HK1211032A1 - Solid forms of a selective cdk4/6 inhibitor cdk4/6 - Google Patents

Solid forms of a selective cdk4/6 inhibitor cdk4/6

Info

Publication number
HK1211032A1
HK1211032A1 HK15111953.5A HK15111953A HK1211032A1 HK 1211032 A1 HK1211032 A1 HK 1211032A1 HK 15111953 A HK15111953 A HK 15111953A HK 1211032 A1 HK1211032 A1 HK 1211032A1
Authority
HK
Hong Kong
Prior art keywords
cdk4
inhibitor
solid forms
selective
selective cdk4
Prior art date
Application number
HK15111953.5A
Other languages
English (en)
Chinese (zh)
Inventor
．柴卡爾
．伊德
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50151343&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1211032(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of HK1211032A1 publication Critical patent/HK1211032A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HK15111953.5A 2013-02-21 2015-12-03 Solid forms of a selective cdk4/6 inhibitor cdk4/6 HK1211032A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361767761P 2013-02-21 2013-02-21
PCT/IB2014/058865 WO2014128588A1 (en) 2013-02-21 2014-02-08 Solid forms of a selective cdk4/6 inhibitor

Publications (1)

Publication Number Publication Date
HK1211032A1 true HK1211032A1 (en) 2016-05-13

Family

ID=50151343

Family Applications (2)

Application Number Title Priority Date Filing Date
HK18107562.3A HK1248217A1 (zh) 2013-02-21 2015-12-03 選擇性cdk4/6抑制劑的固態形式
HK15111953.5A HK1211032A1 (en) 2013-02-21 2015-12-03 Solid forms of a selective cdk4/6 inhibitor cdk4/6

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HK18107562.3A HK1248217A1 (zh) 2013-02-21 2015-12-03 選擇性cdk4/6抑制劑的固態形式

Country Status (24)

Country Link
US (2) US20160002223A1 (sl)
EP (2) EP2958916B1 (sl)
JP (3) JP6381016B2 (sl)
KR (2) KR101858913B1 (sl)
CN (3) CN107759594A (sl)
AR (1) AR094842A1 (sl)
AU (1) AU2014220354B2 (sl)
BR (1) BR112015019508A8 (sl)
CA (1) CA2900322C (sl)
CY (2) CY1120734T1 (sl)
DK (2) DK3431475T3 (sl)
ES (2) ES2869277T3 (sl)
HK (2) HK1248217A1 (sl)
HU (2) HUE054212T2 (sl)
IL (1) IL240277B (sl)
MX (2) MX363715B (sl)
PL (2) PL3431475T3 (sl)
PT (2) PT2958916T (sl)
RU (1) RU2619944C2 (sl)
SG (1) SG11201505680RA (sl)
SI (2) SI2958916T1 (sl)
TR (1) TR201816077T4 (sl)
TW (2) TWI633103B (sl)
WO (1) WO2014128588A1 (sl)

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