HRP20161408T1 - Cefalosporin koji sadrži katehol skupinu - Google Patents

Cefalosporin koji sadrži katehol skupinu Download PDF

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Publication number
HRP20161408T1
HRP20161408T1 HRP20161408TT HRP20161408T HRP20161408T1 HR P20161408 T1 HRP20161408 T1 HR P20161408T1 HR P20161408T T HRP20161408T T HR P20161408TT HR P20161408 T HRP20161408 T HR P20161408T HR P20161408 T1 HRP20161408 T1 HR P20161408T1
Authority
HR
Croatia
Prior art keywords
compound
cephalosporin
ester
amino
pharmaceutically acceptable
Prior art date
Application number
HRP20161408TT
Other languages
English (en)
Inventor
Yasuhiro Nishitani
Kenji Yamawaki
Yusuke Takeoka
Hideki Sugimoto
Shinya Hisakawa
Toshiaki Aoki
Original Assignee
Shionogi & Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42128829&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20161408(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Shionogi & Co., Ltd. filed Critical Shionogi & Co., Ltd.
Publication of HRP20161408T1 publication Critical patent/HRP20161408T1/hr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D505/10—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D505/12—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 substituted in position 7
    • C07D505/14—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 substituted in position 7 with hetero atoms directly attached in position 7
    • C07D505/16—Nitrogen atoms
    • C07D505/18—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof
    • C07D505/20—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D505/24—Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen further substituted by doubly-bound nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C07D519/06—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00 containing at least one condensed beta-lactam ring system, provided for by groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00, e.g. a penem or a cepham system
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Claims (4)

1. Spoj s formulom: [image] ili njegov ester, zaštićeni spoj na amino na prstenu u 7-bočnom lancu, njegova farmaceutski prihvatljiva sol, ili njegov solvat.
2. Farmaceutski pripravak, naznačen time da sadrži spoj ili njegov ester, zaštićeni spoj na amino na prstenu u 7-bočnom lancu, njegova farmaceutski prihvatljiva sol, ili njegov solvat prema zahtjevu 1.
3. Farmaceutski pripravak prema patentnom zahtjevu 2, naznačen time da je za uporabu za liječenje antimikrobne infekcije.
4. Spoj ili njegov ester, zaštićeni spoj na amino na prstenu u 7-bočnom lancu, njegova farmaceutski prihvatljiva sol, ili njegov solvat u skladu sa zahtjevom 1, naznačen time da je namijenjen upotrebi za liječenje zarazne bolesti.
HRP20161408TT 2008-10-31 2016-10-27 Cefalosporin koji sadrži katehol skupinu HRP20161408T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2008280828 2008-10-31
EP15175084.1A EP2960244B1 (en) 2008-10-31 2009-10-27 Cephalosporin having catechol group

Publications (1)

Publication Number Publication Date
HRP20161408T1 true HRP20161408T1 (hr) 2016-12-02

Family

ID=42128829

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20161408TT HRP20161408T1 (hr) 2008-10-31 2016-10-27 Cefalosporin koji sadrži katehol skupinu

Country Status (38)

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US (1) US9238657B2 (hr)
EP (2) EP2960244B1 (hr)
JP (2) JP5498393B2 (hr)
KR (1) KR101655961B1 (hr)
CN (1) CN102203100B (hr)
AU (1) AU2009310959B2 (hr)
BR (1) BRPI0921701B8 (hr)
CA (1) CA2736953C (hr)
CL (1) CL2011000939A1 (hr)
CO (1) CO6331443A2 (hr)
CR (1) CR20110144A (hr)
CY (2) CY1118536T1 (hr)
DK (1) DK2960244T3 (hr)
EA (1) EA019520B1 (hr)
ES (2) ES2602969T3 (hr)
FI (1) FIC20200039I1 (hr)
FR (1) FR20C1050I2 (hr)
HR (1) HRP20161408T1 (hr)
HU (2) HUE031802T2 (hr)
IL (1) IL211720A (hr)
LT (2) LT2960244T (hr)
MA (1) MA32731B1 (hr)
ME (1) ME02666B (hr)
MX (1) MX2011004636A (hr)
MY (1) MY155655A (hr)
NL (1) NL301067I2 (hr)
NO (1) NO2020035I1 (hr)
NZ (1) NZ591728A (hr)
PE (1) PE20120010A1 (hr)
PL (1) PL2960244T3 (hr)
PT (1) PT2960244T (hr)
RS (1) RS55365B1 (hr)
SI (1) SI2960244T1 (hr)
SM (1) SMT201600397B (hr)
TW (1) TWI535727B (hr)
UA (1) UA105190C2 (hr)
WO (1) WO2010050468A1 (hr)
ZA (1) ZA201102024B (hr)

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UA105190C2 (ru) 2014-04-25
WO2010050468A1 (ja) 2010-05-06
DK2960244T3 (en) 2016-11-28
PE20120010A1 (es) 2012-02-07
CY2020034I2 (el) 2021-05-05
PL2960244T3 (pl) 2017-03-31
SI2960244T1 (sl) 2017-02-28
ZA201102024B (en) 2014-08-27
ME02666B (me) 2017-06-20
CY1118536T1 (el) 2017-07-12
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