IL101560A - Compressed diazepines, their preparation and pharmaceutical preparations containing them - Google Patents

Compressed diazepines, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL101560A
IL101560A IL10156092A IL10156092A IL101560A IL 101560 A IL101560 A IL 101560A IL 10156092 A IL10156092 A IL 10156092A IL 10156092 A IL10156092 A IL 10156092A IL 101560 A IL101560 A IL 101560A
Authority
IL
Israel
Prior art keywords
dihydro
formula
piperidinyl
acetyl
benzodiazepin
Prior art date
Application number
IL10156092A
Other languages
English (en)
Hebrew (he)
Other versions
IL101560A0 (en
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of IL101560A0 publication Critical patent/IL101560A0/xx
Publication of IL101560A publication Critical patent/IL101560A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
IL10156092A 1991-04-12 1992-04-10 Compressed diazepines, their preparation and pharmaceutical preparations containing them IL101560A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4112014A DE4112014A1 (de) 1991-04-12 1991-04-12 Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende mittel zur behandlung von erkrankungen des zentralnervensystems und zur foerderung der cerebralen durchblutung

Publications (2)

Publication Number Publication Date
IL101560A0 IL101560A0 (en) 1992-12-30
IL101560A true IL101560A (en) 1996-03-31

Family

ID=6429483

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10156092A IL101560A (en) 1991-04-12 1992-04-10 Compressed diazepines, their preparation and pharmaceutical preparations containing them

Country Status (28)

Country Link
US (1) US5641772A (sk)
EP (1) EP0508370B1 (sk)
JP (1) JPH0597845A (sk)
KR (1) KR100196969B1 (sk)
AT (1) ATE140004T1 (sk)
AU (1) AU653802B2 (sk)
CA (1) CA2065800A1 (sk)
CZ (1) CZ283399B6 (sk)
DE (2) DE4112014A1 (sk)
DK (1) DK0508370T3 (sk)
ES (1) ES2090396T3 (sk)
FI (1) FI97470C (sk)
GR (1) GR3020860T3 (sk)
HR (1) HRP940753A2 (sk)
HU (2) HUT61301A (sk)
IE (1) IE921147A1 (sk)
IL (1) IL101560A (sk)
MX (1) MX9201675A (sk)
NO (1) NO180303C (sk)
NZ (1) NZ242305A (sk)
PL (1) PL169745B1 (sk)
RU (1) RU2081870C1 (sk)
SG (1) SG48793A1 (sk)
SI (1) SI9210325A (sk)
SK (1) SK279466B6 (sk)
TW (1) TW205551B (sk)
YU (1) YU48645B (sk)
ZA (1) ZA922617B (sk)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4332168A1 (de) * 1993-02-22 1995-03-23 Thomae Gmbh Dr K Cyclische Derivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
ATE221067T1 (de) * 1993-04-05 2002-08-15 Pharmaceutical Discovery Corp Pyrido(2,3-b)(1,4)benzodiazepinone als m2- rezeptorligand zur behandlung neurologischer störungen
AU3754495A (en) * 1994-10-31 1996-05-23 Yamanouchi Pharmaceutical Co., Ltd. Novel benzodiazepinone derivative and medicinal composition thereof
WO2007056388A2 (en) * 2005-11-07 2007-05-18 The General Hospital Corporation Compositions and methods for modulating poly (adp-ribose) polymerase activity
EP2173355A2 (en) * 2007-07-02 2010-04-14 AC Immune S.A. Pirenzepine and derivatives thereof as anti-amyloid agents
KR102478480B1 (ko) 2021-11-17 2022-12-19 주식회사 지농 통신 데이터 사용량을 최소화한 스마트팜 제어 및 동작확인 장치
KR20240109659A (ko) 2023-01-04 2024-07-12 주식회사 다온정보기술 스마트기기를 이용한 스마트팜 제어시스템

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3409237A1 (de) * 1984-03-14 1985-09-19 Dr. Karl Thomae Gmbh, 7950 Biberach Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3735895A1 (de) * 1987-10-23 1989-05-03 Thomae Gmbh Dr K Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3919076A1 (de) * 1989-06-10 1990-12-13 Thomae Gmbh Dr K Mittel zur behandlung von erkrankungen des zentralnervensystems und zur foerderung der cerebralen durchblutung

Also Published As

Publication number Publication date
HRP940753A2 (en) 1997-08-31
FI921589A (fi) 1992-10-13
HU9201247D0 (en) 1992-07-28
MX9201675A (es) 1992-10-01
FI97470C (fi) 1996-12-27
ES2090396T3 (es) 1996-10-16
IE921147A1 (en) 1992-10-21
NZ242305A (en) 1994-09-27
US5641772A (en) 1997-06-24
SK279466B6 (sk) 1998-11-04
KR920019792A (ko) 1992-11-20
EP0508370A1 (de) 1992-10-14
ATE140004T1 (de) 1996-07-15
PL294184A1 (en) 1993-05-04
FI97470B (fi) 1996-09-13
IL101560A0 (en) 1992-12-30
PL169745B1 (pl) 1996-08-30
AU1481492A (en) 1992-10-15
YU32592A (sh) 1998-09-18
SI9210325A (en) 1995-04-30
CA2065800A1 (en) 1992-10-13
JPH0597845A (ja) 1993-04-20
HU211156A9 (en) 1995-10-30
NO180303B (no) 1996-12-16
DE4112014A1 (de) 1992-10-15
CZ283399B6 (cs) 1998-04-15
ZA922617B (en) 1993-10-11
CZ111192A3 (en) 1993-04-14
SG48793A1 (en) 1998-05-18
RU2081870C1 (ru) 1997-06-20
TW205551B (sk) 1993-05-11
GR3020860T3 (en) 1996-11-30
HUT61301A (en) 1992-12-28
FI921589A0 (fi) 1992-04-10
NO180303C (no) 1997-03-26
DK0508370T3 (da) 1996-11-04
DE59206679D1 (de) 1996-08-08
SK111192A3 (en) 1995-04-12
EP0508370B1 (de) 1996-07-03
NO921447D0 (no) 1992-04-10
NO921447L (no) 1992-10-13
YU48645B (sh) 1999-06-15
KR100196969B1 (ko) 1999-06-15
AU653802B2 (en) 1994-10-13

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees