ATE124941T1 - (1h-azol-1-ylmethyl)substituierte quinolin-, quinazolin- oder quinoxalin-derivate. - Google Patents

(1h-azol-1-ylmethyl)substituierte quinolin-, quinazolin- oder quinoxalin-derivate.

Info

Publication number
ATE124941T1
ATE124941T1 AT89203014T AT89203014T ATE124941T1 AT E124941 T1 ATE124941 T1 AT E124941T1 AT 89203014 T AT89203014 T AT 89203014T AT 89203014 T AT89203014 T AT 89203014T AT E124941 T1 ATE124941 T1 AT E124941T1
Authority
AT
Austria
Prior art keywords
quinazoline
ylmethyl
chem
compounds
quinoxaline derivatives
Prior art date
Application number
AT89203014T
Other languages
English (en)
Inventor
Eddy Jean Edgard Freyne
Marc Gaston Venet
Alfons Herman Marg Raeymaekers
Gerard Charles Sanz
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB888827820A external-priority patent/GB8827820D0/en
Priority claimed from GB888827822A external-priority patent/GB8827822D0/en
Priority claimed from GB888827821A external-priority patent/GB8827821D0/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of ATE124941T1 publication Critical patent/ATE124941T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Quinoline Compounds (AREA)
  • Developing Agents For Electrophotography (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AT89203014T 1988-11-29 1989-11-28 (1h-azol-1-ylmethyl)substituierte quinolin-, quinazolin- oder quinoxalin-derivate. ATE124941T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB888827820A GB8827820D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives
GB888827822A GB8827822D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives
GB888827821A GB8827821D0 (en) 1988-11-29 1988-11-29 (1h-azol-1-ylmethyl)substituted quinoline derivatives

Publications (1)

Publication Number Publication Date
ATE124941T1 true ATE124941T1 (de) 1995-07-15

Family

ID=27264207

Family Applications (1)

Application Number Title Priority Date Filing Date
AT89203014T ATE124941T1 (de) 1988-11-29 1989-11-28 (1h-azol-1-ylmethyl)substituierte quinolin-, quinazolin- oder quinoxalin-derivate.

Country Status (22)

Country Link
EP (1) EP0371564B1 (de)
JP (1) JP2916181B2 (de)
CN (3) CN1033752C (de)
AT (1) ATE124941T1 (de)
AU (1) AU620946B2 (de)
CA (1) CA2002864C (de)
CY (1) CY1920A (de)
DE (1) DE68923430T2 (de)
DK (1) DK172748B1 (de)
ES (1) ES2088889T3 (de)
FI (1) FI101964B1 (de)
GR (1) GR3017351T3 (de)
HK (1) HK118196A (de)
HU (2) HU205106B (de)
IE (1) IE67803B1 (de)
IL (1) IL92486A (de)
MY (1) MY105871A (de)
NO (1) NO174509B (de)
NZ (1) NZ231441A (de)
PT (1) PT92448B (de)
RU (1) RU1780536C (de)
ZW (1) ZW15889A1 (de)

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AU2001293835A1 (en) 2000-09-25 2002-04-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives
AU2001293829A1 (en) 2000-09-25 2002-04-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting 6-((substituted phenyl)methyl)-quinoline and quinazoline derivatives
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Also Published As

Publication number Publication date
DE68923430T2 (de) 1996-02-15
CN1033752C (zh) 1997-01-08
CY1920A (en) 1997-03-07
ES2088889T3 (es) 1996-10-01
CN1106004A (zh) 1995-08-02
CN1042912A (zh) 1990-06-13
CN1036002C (zh) 1997-10-01
IE67803B1 (en) 1996-05-01
AU4564689A (en) 1990-06-07
NO174509C (de) 1994-05-18
CN1106005A (zh) 1995-08-02
JPH02223579A (ja) 1990-09-05
DK172748B1 (da) 1999-06-28
DK599489A (da) 1990-05-30
AU620946B2 (en) 1992-02-27
NO894734L (no) 1990-05-30
EP0371564B1 (de) 1995-07-12
MY105871A (en) 1995-02-28
HK118196A (en) 1996-07-12
FI101964B (fi) 1998-09-30
FI895687A0 (fi) 1989-11-28
DE68923430D1 (de) 1995-08-17
IL92486A (en) 1993-07-08
DK599489D0 (da) 1989-11-28
PT92448B (pt) 1995-07-18
HU205106B (en) 1992-03-30
EP0371564A3 (de) 1991-05-29
HU896220D0 (en) 1990-02-28
EP0371564A2 (de) 1990-06-06
CN1036003C (zh) 1997-10-01
NO174509B (no) 1994-02-07
IE893782L (en) 1990-05-29
CA2002864C (en) 1999-11-16
IL92486A0 (en) 1990-08-31
FI101964B1 (fi) 1998-09-30
ZW15889A1 (en) 1991-07-17
CA2002864A1 (en) 1990-05-29
GR3017351T3 (en) 1995-12-31
PT92448A (pt) 1990-05-31
NO894734D0 (no) 1989-11-28
NZ231441A (en) 1991-05-28
RU1780536C (ru) 1992-12-07
HUT52498A (en) 1990-07-28
HU211686A9 (en) 1995-12-28
JP2916181B2 (ja) 1999-07-05

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