HK1200438A1 - Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors - Google Patents

Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors

Info

Publication number
HK1200438A1
HK1200438A1 HK15100806.7A HK15100806A HK1200438A1 HK 1200438 A1 HK1200438 A1 HK 1200438A1 HK 15100806 A HK15100806 A HK 15100806A HK 1200438 A1 HK1200438 A1 HK 1200438A1
Authority
HK
Hong Kong
Prior art keywords
phenyl substituted
reuptake inhibitors
monoamine reuptake
substituted cycloalkylamines
cycloalkylamines
Prior art date
Application number
HK15100806.7A
Other languages
English (en)
Chinese (zh)
Inventor
邵黎明
王鳳江
．瑪爾科姆
．赫維特
馬建國
．萊布
．瓦尼
．坎貝爾
．恩格爾
．哈迪
．科克
．施雷伯
．斯皮爾
Original Assignee
Sunovion Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sunovion Pharmaceuticals Inc filed Critical Sunovion Pharmaceuticals Inc
Publication of HK1200438A1 publication Critical patent/HK1200438A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/42—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having amino groups or hydroxy groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/52—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups or amino groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/76—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings and etherified hydroxy groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK15100806.7A 2007-05-31 2015-01-23 Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors HK1200438A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US94124207P 2007-05-31 2007-05-31

Publications (1)

Publication Number Publication Date
HK1200438A1 true HK1200438A1 (en) 2015-08-07

Family

ID=40094167

Family Applications (1)

Application Number Title Priority Date Filing Date
HK15100806.7A HK1200438A1 (en) 2007-05-31 2015-01-23 Phenyl substituted cycloalkylamines as monoamine reuptake inhibitors

Country Status (15)

Country Link
US (3) US8669291B2 (hu)
EP (3) EP2617704B1 (hu)
JP (3) JP5420534B2 (hu)
KR (1) KR101581289B1 (hu)
CN (3) CN101686672A (hu)
AU (1) AU2008259841B2 (hu)
BR (1) BRPI0811639A2 (hu)
CA (1) CA2688493C (hu)
HK (1) HK1200438A1 (hu)
IL (1) IL202405A (hu)
MX (1) MX2009012685A (hu)
NZ (1) NZ580429A (hu)
RU (1) RU2470011C2 (hu)
WO (1) WO2008151156A1 (hu)
ZA (1) ZA200907171B (hu)

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US20230212144A1 (en) 2020-05-29 2023-07-06 Daegu-Gyeongbuk Medical Innovation Foundation 5-membered heteroaryl derivative containing at least one n, and pharmaceutical composition for preventing or treating mental disorders, containing same as active ingredient
JP2023528545A (ja) 2020-05-29 2023-07-04 テグ－キョンプク メディカル イノベーション ファウンデーション スルホンアミド誘導体およびそれを有効成分とする精神病の予防または治療に使用するための医薬組成物

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IL202405A (en) 2014-05-28
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