HK1133878A1 - Inhibitors of c-fms kinase c-fms - Google Patents

Inhibitors of c-fms kinase c-fms

Info

Publication number
HK1133878A1
HK1133878A1 HK09112210.0A HK09112210A HK1133878A1 HK 1133878 A1 HK1133878 A1 HK 1133878A1 HK 09112210 A HK09112210 A HK 09112210A HK 1133878 A1 HK1133878 A1 HK 1133878A1
Authority
HK
Hong Kong
Prior art keywords
fms
inhibitors
kinase
fms kinase
Prior art date
Application number
HK09112210.0A
Other languages
English (en)
Chinese (zh)
Inventor
Carl R Illig
Shelley K Ballentine
Jinsheng Chen
Renee Louise Desjarlais
Sanath K Meegalla
Bruce E Tomczuk
Mark Wall
Kenneth Wilson
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1133878A1 publication Critical patent/HK1133878A1/xx

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    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Genetics & Genomics (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • General Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Microbiology (AREA)
  • Biotechnology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Virology (AREA)
HK09112210.0A 2006-04-20 2009-12-28 Inhibitors of c-fms kinase c-fms HK1133878A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79366706P 2006-04-20 2006-04-20
PCT/US2007/066868 WO2007124319A1 (en) 2006-04-20 2007-04-18 Inhibitors of c-fms kinase

Publications (1)

Publication Number Publication Date
HK1133878A1 true HK1133878A1 (en) 2010-04-09

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HK09112210.0A HK1133878A1 (en) 2006-04-20 2009-12-28 Inhibitors of c-fms kinase c-fms

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Country Link
US (7) US8859602B2 (ru)
EP (3) EP2016074B1 (ru)
JP (3) JP5331681B2 (ru)
KR (3) KR101367646B1 (ru)
CN (1) CN101472914B (ru)
AR (3) AR060610A1 (ru)
AU (3) AU2007240442B2 (ru)
BR (1) BRPI0710548B8 (ru)
CA (3) CA2650057C (ru)
ES (3) ES2565238T3 (ru)
HK (1) HK1133878A1 (ru)
IL (1) IL194845A (ru)
MX (3) MX2008013530A (ru)
NO (1) NO20084896L (ru)
NZ (3) NZ572070A (ru)
PE (1) PE20080074A1 (ru)
RU (1) RU2475483C2 (ru)
SG (1) SG171593A1 (ru)
TW (3) TWI411612B (ru)
UA (1) UA93085C2 (ru)
UY (1) UY30297A1 (ru)
WO (3) WO2007124321A1 (ru)
ZA (1) ZA200809873B (ru)

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US20060281788A1 (en) * 2005-06-10 2006-12-14 Baumann Christian A Synergistic modulation of flt3 kinase using a flt3 inhibitor and a farnesyl transferase inhibitor
US20090246208A1 (en) * 2006-01-05 2009-10-01 Novartis Ag Methods for preventing and treating cancer metastasis and bone loss associated with cancer metastasis
US8697716B2 (en) 2006-04-20 2014-04-15 Janssen Pharmaceutica Nv Method of inhibiting C-KIT kinase
KR101367645B1 (ko) 2006-04-20 2014-02-27 얀센 파마슈티카 엔.브이. Ｃ-ｆｍｓ 키나제의 저해제로서의 복소환식 화합물
US8859602B2 (en) * 2006-04-20 2014-10-14 Janssen Pharmaceutica Nv Inhibitors of c-fms kinase
CA2649755C (en) * 2006-04-20 2014-12-02 Janssen Pharmaceutica N.V. Method of inhibiting c-kit kinase
NZ572201A (en) * 2006-04-20 2011-09-30 Janssen Pharmaceutica Nv Inhibitors of c-fms kinase
JO3240B1 (ar) * 2007-10-17 2018-03-08 Janssen Pharmaceutica Nv c-fms مثبطات كيناز
US10106798B2 (en) 2010-01-05 2018-10-23 Institut National De La Sante Et De La Recherche Medicale (Inserm) FLT3 receptor antagonists for the treatment or the prevention of pain disorders
US9109227B2 (en) 2010-01-05 2015-08-18 Institut National De La Sante Et De La Recherche Medicale (Inserm) FLT3 receptor antagonists for the treatment or the prevention of pain disorders
EP2704713B1 (en) 2011-05-05 2017-01-18 Novartis AG Csf-1r inhibitors for treatment of brain tumors
US8940742B2 (en) * 2012-04-10 2015-01-27 Infinity Pharmaceuticals, Inc. Heterocyclic compounds and uses thereof
ES2608628T3 (es) 2012-08-07 2017-04-12 Janssen Pharmaceutica Nv Procedimiento para la preparacion de derivados de ester heterociclicos
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