ID28695A - TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA - Google Patents

TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA

Info

Publication number
ID28695A
ID28695A IDW20002562A ID20002562A ID28695A ID 28695 A ID28695 A ID 28695A ID W20002562 A IDW20002562 A ID W20002562A ID 20002562 A ID20002562 A ID 20002562A ID 28695 A ID28695 A ID 28695A
Authority
ID
Indonesia
Prior art keywords
tiepin
benzo
designs
dioxide
compounds
Prior art date
Application number
IDW20002562A
Other languages
English (en)
Indonesian (id)
Inventor
Wendelin Dr Frick
Alfons Dr Enhsen
Heiner Dr Glombik
Hubert Dr Heuer
Original Assignee
Aventis Pharma Deutschland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Deutschland filed Critical Aventis Pharma Deutschland
Publication of ID28695A publication Critical patent/ID28695A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02—Seven-membered rings
    • C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/04—Drugs for disorders of the urinary system for urolithiasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08G—MACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G65/00—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule
    • C08G65/02—Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule from cyclic ethers by opening of the heterocyclic ring
    • C08G65/32—Polymers modified by chemical after-treatment
    • C08G65/329—Polymers modified by chemical after-treatment with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Genetics & Genomics (AREA)
  • Polymers & Plastics (AREA)
  • Urology & Nephrology (AREA)
  • Biophysics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
IDW20002562A 1998-06-10 1999-05-28 TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA ID28695A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19825804A DE19825804C2 (de) 1998-06-10 1998-06-10 1,4-Benzothiepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
ID28695A true ID28695A (id) 2001-06-28

Family

ID=7870440

Family Applications (2)

Application Number Title Priority Date Filing Date
IDW20002562A ID28695A (id) 1998-06-10 1999-05-28 TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA
IDW20002564A ID26876A (id) 1998-06-10 1999-05-29 Derivat-derivat benzotiepin 1,1-dioksida, proses pembuatannya, bahan-bahan farmasi yang terdiri dari senyawa-senyawa ini dan penggunaannya

Family Applications After (1)

Application Number Title Priority Date Filing Date
IDW20002564A ID26876A (id) 1998-06-10 1999-05-29 Derivat-derivat benzotiepin 1,1-dioksida, proses pembuatannya, bahan-bahan farmasi yang terdiri dari senyawa-senyawa ini dan penggunaannya

Country Status (26)

Country Link
US (1) US6387944B1 (ja)
EP (2) EP1086092B1 (ja)
JP (2) JP4374426B2 (ja)
KR (2) KR100681721B1 (ja)
CN (2) CN1127497C (ja)
AR (2) AR018633A1 (ja)
AT (2) ATE227715T1 (ja)
AU (2) AU753275B2 (ja)
BR (2) BR9912188B1 (ja)
CA (2) CA2334775C (ja)
CZ (2) CZ297989B6 (ja)
DE (3) DE19825804C2 (ja)
DK (2) DK1086092T3 (ja)
ES (2) ES2182535T3 (ja)
HK (2) HK1039490A1 (ja)
HU (2) HU229761B1 (ja)
ID (2) ID28695A (ja)
IL (1) IL140078A (ja)
NO (1) NO327075B1 (ja)
NZ (1) NZ508681A (ja)
PL (2) PL196074B1 (ja)
PT (2) PT1086092E (ja)
RU (2) RU2215001C2 (ja)
TR (2) TR200003634T2 (ja)
WO (2) WO1999064410A1 (ja)
ZA (2) ZA200007060B (ja)

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SE0000772D0 (sv) 2000-03-08 2000-03-08 Astrazeneca Ab Chemical compounds
DE50111751D1 (de) * 2000-12-21 2007-02-08 Sanofi Aventis Deutschland Neue diphenzylazetidinone, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung zur behandlung von lipidstoffwechselstörungen
EG26979A (en) 2000-12-21 2015-03-01 Astrazeneca Ab Chemical compounds
CA2457976A1 (en) * 2001-08-22 2003-03-06 Aventis Pharma Deutschland Gmbh Combined preparations, containing 1,4-benzothiepine-1,1-dioxide derivatives and other active substances, and the use thereof
GB0121337D0 (en) 2001-09-04 2001-10-24 Astrazeneca Ab Chemical compounds
GB0121622D0 (en) 2001-09-07 2001-10-31 Astrazeneca Ab Chemical compounds
GB0121621D0 (en) 2001-09-07 2001-10-31 Astrazeneca Ab Chemical compounds
RU2305681C2 (ru) 2001-09-08 2007-09-10 Астразенека Аб Производные бензотиадиазепина, способ их получения (варианты)
GB0209467D0 (en) 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
GB0213669D0 (en) 2002-06-14 2002-07-24 Astrazeneca Ab Chemical compounds
SE0201937D0 (sv) 2002-06-20 2002-06-20 Astrazeneca Ab Therapeutic agents
FR2848452B1 (fr) * 2002-12-12 2007-04-06 Aventis Pharma Sa Application des inhibiteurs de recapture intestinale des acides biliaires pour la prevention et le traitement de la maladie d'alzheimer
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GB0304194D0 (en) 2003-02-25 2003-03-26 Astrazeneca Ab Chemical compounds
GB0307918D0 (en) 2003-04-05 2003-05-14 Astrazeneca Ab Therapeutic use
DE102006053636B4 (de) * 2006-11-14 2008-09-18 Sanofi-Aventis Deutschland Gmbh Neue mit Cyclohexylresten substituierte 1,4-Benzothiepin-1,1-Dioxidderivate und deren Verwendung
DE102006053635B4 (de) * 2006-11-14 2011-06-30 Sanofi-Aventis Deutschland GmbH, 65929 Neue mit Benzylresten substituierte 1,4-Benzothiepin-1,1-Dioxidderivate, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
US20100221513A1 (en) * 2008-09-05 2010-09-02 Wisconsin Alumni Research Foundation Self sintering transparent nanoporous thin-films for use in self-cleaning, anti-fogging, anti-corrosion, anti-erosion electronic and optical applications
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AU2011326872C1 (en) 2010-11-08 2015-02-19 Albireo Ab A pharmaceutical combination comprising an IBAT inhibitor and a bile acid binder
BR112013010157B1 (pt) 2010-11-08 2020-02-04 Albireo Ab iinibidores do ibat, seus usos, e composição e combinações farmacêuticas
KR102051030B1 (ko) * 2011-10-28 2019-12-02 루메나 파마수티컬즈, 인코포레이티드 소아 담즙울체성 간 질환 치료용 담즙산 재순환 억제제
CN104023718B (zh) 2011-10-28 2017-04-05 鲁美纳医药公司 用于治疗高胆血症和胆汁淤积性肝病的胆汁酸再循环抑制剂
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CN106659726A (zh) 2014-06-25 2017-05-10 Ea制药株式会社 固体制剂及其着色防止或着色减少方法
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JP3304093B2 (ja) * 1994-09-13 2002-07-22 モンサント カンパニー 回腸の胆汁酸輸送及びタウロコール酸塩吸収の阻害活性を有する新規ベンゾチエピン類
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Also Published As

Publication number Publication date
AU4501999A (en) 1999-12-30
CZ297925B6 (cs) 2007-05-02
RU2215001C2 (ru) 2003-10-27
KR100562184B1 (ko) 2006-03-20
EP1086113A2 (de) 2001-03-28
HUP0102256A1 (hu) 2001-12-28
BR9911123A (pt) 2006-01-03
JP2002517490A (ja) 2002-06-18
AR018634A1 (es) 2001-11-28
RU2220141C2 (ru) 2003-12-27
US6387944B1 (en) 2002-05-14
PL196074B1 (pl) 2007-12-31
ZA200007061B (en) 2001-07-18
ES2182535T3 (es) 2003-03-01
AR018633A1 (es) 2001-11-28
CZ297989B6 (cs) 2007-05-16
PL344827A1 (en) 2001-11-19
IL140078A0 (en) 2002-02-10
WO1999064409A2 (de) 1999-12-16
EP1086092B1 (de) 2002-11-13
WO1999064410A1 (de) 1999-12-16
ATE227715T1 (de) 2002-11-15
ES2215387T3 (es) 2004-10-01
AU4503199A (en) 1999-12-30
PL345901A1 (en) 2002-01-14
DE19825804C2 (de) 2000-08-24
CA2334775C (en) 2009-10-13
KR20010052682A (ko) 2001-06-25
CZ20004592A3 (cs) 2001-04-11
CN1152039C (zh) 2004-06-02
DE59908522D1 (de) 2004-03-18
EP1086113B1 (de) 2004-02-11
HU228570B1 (en) 2013-04-29
HK1039490A1 (en) 2002-04-26
ID26876A (id) 2001-02-15
JP2002517491A (ja) 2002-06-18
EP1086092A1 (de) 2001-03-28
BR9912188B1 (pt) 2010-12-14
ZA200007060B (en) 2001-07-18
DE59903411D1 (de) 2002-12-19
HUP0102554A3 (en) 2002-12-28
DK1086113T3 (da) 2004-05-24
NO20006251L (no) 2001-02-07
DK1086092T3 (da) 2003-03-10
AU752633B2 (en) 2002-09-26
TR200003634T2 (tr) 2001-06-21
JP4374426B2 (ja) 2009-12-02
BR9912188A (pt) 2001-04-10
NO327075B1 (no) 2009-04-20
NZ508681A (en) 2002-06-28
DE19825804A1 (de) 1999-12-16
CZ20004591A3 (cs) 2001-04-11
HK1036799A1 (en) 2002-01-18
AU753275B2 (en) 2002-10-10
IL140078A (en) 2004-08-31
KR100681721B1 (ko) 2007-02-15
CA2334773A1 (en) 1999-12-16
TR200003632T2 (tr) 2001-04-20
PL196057B1 (pl) 2007-11-30
CN1127497C (zh) 2003-11-12
WO1999064409A3 (de) 2000-03-02
ATE259372T1 (de) 2004-02-15
HU229761B1 (hu) 2014-06-30
HUP0102256A3 (en) 2002-04-29
CN1305487A (zh) 2001-07-25
CA2334773C (en) 2009-05-26
HUP0102554A1 (hu) 2001-10-28
KR20010052701A (ko) 2001-06-25
CN1305469A (zh) 2001-07-25
PT1086092E (pt) 2003-03-31
BR9911123B1 (pt) 2010-12-14
CA2334775A1 (en) 1999-12-16
JP3374129B2 (ja) 2003-02-04
PT1086113E (pt) 2004-06-30
NO20006251D0 (no) 2000-12-08

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