HUP0300992A3 - Method for producing 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinones - Google Patents

Method for producing 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinones

Info

Publication number
HUP0300992A3
HUP0300992A3 HU0300992A HUP0300992A HUP0300992A3 HU P0300992 A3 HUP0300992 A3 HU P0300992A3 HU 0300992 A HU0300992 A HU 0300992A HU P0300992 A HUP0300992 A HU P0300992A HU P0300992 A3 HUP0300992 A3 HU P0300992A3
Authority
HU
Hungary
Prior art keywords
phthalazinones
heteroaryl
halogen
methyl
producing
Prior art date
Application number
HU0300992A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of HUP0300992A2 publication Critical patent/HUP0300992A2/hu
Publication of HUP0300992A3 publication Critical patent/HUP0300992A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
HU0300992A 1999-12-23 2000-12-20 Method for producing 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinones HUP0300992A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19963607A DE19963607B4 (de) 1999-12-23 1999-12-23 Verfahren zur Herstellung von 4-(Heteroaryl-methyl) halogen-1(2H)-phthalazinonen
PCT/EP2000/013027 WO2001047912A1 (de) 1999-12-23 2000-12-20 Verfahren zur herstellung von 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinonen

Publications (2)

Publication Number Publication Date
HUP0300992A2 HUP0300992A2 (hu) 2003-08-28
HUP0300992A3 true HUP0300992A3 (en) 2005-11-28

Family

ID=7934888

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0300992A HUP0300992A3 (en) 1999-12-23 2000-12-20 Method for producing 4-(heteroaryl-methyl)-halogen-1(2h)-phthalazinones

Country Status (31)

Country Link
US (1) US6891041B2 (enExample)
EP (1) EP1242405B1 (enExample)
JP (1) JP2003529555A (enExample)
KR (1) KR100654265B1 (enExample)
CN (1) CN1221545C (enExample)
AT (1) ATE273972T1 (enExample)
AU (1) AU772981B2 (enExample)
BG (1) BG65387B1 (enExample)
BR (1) BR0016634A (enExample)
CA (1) CA2395407C (enExample)
CZ (1) CZ20022146A3 (enExample)
DE (2) DE19963607B4 (enExample)
DK (1) DK1242405T3 (enExample)
EE (1) EE04940B1 (enExample)
ES (1) ES2223626T3 (enExample)
HR (1) HRP20020605B1 (enExample)
HU (1) HUP0300992A3 (enExample)
IL (2) IL150017A0 (enExample)
MX (1) MXPA02006224A (enExample)
NO (1) NO321357B1 (enExample)
NZ (1) NZ519285A (enExample)
PL (1) PL200714B1 (enExample)
PT (1) PT1242405E (enExample)
RO (1) RO121211B1 (enExample)
RS (1) RS50458B (enExample)
RU (1) RU2250900C2 (enExample)
SI (1) SI1242405T1 (enExample)
SK (1) SK285522B6 (enExample)
UA (1) UA72021C2 (enExample)
WO (1) WO2001047912A1 (enExample)
ZA (1) ZA200205853B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1296984B1 (it) * 1997-12-19 1999-08-03 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
US7151102B2 (en) * 2000-10-30 2006-12-19 Kudos Pharmaceuticals Limited Phthalazinone derivatives
GB0419072D0 (en) * 2004-08-26 2004-09-29 Kudos Pharm Ltd Phthalazinone derivatives
TWI404716B (zh) * 2006-10-17 2013-08-11 Kudos Pharm Ltd 酞嗪酮（ｐｈｔｈａｌａｚｉｎｏｎｅ）衍生物
KR101598231B1 (ko) * 2007-10-17 2016-02-26 쿠도스 파마슈티칼스 리미티드 4-[3-(4-시클로프로판카르보닐-피페라진-1-카르보닐)-4-플루오로-벤질]-2ｈ-프탈라진-1-온
CA2737400C (en) * 2008-10-07 2016-11-22 Astrazeneca Uk Limited Pharmaceutical formulation 514
JP6545148B2 (ja) 2013-03-13 2019-07-17 フラットリー ディスカバリー ラブ，エルエルシー ピリダジノン化合物及び嚢胞性線維症の治療のための方法
WO2016146303A1 (en) * 2015-03-19 2016-09-22 Clariant International Ltd Biodegradable sugar-amide-surfactants for enhanced oil recovery

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE567431A (enExample) * 1957-05-07
GB1293565A (en) * 1969-05-03 1972-10-18 Aspro Nicholas Ltd Aminophthalazines and pharmaceutical compositions thereof
IE47592B1 (en) * 1977-12-29 1984-05-02 Ici Ltd Enzyme inhibitory phthalazin-4-ylacetic acid derivatives, pharmaceutical compositions thereof,and process for their manufacture
EP0634404A1 (en) * 1993-07-13 1995-01-18 Rhone Poulenc Agriculture Ltd. Phtalazin derivatives and their use as pesticides
JP3919835B2 (ja) * 1994-08-09 2007-05-30 エーザイ・アール・アンド・ディー・マネジメント株式会社 縮合ピリダジン系化合物
NZ290952A (en) * 1994-08-09 1998-05-27 Eisai Co Ltd Phthalazine derivatives optionally substituted in position-1 by (generally benzyl) amino groups
RU2128175C1 (ru) * 1994-08-09 1999-03-27 Эйсай Ко., Лтд. Конденсированный пиридазин или его фармакологически приемлемая соль, средство, проявляющее ингибирующую активность в отношении циклической гмф- фосфодиэстеразы
CA2275686C (en) * 1996-12-18 2006-10-17 Neurogen Corporation Isoquinolinamine and phthalazinamine derivatives which interact with crf receptors
CO4950519A1 (es) * 1997-02-13 2000-09-01 Novartis Ag Ftalazinas, preparaciones farmaceuticas que las comprenden y proceso para su preparacion
IT1296984B1 (it) * 1997-12-19 1999-08-03 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
ITMI981671A1 (it) * 1998-07-21 2000-01-21 Zambon Spa Derivati ftalazinici inibitori della fosfodisterasi 4
ITMI981670A1 (it) * 1998-07-21 2000-01-21 Zambon Spa Derivati ftalazinici inibitori della fosfodiesterasi 4
ITMI20000261A1 (it) * 2000-02-16 2001-08-16 Zambon Group Processo per la preparazione di piridiniliden-ftalidi

Also Published As

Publication number Publication date
DK1242405T3 (da) 2004-11-01
DE19963607B4 (de) 2005-12-15
RS50458B (sr) 2010-03-02
DE50007520D1 (de) 2004-09-23
US20040192695A1 (en) 2004-09-30
EE04940B1 (et) 2007-12-17
PT1242405E (pt) 2004-11-30
HK1055296A1 (en) 2004-01-02
HRP20020605B1 (en) 2007-06-30
EE200200307A (et) 2003-06-16
BG106843A (en) 2003-02-28
YU47302A (sh) 2005-06-10
MXPA02006224A (es) 2002-12-05
CA2395407C (en) 2009-04-28
NO20023014D0 (no) 2002-06-21
PL200714B1 (pl) 2009-01-30
CN1413203A (zh) 2003-04-23
NZ519285A (en) 2004-12-24
EP1242405A1 (de) 2002-09-25
KR100654265B1 (ko) 2006-12-07
JP2003529555A (ja) 2003-10-07
NO321357B1 (no) 2006-05-02
ES2223626T3 (es) 2005-03-01
IL150017A0 (en) 2002-12-01
KR20020062363A (ko) 2002-07-25
ZA200205853B (en) 2004-02-18
CA2395407A1 (en) 2001-07-05
SI1242405T1 (en) 2005-02-28
EP1242405B1 (de) 2004-08-18
BG65387B1 (bg) 2008-05-30
US6891041B2 (en) 2005-05-10
PL355525A1 (en) 2004-05-04
IL150017A (en) 2006-12-31
RU2002119559A (ru) 2004-01-10
AU772981B2 (en) 2004-05-13
SK8922002A3 (en) 2002-11-06
HRP20020605A2 (en) 2004-12-31
CN1221545C (zh) 2005-10-05
CZ20022146A3 (cs) 2002-09-11
AU2012201A (en) 2001-07-09
ATE273972T1 (de) 2004-09-15
DE19963607A1 (de) 2001-07-12
UA72021C2 (en) 2005-01-17
RU2250900C2 (ru) 2005-04-27
BR0016634A (pt) 2002-10-15
HUP0300992A2 (hu) 2003-08-28
NO20023014L (no) 2002-06-21
SK285522B6 (sk) 2007-03-01
WO2001047912A1 (de) 2001-07-05
RO121211B1 (ro) 2007-01-30

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Legal Events

Date Code Title Description
FD9A Lapse of provisional protection due to non-payment of fees