HRP20171175T1 - Novi triciklički spojevi - Google Patents
Novi triciklički spojevi Download PDFInfo
- Publication number
- HRP20171175T1 HRP20171175T1 HRP20171175TT HRP20171175T HRP20171175T1 HR P20171175 T1 HRP20171175 T1 HR P20171175T1 HR P20171175T T HRP20171175T T HR P20171175TT HR P20171175 T HRP20171175 T HR P20171175T HR P20171175 T1 HRP20171175 T1 HR P20171175T1
- Authority
- HR
- Croatia
- Prior art keywords
- tricyclic compounds
- novel tricyclic
- pharmaceutically acceptable
- image
- following formula
- Prior art date
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- 150000001875 compounds Chemical class 0.000 title claims 5
- 150000003839 salts Chemical class 0.000 claims 2
- 239000012752 auxiliary agent Substances 0.000 claims 1
- 239000003937 drug carrier Substances 0.000 claims 1
- 239000000825 pharmaceutical preparation Substances 0.000 claims 1
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Claims (3)
1. Spoj predstavljen slijedećom formulom:
[image]
2. Farmaceutski prihvatljiva sol spoja predstavljenog slijedećom formulom:
[image]
3. Farmaceutski pripravak, naznačen time, da sadrži spoj prema zahtjevu 1 ili farmaceutski prihvatljivu sol spoja prema zahtjevu 2, te farmaceutski prihvatljiv nosač i pomoćno sredstvo.
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US26556309P | 2009-12-01 | 2009-12-01 | |
US36411610P | 2010-07-14 | 2010-07-14 | |
EP10835061.2A EP2506716B1 (en) | 2009-12-01 | 2010-12-01 | Novel tricyclic compounds |
PCT/US2010/058572 WO2011068881A1 (en) | 2009-12-01 | 2010-12-01 | Novel tricyclic compounds |
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HRP20171175T1 true HRP20171175T1 (hr) | 2017-10-06 |
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