IL145986A0 - Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a - Google Patents

Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a

Info

Publication number
IL145986A0
IL145986A0 IL14598600A IL14598600A IL145986A0 IL 145986 A0 IL145986 A0 IL 145986A0 IL 14598600 A IL14598600 A IL 14598600A IL 14598600 A IL14598600 A IL 14598600A IL 145986 A0 IL145986 A0 IL 145986A0
Authority
IL
Israel
Prior art keywords
meaning
halo
deoxo
aza
homerythromycin
Prior art date
Application number
IL14598600A
Other languages
English (en)
Original Assignee
Pliva Farmaceutska Ind Dionic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Farmaceutska Ind Dionic filed Critical Pliva Farmaceutska Ind Dionic
Publication of IL145986A0 publication Critical patent/IL145986A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL14598600A 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a IL145986A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HR990130A HRP990130B1 (en) 1999-05-03 1999-05-03 HALOGEN DERIVATIVES 9a-N-(N'-ARYLCARBAMOYL)- AND 9a-N-(N'-ARYLTHIOCARBAMOYL)-9-DEOXO-9a-AZA-9a OF HOMOERYTHROMYCIN A
PCT/HR2000/000013 WO2000066603A1 (en) 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a

Publications (1)

Publication Number Publication Date
IL145986A0 true IL145986A0 (en) 2002-07-25

Family

ID=10946916

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14598600A IL145986A0 (en) 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a
IL145986A IL145986A (en) 1999-05-03 2001-10-17 History of a9 - deoxo - 9a - aza 9a - (Aril (Thio) Karbmobil) - 9a - Humarithromycin A Preparation, and pharmaceutical preparations containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL145986A IL145986A (en) 1999-05-03 2001-10-17 History of a9 - deoxo - 9a - aza 9a - (Aril (Thio) Karbmobil) - 9a - Humarithromycin A Preparation, and pharmaceutical preparations containing them

Country Status (33)

Country Link
US (1) US6872707B1 (ja)
EP (1) EP1175429B1 (ja)
JP (1) JP2002543213A (ja)
KR (1) KR100714740B1 (ja)
CN (1) CN1140535C (ja)
AT (1) ATE244258T1 (ja)
AU (1) AU767681B2 (ja)
BG (1) BG106173A (ja)
BR (1) BR0010231A (ja)
CA (1) CA2372977A1 (ja)
CZ (1) CZ20013913A3 (ja)
DE (1) DE60003671T2 (ja)
DK (1) DK1175429T3 (ja)
EA (1) EA005214B1 (ja)
EE (1) EE05007B1 (ja)
ES (1) ES2202107T3 (ja)
GE (1) GEP20032928B (ja)
HK (1) HK1045522B (ja)
HR (1) HRP990130B1 (ja)
HU (1) HUP0201146A3 (ja)
IL (2) IL145986A0 (ja)
IS (1) IS6115A (ja)
MX (1) MXPA01011038A (ja)
NO (1) NO320138B1 (ja)
NZ (1) NZ515278A (ja)
PL (1) PL351402A1 (ja)
PT (1) PT1175429E (ja)
SI (1) SI1175429T1 (ja)
SK (1) SK284513B6 (ja)
TR (1) TR200103143T2 (ja)
UA (1) UA71962C2 (ja)
WO (1) WO2000066603A1 (ja)
ZA (1) ZA200108484B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010146B1 (en) * 2001-02-28 2005-10-31 Pliva D.D. 9a-N-(N'-(PHENYLSULFONYL)CARBAMOYL) DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMYCIN A AND OF 5-O-DESOSAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHRONOLIDE A
HRP20020886A2 (en) * 2002-11-11 2005-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. SUBSTITUTED 9a-N-[N'-(BENZENSULFONYL)CARBAMOYL-γ-AMINOPROPYL) AND 9a-N(N' -(?-CYANOETHIL)-N' -(b
HRP20020885B1 (en) * 2002-11-11 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A
HRP20020991A2 (en) * 2002-12-12 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de
HRP20030381B1 (en) * 2003-05-14 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. 3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
JP2008526948A (ja) * 2005-01-14 2008-07-24 グラクソスミスクライン・イストラジヴァッキ・センタル・ザグレブ・ドルズバ・ゼー・オメイェノ・オドゴヴォルノスティオ 抗マラリア活性を有する9a−カルバモイルおよびチオカルバモイルアザライド
NZ584159A (en) * 2007-09-17 2012-08-31 Enanta Pharm Inc 6,11-bridged biaryl macrolides

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI7910768A8 (en) * 1979-04-02 1996-06-30 Pliva Pharm & Chem Works Process for pripering 11-aza-4-0-cladinosyl-6-0-desosaminyl-15-ethyl- 7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl- oxacyclopentadecane-2-one and their derivatives
EP0553353A1 (en) * 1990-10-15 1993-08-04 Taisho Pharmaceutical Co. Ltd 2'-modified erythromycin or derivative thereof
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A

Also Published As

Publication number Publication date
EE05007B1 (et) 2008-04-15
EP1175429A1 (en) 2002-01-30
BG106173A (bg) 2002-07-31
CN1351606A (zh) 2002-05-29
HK1045522B (zh) 2004-08-20
CN1140535C (zh) 2004-03-03
NO320138B1 (no) 2005-10-31
DE60003671D1 (de) 2003-08-07
CA2372977A1 (en) 2000-11-09
HK1045522A1 (en) 2002-11-29
US6872707B1 (en) 2005-03-29
HUP0201146A2 (hu) 2002-07-29
PT1175429E (pt) 2003-11-28
ZA200108484B (en) 2003-03-26
NO20015346D0 (no) 2001-11-01
CZ20013913A3 (cs) 2002-04-17
PL351402A1 (en) 2003-04-07
NZ515278A (en) 2003-06-30
SK15702001A3 (sk) 2002-04-04
BR0010231A (pt) 2002-02-19
HRP990130A2 (en) 2001-10-31
DK1175429T3 (da) 2003-10-20
EP1175429B1 (en) 2003-07-02
WO2000066603A1 (en) 2000-11-09
ATE244258T1 (de) 2003-07-15
IL145986A (en) 2006-10-31
SI1175429T1 (en) 2003-12-31
IS6115A (is) 2001-10-19
KR100714740B1 (ko) 2007-05-07
UA71962C2 (en) 2005-01-17
JP2002543213A (ja) 2002-12-17
SK284513B6 (sk) 2005-05-05
EA005214B1 (ru) 2004-12-30
AU4135000A (en) 2000-11-17
HRP990130B1 (en) 2004-06-30
TR200103143T2 (tr) 2002-04-22
EE200100582A (et) 2003-02-17
EA200101170A1 (ru) 2002-04-25
NO20015346L (no) 2001-11-01
DE60003671T2 (de) 2004-06-17
MXPA01011038A (es) 2002-07-22
AU767681B2 (en) 2003-11-20
GEP20032928B (en) 2003-03-25
HUP0201146A3 (en) 2003-03-28
ES2202107T3 (es) 2004-04-01
KR20020007397A (ko) 2002-01-26

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