HK1206592A1 - Therapeutic compositions comprising rilpivirin hcl and tenofovir disoproxil fumarate - Google Patents

Therapeutic compositions comprising rilpivirin hcl and tenofovir disoproxil fumarate

Info

Publication number
HK1206592A1
HK1206592A1 HK15106347.0A HK15106347A HK1206592A1 HK 1206592 A1 HK1206592 A1 HK 1206592A1 HK 15106347 A HK15106347 A HK 15106347A HK 1206592 A1 HK1206592 A1 HK 1206592A1
Authority
HK
Hong Kong
Prior art keywords
rilpivirin
hcl
therapeutic compositions
tenofovir disoproxil
disoproxil fumarate
Prior art date
Application number
HK15106347.0A
Other languages
English (en)
Chinese (zh)
Inventor
Reza Oliyai
Lauren Wiser
Mark Menning
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45094284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1206592(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of HK1206592A1 publication Critical patent/HK1206592A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/675Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK15106347.0A 2010-11-19 2014-03-21 Therapeutic compositions comprising rilpivirin hcl and tenofovir disoproxil fumarate HK1206592A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US41560010P 2010-11-19 2010-11-19

Publications (1)

Publication Number Publication Date
HK1206592A1 true HK1206592A1 (en) 2016-01-15

Family

ID=45094284

Family Applications (2)

Application Number Title Priority Date Filing Date
HK15106347.0A HK1206592A1 (en) 2010-11-19 2014-03-21 Therapeutic compositions comprising rilpivirin hcl and tenofovir disoproxil fumarate
HK14102832.2A HK1190064A1 (en) 2010-11-19 2014-03-21 Therapeutic compositions comprising rilpivirin hcl and tenovofir disoproxil fumarate

Family Applications After (1)

Application Number Title Priority Date Filing Date
HK14102832.2A HK1190064A1 (en) 2010-11-19 2014-03-21 Therapeutic compositions comprising rilpivirin hcl and tenovofir disoproxil fumarate

Country Status (35)

Country Link
US (1) US10857102B2 (ru)
EP (2) EP2826466A1 (ru)
JP (2) JP2014500261A (ru)
KR (1) KR101923103B1 (ru)
CN (2) CN106511357A (ru)
AP (1) AP3816A (ru)
AR (2) AR084500A1 (ru)
AU (3) AU2011329642B2 (ru)
BR (1) BR112013012245B1 (ru)
CA (1) CA2818097C (ru)
CL (1) CL2013001402A1 (ru)
CO (1) CO6761300A2 (ru)
CR (1) CR20130293A (ru)
DK (1) DK2640362T4 (ru)
EA (2) EA201691695A1 (ru)
EC (2) ECSP13012700A (ru)
ES (1) ES2524408T5 (ru)
HK (2) HK1206592A1 (ru)
HR (1) HRP20140946T1 (ru)
IL (1) IL226300B (ru)
MA (1) MA34735B1 (ru)
ME (1) ME01980B (ru)
MX (1) MX347512B (ru)
MY (1) MY185604A (ru)
NZ (1) NZ610729A (ru)
PE (3) PE20211657A1 (ru)
PL (1) PL2640362T5 (ru)
PT (1) PT2640362E (ru)
RS (1) RS53691B1 (ru)
SG (3) SG10201509521WA (ru)
SM (1) SMT201400150B (ru)
TW (1) TWI556840B (ru)
UA (1) UA114075C2 (ru)
WO (1) WO2012068535A1 (ru)
ZA (1) ZA201304481B (ru)

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TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
TWI556840B (zh) 2010-11-19 2016-11-11 吉李德科學股份有限公司 治療用組成物
RS55353B2 (sr) 2011-08-16 2023-11-30 Gilead Sciences Inc Tenofovir alafenamid hemifumarat
CA2779052A1 (en) * 2012-05-31 2013-11-30 Pharmascience Inc. Pharmaceutical composition of entecavir and process of manufacturing
DK3067358T3 (da) 2012-12-21 2019-11-04 Gilead Sciences Inc Polycykliske carbamoylpyridon-forbindelser og deres farmaceutiske anvendelse
WO2015014737A1 (en) * 2013-07-29 2015-02-05 Sanovel Ilac Sanayi Ve Ticaret A.S. Multilayer tablet formulations comprising tenofovir and entecavir
CZ2013985A3 (cs) * 2013-12-09 2015-06-17 Zentiva, K.S. Stabilní farmaceutická kompozice obsahující tenofovir disoproxil fumarát
WO2015152433A1 (en) * 2014-03-31 2015-10-08 Hanmi Pharm. Co., Ltd. Amorphous solid dispersion comprising paclitaxel, tablet comprising the same, and method for preparing the same
KR20170123308A (ko) 2014-12-26 2017-11-07 에모리 유니버시티 N4-하이드록시시티딘, 이와 관련된 유도체 및 이의 항 바이러스적 용도
US9839212B2 (en) 2015-04-16 2017-12-12 Bio-Lab, Inc. Multicomponent and multilayer compacted tablets
KR20170003063A (ko) * 2015-06-30 2017-01-09 한미약품 주식회사 테노포비어 디소프록실 함유 경구용 고형제제 및 그 제조방법
CA2921336A1 (en) * 2015-06-30 2016-12-30 Gilead Sciences, Inc. Pharmaceutical formulations
CN113546052A (zh) 2015-11-09 2021-10-26 吉利德科学公司 治疗人免疫缺陷病毒的治疗组合物
US20190060325A1 (en) * 2016-04-08 2019-02-28 Shionogi & Co., Ltd. Stabilized solid dosage form
TR201617448A2 (tr) * 2016-11-29 2018-06-21 Arven Ilac Sanayi Ve Ticaret Anonim Sirketi Tenofovi̇r ve emtri̇si̇tabi̇n i̇çeren kati oral farmasöti̇k bi̇leşi̇mler
US10561614B2 (en) * 2017-01-27 2020-02-18 Steerlife India Private Limited Tenofovir granules
EP3645003A4 (en) * 2017-06-30 2021-03-10 VIIV Healthcare Company COMBINATION AND USES AND TREATMENTS THEREOF
BR122022008466B1 (pt) 2017-12-07 2023-12-05 Emory University Uso de um composto
US20210000823A1 (en) * 2019-07-03 2021-01-07 Janssen Sciences Ireland Unlimited Company Methods of treating hiv
CN112137981A (zh) * 2020-11-02 2020-12-29 成都晶富医药科技有限公司 富马酸丙酚替诺福韦片及其制备工艺

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MY169670A (en) 2003-09-03 2019-05-08 Tibotec Pharm Ltd Combinations of a pyrimidine containing nnrti with rt inhibitors
JO3429B1 (ar) 2001-08-13 2019-10-20 Janssen Pharmaceutica Nv مشتقات برميدينات مثبطة فيروس الايدز
EP1448170A4 (en) 2001-11-27 2010-05-12 Bristol Myers Squibb Co EFAVIRENZ STAMP PREPARATIONS HAVING UNIQUE BIOPHARMACEUTICAL CHARACTERISTICS
DE602004014470D1 (de) 2003-01-14 2008-07-31 Gilead Sciences Inc Zusammensetzungen und verfahren zur antiviralen kombinationstherapie
KR101284361B1 (ko) 2004-09-02 2013-07-15 얀센 파마슈티카 엔.브이. 4-((4-((4-(2-시아노에텐일)-2,6-디메틸페닐)아미노-2-피리미딘일)아미노)벤조니트릴의 하이드로클로라이드
JP4912309B2 (ja) 2004-09-02 2012-04-11 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 4−[[4−[[4−(2−シアノエテニル)−2,6−ジメチルフェニル]アミノ]−2−ピリミジニル]アミノ]ベンゾニトリルの塩酸塩
TWI375560B (en) 2005-06-13 2012-11-01 Gilead Sciences Inc Composition comprising dry granulated emtricitabine and tenofovir df and method for making the same
TWI471145B (zh) 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
JP2009511191A (ja) 2005-10-14 2009-03-19 マイクロドース・テクノロジーズ・インコーポレーテッド 経口投与剤組合せ型医薬パッケージ法
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WO2009106960A2 (en) 2008-02-27 2009-09-03 Aurobindo Pharma Limited Stable compositions of lamivudine, tenofovir and efavirenz
PL2296633T3 (pl) 2008-05-02 2016-03-31 Gilead Sciences Inc Zastosowanie cząsteczek stałych nośników dla udoskonalenia przetwarzalności środka farmaceutycznego
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TWI556840B (zh) 2010-11-19 2016-11-11 吉李德科學股份有限公司 治療用組成物

Also Published As

Publication number Publication date
AU2018202635A1 (en) 2018-05-10
TW201238612A (en) 2012-10-01
KR20140037799A (ko) 2014-03-27
ECSP13012700A (es) 2013-08-30
SMT201400150B (it) 2015-01-15
AP2013006931A0 (en) 2013-06-30
AU2016208417A1 (en) 2016-08-18
CL2013001402A1 (es) 2013-12-27
EP2826466A1 (en) 2015-01-21
PL2640362T3 (pl) 2015-03-31
AP3816A (en) 2016-09-30
MX347512B (es) 2017-04-28
EP2640362B2 (en) 2021-12-01
SG10201509521WA (en) 2015-12-30
CN103491948B (zh) 2016-11-02
KR101923103B1 (ko) 2018-11-28
PE20211657A1 (es) 2021-08-24
EP2640362A1 (en) 2013-09-25
ES2524408T3 (es) 2014-12-09
WO2012068535A1 (en) 2012-05-24
AU2011329642B2 (en) 2016-08-11
CN106511357A (zh) 2017-03-22
MY185604A (en) 2021-05-25
EP2640362B1 (en) 2014-09-10
DK2640362T3 (en) 2014-12-01
PE20140163A1 (es) 2014-02-08
MA34735B1 (fr) 2013-12-03
HK1190064A1 (en) 2014-06-27
BR112013012245A2 (pt) 2016-08-09
BR112013012245B1 (pt) 2022-09-27
CA2818097C (en) 2019-07-30
US20130243857A1 (en) 2013-09-19
SG10201912527XA (en) 2020-02-27
AR123409A2 (es) 2022-11-30
PL2640362T5 (pl) 2022-05-02
ES2524408T5 (es) 2022-04-25
CN103491948A (zh) 2014-01-01
JP2014500261A (ja) 2014-01-09
IL226300B (en) 2019-05-30
CR20130293A (es) 2013-10-03
CO6761300A2 (es) 2013-09-30
AR084500A1 (es) 2013-05-22
HRP20140946T1 (hr) 2015-02-13
AU2016208417B2 (en) 2018-04-05
JP2015131853A (ja) 2015-07-23
ZA201304481B (en) 2022-03-30
EA201691695A1 (ru) 2017-11-30
EA025852B1 (ru) 2017-02-28
PE20170521A1 (es) 2017-05-27
RS53691B1 (en) 2015-04-30
AU2011329642A1 (en) 2013-05-02
US10857102B2 (en) 2020-12-08
UA114075C2 (xx) 2017-04-25
MX2013005669A (es) 2013-11-04
DK2640362T4 (da) 2022-03-07
ECSP19078196A (es) 2019-11-30
JP6138851B2 (ja) 2017-05-31
ME01980B (me) 2015-05-20
TWI556840B (zh) 2016-11-11
NZ610729A (en) 2015-10-30
CA2818097A1 (en) 2012-05-24
PT2640362E (pt) 2014-11-28
SG190333A1 (en) 2013-06-28
EA201390651A1 (ru) 2013-11-29

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