GT199700015AA - Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen ysuusofarmaceuticoymetodosyeficazproductointermedio para su preparacion. - Google Patents

Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen ysuusofarmaceuticoymetodosyeficazproductointermedio para su preparacion.

Info

Publication number
GT199700015AA
GT199700015AA GT199700015AK GT199700015K GT199700015AA GT 199700015A A GT199700015A A GT 199700015AA GT 199700015A K GT199700015A K GT 199700015AK GT 199700015 K GT199700015 K GT 199700015K GT 199700015A A GT199700015A A GT 199700015AA
Authority
GT
Guatemala
Prior art keywords
medicine
preparation
methods
pharmaceutical compositions
compositions containing
Prior art date
Application number
GT199700015AK
Other languages
English (en)
Spanish (es)
Inventor
Scott E Zook
Raymond Dagnino Jr
Michael E Deason
Steven L Bender
Michael J Melnick
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199700015AA publication Critical patent/GT199700015AA/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/04Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
GT199700015AK 1995-12-08 1997-01-29 Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen ysuusofarmaceuticoymetodosyeficazproductointermedio para su preparacion. GT199700015AA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56976695A 1995-12-08 1995-12-08

Publications (1)

Publication Number Publication Date
GT199700015AA true GT199700015AA (es) 1998-07-23

Family

ID=24276764

Family Applications (2)

Application Number Title Priority Date Filing Date
GT199700015A GT199700015A (es) 1995-12-08 1997-01-29 Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen y su uso farmaceutico y metodosyeficazproducto intermedio para su preparacion.
GT199700015AK GT199700015AA (es) 1995-12-08 1997-01-29 Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen ysuusofarmaceuticoymetodosyeficazproductointermedio para su preparacion.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
GT199700015A GT199700015A (es) 1995-12-08 1997-01-29 Inhibidores de metaloproteinasa, composiciones farmaceuticas que las contienen y su uso farmaceutico y metodosyeficazproducto intermedio para su preparacion.

Country Status (39)

Country Link
US (1) US6153757A (fr)
EP (2) EP1095936B1 (fr)
JP (1) JP2000502330A (fr)
KR (1) KR19990072009A (fr)
CN (2) CN1207289C (fr)
AP (2) AP1288A (fr)
AT (2) ATE283264T1 (fr)
AU (1) AU725831C (fr)
BG (1) BG64279B1 (fr)
BR (1) BR9611929A (fr)
CA (1) CA2238306A1 (fr)
CO (1) CO4790150A1 (fr)
CZ (1) CZ292942B6 (fr)
DE (2) DE69633947T2 (fr)
DK (1) DK0874830T3 (fr)
EA (1) EA003294B1 (fr)
ES (2) ES2233275T3 (fr)
GE (1) GEP20012388B (fr)
GT (2) GT199700015A (fr)
HR (1) HRP970031A2 (fr)
HU (1) HUP9902092A3 (fr)
ID (1) ID17624A (fr)
IL (6) IL124559A (fr)
MX (1) MX9804457A (fr)
MY (1) MY117290A (fr)
NO (1) NO311360B1 (fr)
NZ (1) NZ325559A (fr)
OA (1) OA10794A (fr)
PA (1) PA8431301A1 (fr)
PE (1) PE69298A1 (fr)
PL (1) PL327275A1 (fr)
PT (1) PT874830E (fr)
SI (1) SI0874830T1 (fr)
SK (1) SK73898A3 (fr)
SV (1) SV1997000008A (fr)
TR (1) TR199800990T2 (fr)
TW (1) TW546293B (fr)
WO (1) WO1997020824A1 (fr)
YU (1) YU21597A (fr)

Families Citing this family (114)

* Cited by examiner, † Cited by third party
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WO2002074738A2 (fr) 2001-03-15 2002-09-26 Bristol-Myers Squibb Company Derives de beta-aminoacides spirocycliques utilises comme inhibiteurs des metalloproteinases matricielles et de l'enzyme de conversion de tnf-alpha (tage)
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