HUP0201146A3 - Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a, process for their preparation and pharmaceutical compositions containing them - Google Patents

Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a, process for their preparation and pharmaceutical compositions containing them

Info

Publication number
HUP0201146A3
HUP0201146A3 HU0201146A HUP0201146A HUP0201146A3 HU P0201146 A3 HUP0201146 A3 HU P0201146A3 HU 0201146 A HU0201146 A HU 0201146A HU P0201146 A HUP0201146 A HU P0201146A HU P0201146 A3 HUP0201146 A3 HU P0201146A3
Authority
HU
Hungary
Prior art keywords
homerythromycin
deoxo
aza
preparation
pharmaceutical compositions
Prior art date
Application number
HU0201146A
Other languages
English (en)
Original Assignee
Pliva Pharm & Chem Works
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Pharm & Chem Works filed Critical Pliva Pharm & Chem Works
Publication of HUP0201146A2 publication Critical patent/HUP0201146A2/hu
Publication of HUP0201146A3 publication Critical patent/HUP0201146A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
HU0201146A 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a, process for their preparation and pharmaceutical compositions containing them HUP0201146A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HR990130A HRP990130B1 (en) 1999-05-03 1999-05-03 HALOGEN DERIVATIVES 9a-N-(N'-ARYLCARBAMOYL)- AND 9a-N-(N'-ARYLTHIOCARBAMOYL)-9-DEOXO-9a-AZA-9a OF HOMOERYTHROMYCIN A

Publications (2)

Publication Number Publication Date
HUP0201146A2 HUP0201146A2 (hu) 2002-07-29
HUP0201146A3 true HUP0201146A3 (en) 2003-03-28

Family

ID=10946916

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0201146A HUP0201146A3 (en) 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a, process for their preparation and pharmaceutical compositions containing them

Country Status (33)

Country Link
US (1) US6872707B1 (hu)
EP (1) EP1175429B1 (hu)
JP (1) JP2002543213A (hu)
KR (1) KR100714740B1 (hu)
CN (1) CN1140535C (hu)
AT (1) ATE244258T1 (hu)
AU (1) AU767681B2 (hu)
BG (1) BG106173A (hu)
BR (1) BR0010231A (hu)
CA (1) CA2372977A1 (hu)
CZ (1) CZ20013913A3 (hu)
DE (1) DE60003671T2 (hu)
DK (1) DK1175429T3 (hu)
EA (1) EA005214B1 (hu)
EE (1) EE05007B1 (hu)
ES (1) ES2202107T3 (hu)
GE (1) GEP20032928B (hu)
HK (1) HK1045522B (hu)
HR (1) HRP990130B1 (hu)
HU (1) HUP0201146A3 (hu)
IL (2) IL145986A0 (hu)
IS (1) IS6115A (hu)
MX (1) MXPA01011038A (hu)
NO (1) NO320138B1 (hu)
NZ (1) NZ515278A (hu)
PL (1) PL351402A1 (hu)
PT (1) PT1175429E (hu)
SI (1) SI1175429T1 (hu)
SK (1) SK284513B6 (hu)
TR (1) TR200103143T2 (hu)
UA (1) UA71962C2 (hu)
WO (1) WO2000066603A1 (hu)
ZA (1) ZA200108484B (hu)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010146B1 (en) * 2001-02-28 2005-10-31 Pliva D.D. 9a-N-(N'-(PHENYLSULFONYL)CARBAMOYL) DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMYCIN A AND OF 5-O-DESOSAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHRONOLIDE A
HRP20020885B1 (en) 2002-11-11 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A
HRP20020886A2 (en) * 2002-11-11 2005-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. SUBSTITUTED 9a-N-[N'-(BENZENSULFONYL)CARBAMOYL-γ-AMINOPROPYL) AND 9a-N(N' -(?-CYANOETHIL)-N' -(b
HRP20020991A2 (en) * 2002-12-12 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de
HRP20030381B1 (en) * 2003-05-14 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. 3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
ES2326002T3 (es) * 2005-01-14 2009-09-28 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. 9a-carbamoil y tiocarbamoil azalidos con actividad antipaludica.
WO2009039177A1 (en) * 2007-09-17 2009-03-26 Enanta Pharmaceuticals, Inc. 6, 11-bicycloides: bridged biaryl macrolide derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU43116B (en) * 1979-04-02 1989-04-30 Pliva Pharm & Chem Works Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
EP0553353A1 (en) * 1990-10-15 1993-08-04 Taisho Pharmaceutical Co. Ltd 2'-modified erythromycin or derivative thereof
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A

Also Published As

Publication number Publication date
EA200101170A1 (ru) 2002-04-25
PT1175429E (pt) 2003-11-28
EE200100582A (et) 2003-02-17
SI1175429T1 (en) 2003-12-31
HRP990130B1 (en) 2004-06-30
BG106173A (bg) 2002-07-31
CN1140535C (zh) 2004-03-03
KR100714740B1 (ko) 2007-05-07
NO20015346L (no) 2001-11-01
JP2002543213A (ja) 2002-12-17
DE60003671D1 (de) 2003-08-07
HK1045522B (zh) 2004-08-20
NO320138B1 (no) 2005-10-31
CN1351606A (zh) 2002-05-29
US6872707B1 (en) 2005-03-29
SK15702001A3 (sk) 2002-04-04
NZ515278A (en) 2003-06-30
HK1045522A1 (en) 2002-11-29
AU4135000A (en) 2000-11-17
IL145986A (en) 2006-10-31
IS6115A (is) 2001-10-19
GEP20032928B (en) 2003-03-25
UA71962C2 (en) 2005-01-17
TR200103143T2 (tr) 2002-04-22
AU767681B2 (en) 2003-11-20
KR20020007397A (ko) 2002-01-26
SK284513B6 (sk) 2005-05-05
ZA200108484B (en) 2003-03-26
EP1175429B1 (en) 2003-07-02
NO20015346D0 (no) 2001-11-01
CA2372977A1 (en) 2000-11-09
DE60003671T2 (de) 2004-06-17
ES2202107T3 (es) 2004-04-01
IL145986A0 (en) 2002-07-25
CZ20013913A3 (cs) 2002-04-17
WO2000066603A1 (en) 2000-11-09
PL351402A1 (en) 2003-04-07
BR0010231A (pt) 2002-02-19
EA005214B1 (ru) 2004-12-30
HRP990130A2 (en) 2001-10-31
HUP0201146A2 (hu) 2002-07-29
EP1175429A1 (en) 2002-01-30
ATE244258T1 (de) 2003-07-15
MXPA01011038A (es) 2002-07-22
EE05007B1 (et) 2008-04-15
DK1175429T3 (da) 2003-10-20

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Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees