JP2005511727A5 - - Google Patents
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- Publication number
- JP2005511727A5 JP2005511727A5 JP2003551090A JP2003551090A JP2005511727A5 JP 2005511727 A5 JP2005511727 A5 JP 2005511727A5 JP 2003551090 A JP2003551090 A JP 2003551090A JP 2003551090 A JP2003551090 A JP 2003551090A JP 2005511727 A5 JP2005511727 A5 JP 2005511727A5
- Authority
- JP
- Japan
- Prior art keywords
- substituted
- alkyl
- sulfonyl
- amino acid
- phenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/014,304 US6610734B2 (en) | 2000-12-13 | 2001-12-11 | Heterocyclic sulfonamide inhibitors of beta amyloid production |
| US10/166,896 US6657070B2 (en) | 2000-12-13 | 2002-06-11 | Production of chirally pure α-amino acids and N-sulfonyl α-amino acids |
| PCT/US2002/038117 WO2003050062A2 (en) | 2001-12-11 | 2002-11-26 | PRODUCTION OF CHIRALLY PURE α-AMINO ACIDS ADN N-SULFONYL α-AMINO ACIDS |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005511727A JP2005511727A (ja) | 2005-04-28 |
| JP2005511727A5 true JP2005511727A5 (https=) | 2006-01-05 |
| JP4615861B2 JP4615861B2 (ja) | 2011-01-19 |
Family
ID=46204648
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003551090A Expired - Fee Related JP4615861B2 (ja) | 2001-12-11 | 2002-11-26 | キラル的に純粋なα−アミノ酸およびＮ−スルホニルα−アミノ酸の生産 |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1461332A4 (https=) |
| JP (1) | JP4615861B2 (https=) |
| AU (2) | AU2002351170B8 (https=) |
| CA (1) | CA2470111A1 (https=) |
| MX (1) | MXPA04005366A (https=) |
| TW (1) | TWI260316B (https=) |
| WO (1) | WO2003050062A2 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0303857A3 (en) | 2000-12-13 | 2007-07-30 | Wyeth Corp | Heterocyclic sulifonamide inhibitors of beta amyloid production |
| BRPI0408962A (pt) | 2003-03-31 | 2006-04-04 | Wyeth Corp | inibidores sulfonamidas heterocìclicos contendo flúor- e trifluoroalquila da produção de beta amilóide e seus derivados |
| ES2330451T3 (es) | 2004-01-16 | 2009-12-10 | Wyeth | Inhibidores a base de sulfonamidas heterociclicas de la produccion de beta-amiloides que contienen un azol. |
| JP2009534385A (ja) | 2006-04-21 | 2009-09-24 | ワイス | キラル的に純粋なアミノアルコール中間体、それらの誘導体の製造、及びそれらの使用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3802981A1 (de) * | 1988-02-02 | 1989-08-10 | Basf Ag | Verfahren zur reduktion reduzierbarer verbindungen |
| US5264577A (en) * | 1992-04-22 | 1993-11-23 | Warner-Lambert Company | Cyclic amino acids and derivatives thereof |
| ATE218541T1 (de) * | 1992-08-25 | 2002-06-15 | Searle & Co | Hydroxyethylaminosulfonamide verwendbar als inhibitoren retroviraler proteasen |
| US5968942A (en) * | 1992-08-25 | 1999-10-19 | G. D. Searle & Co. | α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors |
| US6191306B1 (en) * | 1999-08-03 | 2001-02-20 | Eastman Chemical Company | Process for the preparation of cyclopropylglycine |
-
2002
- 2002-11-26 JP JP2003551090A patent/JP4615861B2/ja not_active Expired - Fee Related
- 2002-11-26 WO PCT/US2002/038117 patent/WO2003050062A2/en not_active Ceased
- 2002-11-26 CA CA002470111A patent/CA2470111A1/en not_active Abandoned
- 2002-11-26 MX MXPA04005366A patent/MXPA04005366A/es active IP Right Grant
- 2002-11-26 AU AU2002351170A patent/AU2002351170B8/en not_active Ceased
- 2002-11-26 EP EP02786817A patent/EP1461332A4/en not_active Withdrawn
- 2002-12-10 TW TW091135621A patent/TWI260316B/zh active
-
2009
- 2009-12-24 AU AU2009251195A patent/AU2009251195A1/en not_active Abandoned
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