HRP20020381A2 - ?2-adrenergic receptor agonists - Google Patents
?2-adrenergic receptor agonistsInfo
- Publication number
- HRP20020381A2 HRP20020381A2 HR20020381A HRP20020381A HRP20020381A2 HR P20020381 A2 HRP20020381 A2 HR P20020381A2 HR 20020381 A HR20020381 A HR 20020381A HR P20020381 A HRP20020381 A HR P20020381A HR P20020381 A2 HRP20020381 A2 HR P20020381A2
- Authority
- HR
- Croatia
- Prior art keywords
- substituted
- ligand
- compound
- linker
- compounds
- Prior art date
Links
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/68—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings and hydroxy groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/06—Antiabortive agents; Labour repressants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/34—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
- C07C233/42—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
- C07C233/43—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of a saturated carbon skeleton
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Biomedical Technology (AREA)
- Reproductive Health (AREA)
- Neurosurgery (AREA)
- Child & Adolescent Psychology (AREA)
- Emergency Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Vehicle Body Suspensions (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US45761899A | 1999-12-08 | 1999-12-08 | |
US09/637,899 US6576793B1 (en) | 1999-12-08 | 2000-08-14 | β2-adrenergic receptor agonists |
PCT/US2000/033057 WO2001042193A1 (fr) | 1999-12-08 | 2000-12-06 | Agonistes des recepteurs adrenergiques du beta 2 |
Publications (1)
Publication Number | Publication Date |
---|---|
HRP20020381A2 true HRP20020381A2 (en) | 2005-12-31 |
Family
ID=27038674
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HR20020381A HRP20020381A2 (en) | 1999-12-08 | 2002-04-30 | ?2-adrenergic receptor agonists |
Country Status (23)
Country | Link |
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EP (1) | EP1235787B1 (fr) |
KR (1) | KR20070039968A (fr) |
CN (1) | CN1402702A (fr) |
AT (1) | ATE253039T1 (fr) |
AU (1) | AU781466B2 (fr) |
BR (1) | BR0015962A (fr) |
CA (1) | CA2391293C (fr) |
CZ (1) | CZ20021831A3 (fr) |
DE (1) | DE60006280T2 (fr) |
DK (1) | DK1235787T3 (fr) |
EA (1) | EA004263B1 (fr) |
ES (1) | ES2208453T3 (fr) |
HR (1) | HRP20020381A2 (fr) |
HU (1) | HUP0203638A3 (fr) |
IL (1) | IL149317A0 (fr) |
IS (1) | IS2164B (fr) |
MX (1) | MXPA02005599A (fr) |
NO (1) | NO327630B1 (fr) |
OA (1) | OA11558A (fr) |
PT (1) | PT1235787E (fr) |
SK (1) | SK287036B6 (fr) |
TR (1) | TR200302010T4 (fr) |
WO (1) | WO2001042193A1 (fr) |
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EP1487417A4 (fr) | 2001-09-17 | 2010-03-17 | Glaxo Group Ltd | Formulations de medicament en poudre seche |
WO2003042160A1 (fr) * | 2001-11-13 | 2003-05-22 | Theravance, Inc. | Agonistes de recepteur d'aryl aniline beta-2 adrenergique |
TWI249515B (en) * | 2001-11-13 | 2006-02-21 | Theravance Inc | Aryl aniline beta2 adrenergic receptor agonists |
WO2003099764A1 (fr) * | 2002-05-28 | 2003-12-04 | Theravance, Inc. | Agonistes du recepteur adrenergique $g(b)2 alcoxy aryle |
TW200409746A (en) * | 2002-07-26 | 2004-06-16 | Theravance Inc | Crystalline β2 adrenergic receptor agonist |
US6844362B2 (en) | 2002-10-11 | 2005-01-18 | Pfizer Inc | Indole derivatives useful for the treatment of diseases |
DE602004024383D1 (de) | 2003-05-08 | 2010-01-14 | Theravance Inc | Kristalline formen eines arylanilin-beta-2-adrenergenrezeptor-agonists |
TW200510277A (en) | 2003-05-27 | 2005-03-16 | Theravance Inc | Crystalline form of β2-adrenergic receptor agonist |
US7067541B2 (en) | 2003-06-04 | 2006-06-27 | Pfizer Inc | 2-amino-pyridine derivatives useful for the treatment of diseases |
US7375100B2 (en) | 2003-06-04 | 2008-05-20 | Pfizer Inc | 2-amino-pyridine derivatives useful for the treatment of diseases |
GB0316290D0 (en) | 2003-07-11 | 2003-08-13 | Glaxo Group Ltd | Novel compounds |
EP1654312B1 (fr) | 2003-08-11 | 2014-01-15 | Glaxo Group Limited | Aerosol doseur pharmaceutique et procedes associes |
TW200526547A (en) | 2003-09-22 | 2005-08-16 | Theravance Inc | Amino-substituted ethylamino β2 adrenergic receptor agonists |
TW200531692A (en) | 2004-01-12 | 2005-10-01 | Theravance Inc | Aryl aniline derivatives as β2 adrenergic receptor agonists |
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CA2553293C (fr) | 2004-01-22 | 2010-12-14 | Pfizer Inc. | Derives de sulfamides pour traitements medicaux |
BRPI0508927A (pt) * | 2004-03-17 | 2007-08-14 | Pfizer | compostos úteis para o tratamento de doenças |
EP1577291A1 (fr) * | 2004-03-17 | 2005-09-21 | Pfizer Limited | Dérivés béta-2 agonistes de la phényléthanolamine |
AP2315A (en) * | 2004-03-23 | 2011-11-04 | Pfizer | Formamide derivatives useful as adrenoceptor. |
GB0425054D0 (en) * | 2004-03-23 | 2004-12-15 | Pfizer Ltd | Formamide derivatives for the treatment of diseases |
WO2005095328A1 (fr) * | 2004-04-02 | 2005-10-13 | Glaxo Group Limited | Processus chimique et nouvelle forme cristalline |
GB0411056D0 (en) | 2004-05-18 | 2004-06-23 | Novartis Ag | Organic compounds |
AR049384A1 (es) | 2004-05-24 | 2006-07-26 | Glaxo Group Ltd | Derivados de purina |
BRPI0511695A (pt) * | 2004-06-03 | 2008-01-08 | Theravance Inc | agonistas de receptor (beta)2 adrenérgico diamina |
EP1778638A1 (fr) | 2004-07-21 | 2007-05-02 | Theravance, Inc. | Agonistes des recepteurs beta2 adrenergiques derives d'ethers de diaryle |
GB0418045D0 (en) | 2004-08-12 | 2004-09-15 | Glaxo Group Ltd | Compounds |
GT200500281A (es) | 2004-10-22 | 2006-04-24 | Novartis Ag | Compuestos organicos. |
GB0424284D0 (en) | 2004-11-02 | 2004-12-01 | Novartis Ag | Organic compounds |
GB0426164D0 (en) | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
WO2006066907A1 (fr) * | 2004-12-21 | 2006-06-29 | Glaxo Group Limited | Formulations pharmaceutiques |
WO2006072599A2 (fr) | 2005-01-10 | 2006-07-13 | Glaxo Group Limited | Nouveaux composes |
AR053346A1 (es) | 2005-03-25 | 2007-05-02 | Glaxo Group Ltd | Compuesto derivado de 8h -pirido (2,3-d) pirimidin -7 ona 2,4,8- trisustituida composicion farmaceutica y uso para preparar una composicion para tratamiento y profilxis de una enfermedad mediada por la quinasa csbp/ rk/p38 |
GB0507577D0 (en) | 2005-04-14 | 2005-05-18 | Novartis Ag | Organic compounds |
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WO2007017670A1 (fr) | 2005-08-08 | 2007-02-15 | Argenta Discovery Ltd. | Dérivés bicyclo[2,2]hept-7-ylamine et leurs utilisations |
GB0516313D0 (en) | 2005-08-08 | 2005-09-14 | Argenta Discovery Ltd | Azole derivatives and their uses |
TW200738658A (en) | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
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GB0601951D0 (en) | 2006-01-31 | 2006-03-15 | Novartis Ag | Organic compounds |
TW200745084A (en) * | 2006-03-08 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
TW200745067A (en) | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
BRPI0710240A2 (pt) | 2006-04-20 | 2011-08-09 | Glaxo Group Ltd | composto, uso de um composto, método para o tratamento de um paciente humano ou animal com uma condição ou doença, composição farmacêutica, combinação, e, processo para a preparação de um composto |
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WO2009074575A2 (fr) | 2007-12-10 | 2009-06-18 | Novartis Ag | Composés organiques |
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AT322534B (de) * | 1972-03-16 | 1975-05-26 | Thomae Gmbh Dr K | Verfahren zur herstellung von neuen optisch aktiven 1-(4'-amino-3'-halogenphenyl)-2-aminoäthanolen und deren säureadditionssalzen |
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JPH10152460A (ja) * | 1996-11-21 | 1998-06-09 | Kissei Pharmaceut Co Ltd | 2−アミノ−1−(4−ヒドロキシ−2−メチルフェニル)プロパノール誘導体 |
US6362371B1 (en) * | 1998-06-08 | 2002-03-26 | Advanced Medicine, Inc. | β2- adrenergic receptor agonists |
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- 2000-12-06 KR KR1020077004447A patent/KR20070039968A/ko not_active Application Discontinuation
- 2000-12-06 EP EP00986271A patent/EP1235787B1/fr not_active Expired - Lifetime
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NO327630B1 (no) | 2009-09-07 |
ES2208453T3 (es) | 2004-06-16 |
AU2254601A (en) | 2001-06-18 |
IS6350A (is) | 2002-04-19 |
OA11558A (en) | 2004-06-03 |
DK1235787T3 (da) | 2004-03-08 |
DE60006280D1 (de) | 2003-12-04 |
PT1235787E (pt) | 2004-03-31 |
HUP0203638A3 (en) | 2003-04-28 |
IS2164B (is) | 2006-11-15 |
EP1235787B1 (fr) | 2003-10-29 |
WO2001042193A1 (fr) | 2001-06-14 |
EA200200647A1 (ru) | 2002-12-26 |
NO20022655L (no) | 2002-06-05 |
MXPA02005599A (es) | 2002-09-18 |
NO20022655D0 (no) | 2002-06-05 |
IL149317A0 (en) | 2002-11-10 |
SK287036B6 (sk) | 2009-10-07 |
EA004263B1 (ru) | 2004-02-26 |
TR200302010T4 (tr) | 2004-01-21 |
CZ20021831A3 (cs) | 2002-11-13 |
ATE253039T1 (de) | 2003-11-15 |
EP1235787A1 (fr) | 2002-09-04 |
CA2391293A1 (fr) | 2001-06-14 |
SK9922002A3 (en) | 2002-11-06 |
CA2391293C (fr) | 2008-12-30 |
CN1402702A (zh) | 2003-03-12 |
AU781466B2 (en) | 2005-05-26 |
HUP0203638A2 (hu) | 2003-02-28 |
BR0015962A (pt) | 2002-07-30 |
DE60006280T2 (de) | 2004-07-29 |
KR20070039968A (ko) | 2007-04-13 |
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