HUT68667A - Fused ring analogs of nitrogen containing nonaromatic heterocycles - Google Patents

Fused ring analogs of nitrogen containing nonaromatic heterocycles Download PDF

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Publication number
HUT68667A
HUT68667A HU9300898A HU89893A HUT68667A HU T68667 A HUT68667 A HU T68667A HU 9300898 A HU9300898 A HU 9300898A HU 89893 A HU89893 A HU 89893A HU T68667 A HUT68667 A HU T68667A
Authority
HU
Hungary
Prior art keywords
compound
phenyl
alkyl
group
amino
Prior art date
Application number
HU9300898A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9300898D0 (en
Inventor
Manoj Chandrasinhji Desai
Terry Jay Rosen
Harry Ralph Howard
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of HU9300898D0 publication Critical patent/HU9300898D0/hu
Publication of HUT68667A publication Critical patent/HUT68667A/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Indole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Polyoxymethylene Polymers And Polymers With Carbon-To-Carbon Bonds (AREA)
  • Eye Examination Apparatus (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Electroluminescent Light Sources (AREA)
HU9300898A 1990-09-28 1991-08-20 Fused ring analogs of nitrogen containing nonaromatic heterocycles HUT68667A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59042390A 1990-09-28 1990-09-28

Publications (2)

Publication Number Publication Date
HU9300898D0 HU9300898D0 (en) 1993-06-28
HUT68667A true HUT68667A (en) 1995-07-28

Family

ID=24362216

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9300898A HUT68667A (en) 1990-09-28 1991-08-20 Fused ring analogs of nitrogen containing nonaromatic heterocycles

Country Status (22)

Country Link
EP (1) EP0550635B1 (env)
JP (1) JPH0772175B2 (env)
CN (1) CN1060285A (env)
AT (1) ATE121389T1 (env)
AU (1) AU651145B2 (env)
BR (1) BR9106905A (env)
CA (1) CA2089736A1 (env)
CZ (1) CZ387492A3 (env)
DE (1) DE69109125T2 (env)
DK (1) DK0550635T3 (env)
ES (1) ES2071334T3 (env)
FI (1) FI931370A7 (env)
HU (1) HUT68667A (env)
IE (1) IE66042B1 (env)
IL (1) IL99525A0 (env)
MX (1) MX9101274A (env)
NO (1) NO931151L (env)
PT (1) PT99064A (env)
TW (1) TW199144B (env)
WO (1) WO1992006079A1 (env)
YU (1) YU159291A (env)
ZA (1) ZA917744B (env)

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US5719147A (en) * 1992-06-29 1998-02-17 Merck & Co., Inc. Morpholine and thiomorpholine tachykinin receptor antagonists
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GB9216911D0 (en) * 1992-08-10 1992-09-23 Merck Sharp & Dohme Therapeutic agents
US5721255A (en) * 1992-08-19 1998-02-24 Pfizer Inc. Substituted benzylamino nitrogen containing non-aromatic heterocycles
US5387595A (en) * 1992-08-26 1995-02-07 Merck & Co., Inc. Alicyclic compounds as tachykinin receptor antagonists
EP0675886B1 (en) * 1992-12-10 2000-07-05 Pfizer Inc. Aminomethylene substituted non-aromatic heterocycles and use as substance p antagonists
US5344830A (en) * 1992-12-10 1994-09-06 Merck & Co., Inc. N,N-diacylpiperazine tachykinin antagonists
US5830854A (en) * 1992-12-14 1998-11-03 Merck Sharp & Dohme, Limited Method of treating cystic fibrosis using a tachykinin receptor antagonist
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US5393762A (en) * 1993-06-04 1995-02-28 Pfizer Inc. Pharmaceutical agents for treatment of emesis
US5854262A (en) * 1993-10-07 1998-12-29 Pfizer Inc. Aminomethylene substituted non-aromatic heterocycles and use as substance P antagonists
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Also Published As

Publication number Publication date
ES2071334T3 (es) 1995-06-16
MX9101274A (es) 1992-05-04
CZ387492A3 (en) 1994-02-16
EP0550635A1 (en) 1993-07-14
NO931151D0 (no) 1993-03-26
IE66042B1 (en) 1995-12-13
DE69109125T2 (de) 1995-09-28
FI931370L (fi) 1993-03-26
BR9106905A (pt) 1993-08-17
HU9300898D0 (en) 1993-06-28
FI931370A0 (fi) 1993-03-26
JPH0772175B2 (ja) 1995-08-02
CA2089736A1 (en) 1992-03-29
FI931370A7 (fi) 1993-03-26
NO931151L (no) 1993-03-26
EP0550635B1 (en) 1995-04-19
YU159291A (sh) 1994-01-20
DK0550635T3 (da) 1995-09-04
PT99064A (pt) 1992-08-31
CN1060285A (zh) 1992-04-15
AU8746391A (en) 1992-04-28
TW199144B (env) 1993-02-01
IE913396A1 (en) 1992-04-08
ATE121389T1 (de) 1995-05-15
IL99525A0 (en) 1992-08-18
ZA917744B (en) 1993-03-29
AU651145B2 (en) 1994-07-14
JPH06501267A (ja) 1994-02-10
DE69109125D1 (de) 1995-05-24
WO1992006079A1 (en) 1992-04-16

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