HK1199643A1 - Oxazolidin- 2 -one compounds and uses thereof as pi3ks inhibitors -2--3- - Google Patents
Oxazolidin- 2 -one compounds and uses thereof as pi3ks inhibitors -2--3-Info
- Publication number
- HK1199643A1 HK1199643A1 HK15100012.7A HK15100012A HK1199643A1 HK 1199643 A1 HK1199643 A1 HK 1199643A1 HK 15100012 A HK15100012 A HK 15100012A HK 1199643 A1 HK1199643 A1 HK 1199643A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- oxazolidin
- compounds
- pi3ks
- inhibitors
- pi3ks inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261602954P | 2012-02-24 | 2012-02-24 | |
US201261736707P | 2012-12-13 | 2012-12-13 | |
PCT/IB2013/051443 WO2013124826A1 (en) | 2012-02-24 | 2013-02-22 | Oxazolidin- 2 -one compounds and uses thereof as pi3ks inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1199643A1 true HK1199643A1 (en) | 2015-07-10 |
Family
ID=48142031
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK15100012.7A HK1199643A1 (en) | 2012-02-24 | 2015-01-02 | Oxazolidin- 2 -one compounds and uses thereof as pi3ks inhibitors -2--3- |
Country Status (31)
Country | Link |
---|---|
US (2) | US8865894B2 (ja) |
EP (1) | EP2817307B1 (ja) |
JP (1) | JP6154404B2 (ja) |
KR (1) | KR101640698B1 (ja) |
CN (1) | CN104144926B (ja) |
AP (1) | AP2014007835A0 (ja) |
AR (1) | AR090121A1 (ja) |
AU (1) | AU2013223713C1 (ja) |
BR (1) | BR112014020672B1 (ja) |
CA (1) | CA2865372A1 (ja) |
CO (1) | CO7051028A2 (ja) |
CR (1) | CR20140397A (ja) |
DO (1) | DOP2014000194A (ja) |
EA (1) | EA026031B1 (ja) |
ES (1) | ES2598118T3 (ja) |
GE (1) | GEP20156389B (ja) |
GT (1) | GT201400178A (ja) |
HK (1) | HK1199643A1 (ja) |
IL (1) | IL233936A (ja) |
MX (1) | MX353341B (ja) |
NI (1) | NI201400089A (ja) |
NZ (1) | NZ629198A (ja) |
PE (1) | PE20142456A1 (ja) |
PH (1) | PH12014501900A1 (ja) |
PL (1) | PL2817307T3 (ja) |
PT (1) | PT2817307T (ja) |
SG (1) | SG11201404794XA (ja) |
TW (1) | TW201339155A (ja) |
UY (1) | UY34632A (ja) |
WO (1) | WO2013124826A1 (ja) |
ZA (1) | ZA201405446B (ja) |
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US20150259420A1 (en) | 2014-03-14 | 2015-09-17 | Novartis Ag | Antibody molecules to lag-3 and uses thereof |
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