IL208838A0 - Purine pi3k inhibitor compounds and methods of use - Google Patents

Purine pi3k inhibitor compounds and methods of use

Info

Publication number
IL208838A0
IL208838A0 IL208838A IL20883810A IL208838A0 IL 208838 A0 IL208838 A0 IL 208838A0 IL 208838 A IL208838 A IL 208838A IL 20883810 A IL20883810 A IL 20883810A IL 208838 A0 IL208838 A0 IL 208838A0
Authority
IL
Israel
Prior art keywords
purine
methods
inhibitor compounds
pi3k inhibitor
pi3k
Prior art date
Application number
IL208838A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche, Genentech Inc filed Critical Hoffmann La Roche
Publication of IL208838A0 publication Critical patent/IL208838A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL208838A 2008-05-30 2010-10-20 Purine pi3k inhibitor compounds and methods of use IL208838A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5755908P 2008-05-30 2008-05-30
PCT/US2009/045603 WO2009146406A1 (en) 2008-05-30 2009-05-29 Purine pi3k inhibitor compounds and methods of use

Publications (1)

Publication Number Publication Date
IL208838A0 true IL208838A0 (en) 2011-01-31

Family

ID=41017038

Family Applications (1)

Application Number Title Priority Date Filing Date
IL208838A IL208838A0 (en) 2008-05-30 2010-10-20 Purine pi3k inhibitor compounds and methods of use

Country Status (14)

Country Link
US (2) US8158624B2 (enExample)
EP (1) EP2279188B1 (enExample)
JP (1) JP2011521968A (enExample)
KR (1) KR20110042153A (enExample)
CN (1) CN102105474B (enExample)
AU (1) AU2009251291B2 (enExample)
BR (1) BRPI0909614A2 (enExample)
CA (1) CA2721851A1 (enExample)
ES (1) ES2533788T3 (enExample)
IL (1) IL208838A0 (enExample)
MX (1) MX2010012583A (enExample)
RU (1) RU2509081C2 (enExample)
WO (1) WO2009146406A1 (enExample)
ZA (1) ZA201007524B (enExample)

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TW201817731A (zh) * 2016-09-29 2018-05-16 日商第一三共股份有限公司 ［２－（１－甲基－１ｈ－吡唑－４－基）－６－（ 啉－４－基）－９ｈ－嘌呤－８－基］［４－（ 啉－４－基）哌啶－１－基］甲酮及其製藥上容許鹽之結晶
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Also Published As

Publication number Publication date
ZA201007524B (en) 2012-01-25
ES2533788T3 (es) 2015-04-14
US20090318411A1 (en) 2009-12-24
RU2509081C2 (ru) 2014-03-10
CN102105474B (zh) 2014-01-08
BRPI0909614A2 (pt) 2015-09-22
CA2721851A1 (en) 2009-12-03
EP2279188B1 (en) 2015-01-28
US20120135988A1 (en) 2012-05-31
WO2009146406A1 (en) 2009-12-03
AU2009251291A1 (en) 2009-12-03
EP2279188A1 (en) 2011-02-02
AU2009251291B2 (en) 2013-05-02
US8445487B2 (en) 2013-05-21
MX2010012583A (es) 2011-02-24
US8158624B2 (en) 2012-04-17
CN102105474A (zh) 2011-06-22
JP2011521968A (ja) 2011-07-28
KR20110042153A (ko) 2011-04-25
RU2010154428A (ru) 2012-07-10

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