HRP20171168T4 - Modulatori p2x7 - Google Patents
Modulatori p2x7Info
- Publication number
- HRP20171168T4 HRP20171168T4 HRP20171168TT HRP20171168T HRP20171168T4 HR P20171168 T4 HRP20171168 T4 HR P20171168T4 HR P20171168T T HRP20171168T T HR P20171168TT HR P20171168 T HRP20171168 T HR P20171168T HR P20171168 T4 HRP20171168 T4 HR P20171168T4
- Authority
- HR
- Croatia
- Prior art keywords
- modulators
- Prior art date
Links
- 101100135293 Mus musculus P2rx7 gene Proteins 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- C—CHEMISTRY; METALLURGY
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- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
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- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Hematology (AREA)
- Vascular Medicine (AREA)
- Obesity (AREA)
- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Psychology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361786260P | 2013-03-14 | 2013-03-14 | |
PCT/US2014/027522 WO2014152604A1 (en) | 2013-03-14 | 2014-03-14 | P2x7 modulators |
EP14718857.7A EP2970267B3 (en) | 2013-03-14 | 2014-03-14 | P2x7 modulators |
Publications (2)
Publication Number | Publication Date |
---|---|
HRP20171168T1 HRP20171168T1 (hr) | 2017-10-06 |
HRP20171168T4 true HRP20171168T4 (hr) | 2018-09-21 |
Family
ID=50543353
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HRP20171168TT HRP20171168T4 (hr) | 2013-03-14 | 2017-07-31 | Modulatori p2x7 |
Country Status (33)
Country | Link |
---|---|
US (8) | US10112937B2 (hr) |
EP (3) | EP3495365A1 (hr) |
JP (1) | JP6293861B2 (hr) |
KR (4) | KR102516711B1 (hr) |
CN (2) | CN110003200B (hr) |
AR (2) | AR095530A1 (hr) |
AU (5) | AU2014239291B2 (hr) |
BR (1) | BR112015023142B1 (hr) |
CA (1) | CA2906085C (hr) |
CL (3) | CL2015002655A1 (hr) |
CY (1) | CY1119110T1 (hr) |
DK (2) | DK2970267T6 (hr) |
EA (1) | EA028816B1 (hr) |
ES (2) | ES2704024T3 (hr) |
HK (1) | HK1218541A1 (hr) |
HR (1) | HRP20171168T4 (hr) |
HU (1) | HUE032877T2 (hr) |
IL (1) | IL240880B (hr) |
JO (1) | JO3773B1 (hr) |
LT (1) | LT2970267T (hr) |
ME (1) | ME02802B (hr) |
MX (2) | MX364796B (hr) |
PH (1) | PH12015501930A1 (hr) |
PL (1) | PL2970267T6 (hr) |
PT (2) | PT3239151T (hr) |
RS (1) | RS56315B2 (hr) |
SG (2) | SG10201700889PA (hr) |
SI (1) | SI2970267T1 (hr) |
TW (2) | TWI599567B (hr) |
UA (1) | UA116467C2 (hr) |
UY (3) | UY35469A (hr) |
WO (1) | WO2014152604A1 (hr) |
ZA (1) | ZA201507627B (hr) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2654288T3 (es) | 2013-03-14 | 2018-02-13 | Janssen Pharmaceutica, N.V. | Moduladores de P2X7 |
ES2689526T3 (es) | 2013-03-14 | 2018-11-14 | Janssen Pharmaceutica Nv | Moduladores de P2X7 |
EP2970283B1 (en) | 2013-03-14 | 2020-11-11 | Boehringer Ingelheim International GmbH | Substituted 2-aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of cathepsin c |
TWI627174B (zh) | 2013-03-14 | 2018-06-21 | 比利時商健生藥品公司 | P2x7調控劑 |
TWI599567B (zh) | 2013-03-14 | 2017-09-21 | 健生藥品公司 | P2x7調節劑 |
GB201321748D0 (en) * | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
WO2015172196A1 (en) * | 2014-05-13 | 2015-11-19 | Monash University | Heterocyclic compounds and use of same |
LT3191487T (lt) | 2014-09-12 | 2019-10-10 | Boehringer Ingelheim International Gmbh | Katepsino c spirocikliniai inhibitoriai |
AU2015315687B2 (en) | 2014-09-12 | 2019-07-11 | Janssen Pharmaceutica Nv | P2X7 modulators |
CN107709299B (zh) | 2015-04-24 | 2021-07-16 | 盐野义制药株式会社 | 6元杂环衍生物及含有其的药物组合物 |
EP3328857B1 (en) * | 2015-07-31 | 2019-08-14 | Merck Patent GmbH | Bicyclic heterocyclic derivatives |
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