IL125717A0 - Il-8 receptor antagonists - Google Patents

Il-8 receptor antagonists

Info

Publication number
IL125717A0
IL125717A0 IL12571796A IL12571796A IL125717A0 IL 125717 A0 IL125717 A0 IL 125717A0 IL 12571796 A IL12571796 A IL 12571796A IL 12571796 A IL12571796 A IL 12571796A IL 125717 A0 IL125717 A0 IL 125717A0
Authority
IL
Israel
Prior art keywords
receptor antagonists
antagonists
receptor
Prior art date
Application number
IL12571796A
Other languages
English (en)
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Priority to IL14112196A priority Critical patent/IL141121A/en
Publication of IL125717A0 publication Critical patent/IL125717A0/xx

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/30—Oxygen atoms
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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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    • A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
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    • C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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IL12571796A 1995-02-17 1996-08-21 Il-8 receptor antagonists IL125717A0 (en)

Priority Applications (1)

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IL14112196A IL141121A (en) 1995-02-17 1996-08-21 Process for preparing cyano-phenol derivatives

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US39026095A 1995-02-17 1995-02-17
PCT/US1996/002260 WO1996025157A1 (fr) 1995-02-17 1996-02-16 Antagonistes des recepteurs d'il-8
PCT/US1996/013632 WO1997029743A1 (fr) 1995-02-17 1996-08-21 Antagonistes de recepteurs de l'interleukine-8

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JP (2) JPH11503110A (fr)
KR (1) KR19990082622A (fr)
CN (2) CN1539816A (fr)
AU (1) AU725456B2 (fr)
BG (1) BG102690A (fr)
BR (1) BR9612779A (fr)
CA (1) CA2245927A1 (fr)
EA (1) EA001436B1 (fr)
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IL (1) IL125717A0 (fr)
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PL (1) PL328562A1 (fr)
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WO1997029743A1 (fr) 1997-08-21
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US5886044A (en) 1999-03-23
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