酸化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008220344A Expired - Fee Related JP5398199B2 (ja) | 2003-11-12 | 2008-08-28 | 複素環式ボロン酸化合物 |
Country Status (21)
| Country | Link |
|---|---|
| US (3) | US7674913B2 (https=) |
| EP (3) | EP1743676A1 (https=) |
| JP (3) | JP5435841B2 (https=) |
| KR (2) | KR100918322B1 (https=) |
| AR (1) | AR046778A1 (https=) |
| AU (1) | AU2004288831B2 (https=) |
| BR (1) | BRPI0416444B8 (https=) |
| CA (1) | CA2545311C (https=) |
| DK (1) | DK1689757T3 (https=) |
| EA (1) | EA013684B1 (https=) |
| ES (1) | ES2524916T3 (https=) |
| HR (1) | HRP20141155T1 (https=) |
| IL (1) | IL175550A (https=) |
| NO (2) | NO337818B1 (https=) |
| NZ (1) | NZ547752A (https=) |
| PL (1) | PL1689757T3 (https=) |
| PT (1) | PT1689757E (https=) |
| SG (1) | SG134333A1 (https=) |
| SI (1) | SI1689757T1 (https=) |
| TW (1) | TWI337078B (https=) |
| WO (1) | WO2005047297A1 (https=) |
Families Citing this family (79)
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| AR045047A1 (es) | 2003-07-11 | 2005-10-12 | Arena Pharm Inc | Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos |
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| AU2007235876A1 (en) | 2006-04-12 | 2007-10-18 | Probiodrug Ag | Enzyme inhibitors |
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| TWI430806B (zh) * | 2006-09-13 | 2014-03-21 | Smithkline Beecham Corp | 用於投與長效降血糖藥劑之方法 |
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| EP2089383B1 (en) | 2006-11-09 | 2015-09-16 | Probiodrug AG | 3-hydr0xy-1,5-dihydr0-pyrr0l-2-one derivatives as inhibitors of glutaminyl cyclase for the treatment of ulcer, cancer and other diseases |
| US9126987B2 (en) | 2006-11-30 | 2015-09-08 | Probiodrug Ag | Inhibitors of glutaminyl cyclase |
| US20160331729A9 (en) | 2007-04-11 | 2016-11-17 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| US11241420B2 (en) | 2007-04-11 | 2022-02-08 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| EP3788877B1 (en) * | 2007-04-11 | 2024-08-07 | Omeros Corporation | Compositions and methods for prophylaxis and treatment of addictions |
| JP5667440B2 (ja) | 2007-04-18 | 2015-02-12 | プロビオドルグ エージー | グルタミニルシクラーゼ阻害剤としてのチオ尿素誘導体 |
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| UY32030A (es) | 2008-08-06 | 2010-03-26 | Boehringer Ingelheim Int | "tratamiento para diabetes en pacientes inapropiados para terapia con metformina" |
| UA119131C2 (uk) | 2008-08-15 | 2019-05-10 | Бьорінгер Інгельхайм Інтернаціональ Гмбх | Похідні пурину для застосування при лікуванні пов'язаних із fab захворювань |
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| KR20240090632A (ko) | 2009-11-27 | 2024-06-21 | 베링거 인겔하임 인터내셔날 게엠베하 | 리나글립틴과 같은 ｄｐｐ－ｉｖ 억제제를 사용한 유전자형 검사된 당뇨병 환자의 치료 |
| WO2011107530A2 (en) | 2010-03-03 | 2011-09-09 | Probiodrug Ag | Novel inhibitors |
| JP5688745B2 (ja) | 2010-03-10 | 2015-03-25 | プロビオドルグ エージー | グルタミニルシクラーゼ（ｑｃ、ｅｃ２．３．２．５）の複素環阻害剤 |
| CN102286011B (zh) * | 2010-03-16 | 2017-10-03 | 美德（江西）生物科技有限公司 | 吡咯烷硼酸酯二肽基肽酶抑制剂及其药物组合物 |
| JP2013522279A (ja) | 2010-03-18 | 2013-06-13 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 糖尿病及び関連状態の治療で用いるｇｐｒ１１９作動薬とｄｄｐ−ｉｖ阻害薬リナグリプチンの組合せ |
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| CA3070513C (en) | 2010-05-05 | 2023-01-03 | Boehringer Ingelheim International Gmbh | A dpp-4 inhibitor for use in treatment of skin-alterations or necrosis |
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| MX386419B (es) | 2015-01-06 | 2025-03-18 | Arena Pharm Inc | Metodos de condiciones de tratamiento relacionadas con el receptor s1p1. |
| EA201791982A1 (ru) | 2015-03-09 | 2020-02-17 | Интекрин Терапьютикс, Инк. | Способы лечения неалкогольной жировой болезни печени и/или липодистрофии |
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- 2004-11-12 SG SG200705459-6A patent/SG134333A1/en unknown
- 2004-11-12 EP EP06015708A patent/EP1743676A1/en not_active Withdrawn
- 2004-11-12 US US10/514,575 patent/US7674913B2/en active Active - Reinstated
- 2004-11-12 PT PT48108393T patent/PT1689757E/pt unknown
- 2004-11-12 CA CA2545311A patent/CA2545311C/en not_active Expired - Lifetime
- 2004-11-12 PL PL04810839T patent/PL1689757T3/pl unknown
- 2004-11-12 EP EP08013650.0A patent/EP1997533B8/en not_active Expired - Lifetime
- 2004-11-12 EP EP04810839.3A patent/EP1689757B1/en not_active Expired - Lifetime
- 2004-11-12 HR HRP20141155TT patent/HRP20141155T1/hr unknown
- 2004-11-12 WO PCT/US2004/037820 patent/WO2005047297A1/en not_active Ceased
- 2004-11-12 AU AU2004288831A patent/AU2004288831B2/en not_active Ceased
- 2004-11-12 DK DK04810839.3T patent/DK1689757T3/en active
- 2004-11-12 JP JP2006539906A patent/JP5435841B2/ja not_active Expired - Fee Related
- 2004-11-12 AR ARP040104198A patent/AR046778A1/es active IP Right Grant
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- 2004-11-12 TW TW093134766A patent/TWI337078B/zh not_active IP Right Cessation
- 2004-11-12 SI SI200432201T patent/SI1689757T1/sl unknown
- 2004-11-12 EA EA200600935A patent/EA013684B1/ru not_active IP Right Cessation
- 2004-11-12 KR KR1020067011419A patent/KR100918322B1/ko not_active Expired - Fee Related
- 2004-11-12 BR BRPI0416444A patent/BRPI0416444B8/pt not_active IP Right Cessation
- 2004-11-12 KR KR1020077011094A patent/KR20070054762A/ko not_active Withdrawn
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