HK1029979A1 - Inhibitors of alpha4 mediated cell adhesion alpha 4 - Google Patents
Inhibitors of alpha4 mediated cell adhesion alpha 4Info
- Publication number
- HK1029979A1 HK1029979A1 HK01100247A HK01100247A HK1029979A1 HK 1029979 A1 HK1029979 A1 HK 1029979A1 HK 01100247 A HK01100247 A HK 01100247A HK 01100247 A HK01100247 A HK 01100247A HK 1029979 A1 HK1029979 A1 HK 1029979A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- inhibitors
- alpha
- cell adhesion
- mediated cell
- alpha4
- Prior art date
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- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C07C233/51—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
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- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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-
1999
- 1999-01-18 MY MYPI99000210A patent/MY153569A/en unknown
- 1999-01-19 PT PT99904115T patent/PT1049662E/pt unknown
- 1999-01-19 TW TW088100776A patent/TW591007B/zh not_active IP Right Cessation
- 1999-01-19 ES ES99904115T patent/ES2264252T3/es not_active Expired - Lifetime
- 1999-01-19 AU AU24584/99A patent/AU749568B2/en not_active Ceased
- 1999-01-19 CN CNB998022381A patent/CN1301964C/zh not_active Expired - Fee Related
- 1999-01-19 SG SG200204434A patent/SG118147A1/en unknown
- 1999-01-19 NZ NZ506081A patent/NZ506081A/xx not_active IP Right Cessation
- 1999-01-19 KR KR10-2000-7006563A patent/KR100411331B1/ko not_active IP Right Cessation
- 1999-01-19 DE DE69932032T patent/DE69932032T2/de not_active Expired - Lifetime
- 1999-01-19 IL IL13738599A patent/IL137385A0/xx active IP Right Grant
- 1999-01-19 BR BRPI9907040-5A patent/BR9907040B1/pt not_active IP Right Cessation
- 1999-01-19 AT AT99904115T patent/ATE330935T1/de active
- 1999-01-19 WO PCT/US1999/000993 patent/WO1999036393A1/en active IP Right Grant
- 1999-01-19 DK DK99904115T patent/DK1049662T3/da active
- 1999-01-19 JP JP2000540111A patent/JP3634749B2/ja not_active Expired - Fee Related
- 1999-01-19 CA CA002318527A patent/CA2318527C/en not_active Expired - Fee Related
- 1999-01-19 EP EP99904115A patent/EP1049662B1/en not_active Expired - Lifetime
- 1999-01-21 AR ARP990100226A patent/AR014448A1/es active IP Right Grant
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- 2000-07-19 US US09/619,712 patent/US6521666B1/en not_active Expired - Lifetime
- 2000-07-19 IL IL137385A patent/IL137385A/en not_active IP Right Cessation
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DK1049662T3 (da) | 2006-10-23 |
ES2264252T3 (es) | 2006-12-16 |
KR100411331B1 (ko) | 2003-12-18 |
AR014448A1 (es) | 2001-02-28 |
NZ506081A (en) | 2003-02-28 |
PT1049662E (pt) | 2006-09-29 |
JP2005002116A (ja) | 2005-01-06 |
DE69932032T2 (de) | 2006-12-28 |
CY1105433T1 (el) | 2010-04-28 |
WO1999036393A1 (en) | 1999-07-22 |
MY153569A (en) | 2015-02-27 |
KR20010033180A (ko) | 2001-04-25 |
AU749568B2 (en) | 2002-06-27 |
CA2318527C (en) | 2006-10-17 |
CN1301964C (zh) | 2007-02-28 |
TW591007B (en) | 2004-06-11 |
BR9907040B1 (pt) | 2010-11-30 |
IL137385A0 (en) | 2001-07-24 |
US6855843B2 (en) | 2005-02-15 |
IL137385A (en) | 2006-08-20 |
JP3634749B2 (ja) | 2005-03-30 |
SG118147A1 (en) | 2006-01-27 |
DE69932032D1 (de) | 2006-08-03 |
AU2458499A (en) | 1999-08-02 |
JP2002509131A (ja) | 2002-03-26 |
US20030191118A1 (en) | 2003-10-09 |
CA2318527A1 (en) | 1999-07-22 |
US6521666B1 (en) | 2003-02-18 |
ATE330935T1 (de) | 2006-07-15 |
EP1049662A1 (en) | 2000-11-08 |
EP1049662B1 (en) | 2006-06-21 |
CN1288457A (zh) | 2001-03-21 |
BR9907040A (pt) | 2000-10-17 |
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