IL114589A - Intermediates for the preparation of erythromycin derivatives - Google Patents

Intermediates for the preparation of erythromycin derivatives

Info

Publication number
IL114589A
IL114589A IL11458991A IL11458991A IL114589A IL 114589 A IL114589 A IL 114589A IL 11458991 A IL11458991 A IL 11458991A IL 11458991 A IL11458991 A IL 11458991A IL 114589 A IL114589 A IL 114589A
Authority
IL
Israel
Prior art keywords
radical
methyl
formula
carbon atoms
compounds
Prior art date
Application number
IL11458991A
Other languages
English (en)
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9014499A external-priority patent/FR2669337B1/fr
Priority claimed from FR9106333A external-priority patent/FR2677025B1/fr
Priority claimed from FR9110728A external-priority patent/FR2680790B1/fr
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IL114589A publication Critical patent/IL114589A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Virology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
IL11458991A 1990-11-21 1991-11-07 Intermediates for the preparation of erythromycin derivatives IL114589A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9014499A FR2669337B1 (fr) 1990-11-21 1990-11-21 Nouveaux derives descladinosyles de l'erythromycine, leur procede de preparation et leur application comme medicaments.
FR9106333A FR2677025B1 (fr) 1991-05-27 1991-05-27 Nouveaux derives descladinosyles de l'erythromycine, leur procede de preparation et leur application comme medicaments.
FR9110728A FR2680790B1 (fr) 1991-08-29 1991-08-29 Nouveaux derives descladinosyles de l'erythromycine, leur procede de preparation et leur application comme medicaments.
IL99995A IL99995A (en) 1990-11-21 1991-11-07 Erythromycin derivatives, their preparation and pharmaceutical compositions containing them

Publications (1)

Publication Number Publication Date
IL114589A true IL114589A (en) 1999-12-22

Family

ID=27252354

Family Applications (3)

Application Number Title Priority Date Filing Date
IL99995A IL99995A (en) 1990-11-21 1991-11-07 Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
IL11458991A IL114589A (en) 1990-11-21 1991-11-07 Intermediates for the preparation of erythromycin derivatives
IL11458995A IL114589A0 (en) 1990-11-21 1995-07-14 Intermediates for the preparation of erythromycin derivatives

Family Applications Before (1)

Application Number Title Priority Date Filing Date
IL99995A IL99995A (en) 1990-11-21 1991-11-07 Erythromycin derivatives, their preparation and pharmaceutical compositions containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL11458995A IL114589A0 (en) 1990-11-21 1995-07-14 Intermediates for the preparation of erythromycin derivatives

Country Status (26)

Country Link
US (3) US5444051A (pt)
EP (1) EP0487411B1 (pt)
JP (1) JP3130097B2 (pt)
KR (1) KR100189597B1 (pt)
CN (1) CN1033974C (pt)
AT (1) ATE133683T1 (pt)
AU (1) AU640290B2 (pt)
BR (1) BR9105062A (pt)
CA (1) CA2055912C (pt)
CZ (1) CZ290651B6 (pt)
DE (1) DE69116815T2 (pt)
DK (1) DK0487411T3 (pt)
ES (1) ES2082952T3 (pt)
FI (1) FI102281B (pt)
GR (1) GR3018848T3 (pt)
HU (1) HU218787B (pt)
IE (1) IE74713B1 (pt)
IL (3) IL99995A (pt)
MA (1) MA22344A1 (pt)
MX (1) MX9102159A (pt)
NZ (1) NZ240684A (pt)
OA (1) OA09523A (pt)
PL (2) PL169422B1 (pt)
PT (1) PT99569B (pt)
RU (1) RU2100367C1 (pt)
SK (1) SK281550B6 (pt)

Families Citing this family (141)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5523399A (en) * 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
WO1993021199A1 (fr) * 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. Derive de 5-o-desosaminylerythronolide
FR2707088B1 (fr) * 1993-07-02 1995-08-25 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
US5602239A (en) * 1993-01-26 1997-02-11 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
FR2702480B1 (fr) * 1993-03-09 1995-04-28 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2713226B1 (fr) * 1993-12-03 1996-01-05 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2727969B1 (fr) * 1994-12-09 1997-01-17 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
IT1276901B1 (it) * 1994-12-13 1997-11-03 Zambon Spa Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica
FR2732684B1 (fr) * 1995-04-06 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
KR19990067333A (ko) * 1995-11-08 1999-08-16 스티븐 에프. 웨인스톡 에리트로마이신 a 및 b의 3-데옥시-3-데스클라디노즈 유도체
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EP0487411A1 (fr) 1992-05-27
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PL292455A1 (en) 1992-08-10
PT99569B (pt) 1999-04-30
FI102281B1 (fi) 1998-11-13
PT99569A (pt) 1992-10-30
CN1065069A (zh) 1992-10-07
KR100189597B1 (ko) 1999-06-01
CN1033974C (zh) 1997-02-05
MA22344A1 (fr) 1992-07-01
US5770579A (en) 1998-06-23
PL169422B1 (pl) 1996-07-31
ATE133683T1 (de) 1996-02-15
ES2082952T3 (es) 1996-04-01
RU2100367C1 (ru) 1997-12-27
OA09523A (fr) 1992-11-15
EP0487411B1 (fr) 1996-01-31
IL114589A0 (en) 1995-11-27
US5444051A (en) 1995-08-22
IL99995A (en) 1997-11-20
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CA2055912C (fr) 2002-03-19
AU640290B2 (en) 1993-08-19
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HUT61564A (en) 1993-01-28
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IL99995A0 (en) 1992-08-18
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US5561118A (en) 1996-10-01
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