HK118196A - (1H-azol-1-ylmethyl)substituted quinoline quinazoline of quinoxaline derivatives - Google Patents

(1H-azol-1-ylmethyl)substituted quinoline quinazoline of quinoxaline derivatives

Info

Publication number
HK118196A
HK118196A HK118196A HK118196A HK118196A HK 118196 A HK118196 A HK 118196A HK 118196 A HK118196 A HK 118196A HK 118196 A HK118196 A HK 118196A HK 118196 A HK118196 A HK 118196A
Authority
HK
Hong Kong
Prior art keywords
azol
ylmethyl
chem
compounds
quinoxaline derivatives
Prior art date
Application number
HK118196A
Other languages
English (en)
Inventor
Eddy Jean Edgard Freyne
Marc Gaston Venet
Alfons Herman Marg Raeymaekers
Gerard Charles Sanz
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB888827822A external-priority patent/GB8827822D0/en
Priority claimed from GB888827821A external-priority patent/GB8827821D0/en
Priority claimed from GB888827820A external-priority patent/GB8827820D0/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK118196A publication Critical patent/HK118196A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Quinoline Compounds (AREA)
  • Developing Agents For Electrophotography (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
HK118196A 1988-11-29 1996-07-04 (1H-azol-1-ylmethyl)substituted quinoline quinazoline of quinoxaline derivatives HK118196A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB888827822A GB8827822D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives
GB888827821A GB8827821D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives
GB888827820A GB8827820D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives

Publications (1)

Publication Number Publication Date
HK118196A true HK118196A (en) 1996-07-12

Family

ID=27264207

Family Applications (1)

Application Number Title Priority Date Filing Date
HK118196A HK118196A (en) 1988-11-29 1996-07-04 (1H-azol-1-ylmethyl)substituted quinoline quinazoline of quinoxaline derivatives

Country Status (22)

Country Link
EP (1) EP0371564B1 (pt)
JP (1) JP2916181B2 (pt)
CN (3) CN1033752C (pt)
AT (1) ATE124941T1 (pt)
AU (1) AU620946B2 (pt)
CA (1) CA2002864C (pt)
CY (1) CY1920A (pt)
DE (1) DE68923430T2 (pt)
DK (1) DK172748B1 (pt)
ES (1) ES2088889T3 (pt)
FI (1) FI101964B1 (pt)
GR (1) GR3017351T3 (pt)
HK (1) HK118196A (pt)
HU (2) HU205106B (pt)
IE (1) IE67803B1 (pt)
IL (1) IL92486A (pt)
MY (1) MY105871A (pt)
NO (1) NO174509B (pt)
NZ (1) NZ231441A (pt)
PT (1) PT92448B (pt)
RU (1) RU1780536C (pt)
ZW (1) ZW15889A1 (pt)

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KR101159118B1 (ko) * 2003-12-05 2012-06-22 얀센 파마슈티카 엔.브이. 폴리(adp-리보스)폴리머라제 저해제로서의 6-치환된2-퀴놀리논 및 2-퀴녹살리논
CN1890225A (zh) * 2003-12-10 2007-01-03 詹森药业有限公司 作为多聚(adp-核糖)聚合酶抑制剂的被取代的6-环己基烷基取代的2-喹啉酮和2-喹喔啉酮
CN1980913B (zh) 2004-06-30 2011-12-14 詹森药业有限公司 作为parp抑制剂的喹唑啉二酮衍生物
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Also Published As

Publication number Publication date
RU1780536C (ru) 1992-12-07
NO174509C (pt) 1994-05-18
PT92448A (pt) 1990-05-31
DE68923430T2 (de) 1996-02-15
GR3017351T3 (en) 1995-12-31
HUT52498A (en) 1990-07-28
FI895687A0 (fi) 1989-11-28
ATE124941T1 (de) 1995-07-15
FI101964B (fi) 1998-09-30
CN1036003C (zh) 1997-10-01
DK172748B1 (da) 1999-06-28
DK599489A (da) 1990-05-30
CN1036002C (zh) 1997-10-01
IE893782L (en) 1990-05-29
HU205106B (en) 1992-03-30
MY105871A (en) 1995-02-28
DE68923430D1 (de) 1995-08-17
DK599489D0 (da) 1989-11-28
EP0371564A3 (en) 1991-05-29
NZ231441A (en) 1991-05-28
EP0371564B1 (en) 1995-07-12
HU211686A9 (en) 1995-12-28
ES2088889T3 (es) 1996-10-01
JP2916181B2 (ja) 1999-07-05
EP0371564A2 (en) 1990-06-06
NO894734D0 (no) 1989-11-28
IL92486A0 (en) 1990-08-31
FI101964B1 (fi) 1998-09-30
CN1106004A (zh) 1995-08-02
AU620946B2 (en) 1992-02-27
CN1033752C (zh) 1997-01-08
HU896220D0 (en) 1990-02-28
IE67803B1 (en) 1996-05-01
CA2002864A1 (en) 1990-05-29
NO174509B (no) 1994-02-07
NO894734L (no) 1990-05-30
CN1042912A (zh) 1990-06-13
CN1106005A (zh) 1995-08-02
PT92448B (pt) 1995-07-18
AU4564689A (en) 1990-06-07
CY1920A (en) 1997-03-07
JPH02223579A (ja) 1990-09-05
ZW15889A1 (en) 1991-07-17
IL92486A (en) 1993-07-08
CA2002864C (en) 1999-11-16

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PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20061128