JO3773B1 - معدلات p2x7 - Google Patents

معدلات p2x7

Info

Publication number
JO3773B1
JO3773B1 JOP/2014/0094A JOP20140094A JO3773B1 JO 3773 B1 JO3773 B1 JO 3773B1 JO P20140094 A JOP20140094 A JO P20140094A JO 3773 B1 JO3773 B1 JO 3773B1
Authority
JO
Jordan
Prior art keywords
iib
iia
formulas
compounds
rates
Prior art date
Application number
JOP/2014/0094A
Other languages
English (en)
Inventor
Soyode-Johnson Akinola
R Coate Heather
C Rech Jason
A Letavic Michael
C Chrovian Christa
L Wall Jessica
F Gelin Christine
Stenne Brice
De Angelisz Meri
D Allison Brett
S Mani Neelakandha
Jesus Alcazar Vaca Manuel
Ignacio Andres Gil Jose
M Swanson Devin
A Dvorak Curt
Deng Xiaohu
M Savall Brad
T Liang Jimmy
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of JO3773B1 publication Critical patent/JO3773B1/ar

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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Abstract

يتعلق هذا الاختراع بمركبات الصيغة (I، Ia، IIa و IIb): يتعلق الاختراع أيضاً بتركيبات صيدلية تشتمل على مركبات الصيغة (I، Ia، IIa و IIb). وتكون طرق عمل واستخدام مركبات الصيغة (I، Ia، IIa و IIb) أيضاً داخل مجال الاختراع.
JOP/2014/0094A 2013-03-14 2014-03-12 معدلات p2x7 JO3773B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361786260P 2013-03-14 2013-03-14

Publications (1)

Publication Number Publication Date
JO3773B1 true JO3773B1 (ar) 2021-01-31

Family

ID=50543353

Family Applications (1)

Application Number Title Priority Date Filing Date
JOP/2014/0094A JO3773B1 (ar) 2013-03-14 2014-03-12 معدلات p2x7

Country Status (33)

Country Link
US (8) US10112937B2 (ar)
EP (3) EP2970267B3 (ar)
JP (1) JP6293861B2 (ar)
KR (5) KR102516711B1 (ar)
CN (2) CN110003200B (ar)
AR (2) AR095530A1 (ar)
AU (5) AU2014239291B2 (ar)
BR (1) BR112015023142B1 (ar)
CA (1) CA2906085C (ar)
CL (3) CL2015002655A1 (ar)
CY (1) CY1119110T1 (ar)
DK (2) DK2970267T6 (ar)
EA (1) EA028816B1 (ar)
ES (2) ES2704024T3 (ar)
HR (1) HRP20171168T4 (ar)
HU (1) HUE032877T2 (ar)
IL (1) IL240880B (ar)
JO (1) JO3773B1 (ar)
LT (1) LT2970267T (ar)
ME (1) ME02802B (ar)
MX (2) MX364796B (ar)
PH (1) PH12015501930A1 (ar)
PL (1) PL2970267T6 (ar)
PT (2) PT3239151T (ar)
RS (1) RS56315B2 (ar)
SG (2) SG10201700889PA (ar)
SI (1) SI2970267T1 (ar)
SM (1) SMT201700352T1 (ar)
TW (2) TWI644671B (ar)
UA (1) UA116467C2 (ar)
UY (3) UY39887A (ar)
WO (1) WO2014152604A1 (ar)
ZA (1) ZA201507627B (ar)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI627174B (zh) 2013-03-14 2018-06-21 比利時商健生藥品公司 Ｐ２ｘ７調控劑
EP2970304B1 (en) 2013-03-14 2018-08-15 Janssen Pharmaceutica NV P2x7 modulators
JO3773B1 (ar) 2013-03-14 2021-01-31 Janssen Pharmaceutica Nv معدلات p2x7
EP3112366B1 (en) 2013-03-14 2018-02-28 Janssen Pharmaceutica NV P2x7 modulators
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