HRP20020381A2 - ?2-adrenergic receptor agonists - Google Patents

?2-adrenergic receptor agonists

Info

Publication number
HRP20020381A2
HRP20020381A2 HR20020381A HRP20020381A HRP20020381A2 HR P20020381 A2 HRP20020381 A2 HR P20020381A2 HR 20020381 A HR20020381 A HR 20020381A HR P20020381 A HRP20020381 A HR P20020381A HR P20020381 A2 HRP20020381 A2 HR P20020381A2
Authority
HR
Croatia
Prior art keywords
substituted
ligand
compound
linker
compounds
Prior art date
Application number
HR20020381A
Other languages
English (en)
Croatian (hr)
Inventor
Edmound
Choi Seok-Ki
Original Assignee
Theravance
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/637,899 external-priority patent/US6576793B1/en
Application filed by Theravance filed Critical Theravance
Publication of HRP20020381A2 publication Critical patent/HRP20020381A2/hr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/68Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings and hydroxy groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/06Antiabortive agents; Labour repressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00Carboxylic acid amides
    • C07C233/01Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/34Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups
    • C07C233/42Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring
    • C07C233/43Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by amino groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by a carbon atom of a six-membered aromatic ring having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of a saturated carbon skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biomedical Technology (AREA)
  • Reproductive Health (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Vehicle Body Suspensions (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
HR20020381A 1999-12-08 2002-04-30 ?2-adrenergic receptor agonists HRP20020381A2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US45761899A 1999-12-08 1999-12-08
US09/637,899 US6576793B1 (en) 1999-12-08 2000-08-14 β2-adrenergic receptor agonists
PCT/US2000/033057 WO2001042193A1 (fr) 1999-12-08 2000-12-06 Agonistes des recepteurs adrenergiques du beta 2

Publications (1)

Publication Number Publication Date
HRP20020381A2 true HRP20020381A2 (en) 2005-12-31

Family

ID=27038674

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20020381A HRP20020381A2 (en) 1999-12-08 2002-04-30 ?2-adrenergic receptor agonists

Country Status (23)

Country Link
EP (1) EP1235787B1 (fr)
KR (1) KR20070039968A (fr)
CN (1) CN1402702A (fr)
AT (1) ATE253039T1 (fr)
AU (1) AU781466B2 (fr)
BR (1) BR0015962A (fr)
CA (1) CA2391293C (fr)
CZ (1) CZ20021831A3 (fr)
DE (1) DE60006280T2 (fr)
DK (1) DK1235787T3 (fr)
EA (1) EA004263B1 (fr)
ES (1) ES2208453T3 (fr)
HR (1) HRP20020381A2 (fr)
HU (1) HUP0203638A3 (fr)
IL (1) IL149317A0 (fr)
IS (1) IS2164B (fr)
MX (1) MXPA02005599A (fr)
NO (1) NO327630B1 (fr)
OA (1) OA11558A (fr)
PT (1) PT1235787E (fr)
SK (1) SK287036B6 (fr)
TR (1) TR200302010T4 (fr)
WO (1) WO2001042193A1 (fr)

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HUP0203638A3 (en) 2003-04-28
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EP1235787B1 (fr) 2003-10-29
WO2001042193A1 (fr) 2001-06-14
EA200200647A1 (ru) 2002-12-26
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IL149317A0 (en) 2002-11-10
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EA004263B1 (ru) 2004-02-26
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CZ20021831A3 (cs) 2002-11-13
ATE253039T1 (de) 2003-11-15
EP1235787A1 (fr) 2002-09-04
CA2391293A1 (fr) 2001-06-14
SK9922002A3 (en) 2002-11-06
CA2391293C (fr) 2008-12-30
CN1402702A (zh) 2003-03-12
AU781466B2 (en) 2005-05-26
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