FR2775596B1 - Nouvelles compositions pharmaceutiques - Google Patents

Nouvelles compositions pharmaceutiques

Info

Publication number
FR2775596B1
FR2775596B1 FR9902748A FR9902748A FR2775596B1 FR 2775596 B1 FR2775596 B1 FR 2775596B1 FR 9902748 A FR9902748 A FR 9902748A FR 9902748 A FR9902748 A FR 9902748A FR 2775596 B1 FR2775596 B1 FR 2775596B1
Authority
FR
France
Prior art keywords
pharmaceutical compositions
new pharmaceutical
new
compositions
pharmaceutical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9902748A
Other languages
English (en)
Other versions
FR2775596A1 (fr
Inventor
Michael Ambuhl
Barbara Luckel
Friedrich Richter
Barbara Haberlin
Armin Meinzer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269231&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR2775596(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9804742.6A external-priority patent/GB9804742D0/en
Priority claimed from GBGB9805104.8A external-priority patent/GB9805104D0/en
Priority claimed from GBGB9805199.8A external-priority patent/GB9805199D0/en
Application filed by Novartis AG filed Critical Novartis AG
Publication of FR2775596A1 publication Critical patent/FR2775596A1/fr
Application granted granted Critical
Publication of FR2775596B1 publication Critical patent/FR2775596B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P41/00Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
FR9902748A 1998-03-06 1999-03-04 Nouvelles compositions pharmaceutiques Expired - Fee Related FR2775596B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9804742.6A GB9804742D0 (en) 1998-03-06 1998-03-06 Organic compounds
GBGB9805104.8A GB9805104D0 (en) 1998-03-10 1998-03-10 Organic compounds
GBGB9805199.8A GB9805199D0 (en) 1998-03-11 1998-03-11 Organic compounds

Publications (2)

Publication Number Publication Date
FR2775596A1 FR2775596A1 (fr) 1999-09-10
FR2775596B1 true FR2775596B1 (fr) 2004-12-24

Family

ID=27269231

Family Applications (4)

Application Number Title Priority Date Filing Date
FR9902748A Expired - Fee Related FR2775596B1 (fr) 1998-03-06 1999-03-04 Nouvelles compositions pharmaceutiques
FR0013782A Expired - Fee Related FR2800277B1 (fr) 1998-03-06 2000-10-25 Compositions pharmaceutiques comprenant une substance active difficilement soluble et un milieu vehiculeur
FR0403163A Expired - Fee Related FR2853546B1 (fr) 1998-03-06 2004-03-26 Nouvelle composition pharmaceutique contenant la cyclosporine a
FR0600097A Withdrawn FR2881956A1 (fr) 1998-03-06 2006-01-05 Nouvelle composition pharmaceutique contenant la cycloporine a

Family Applications After (3)

Application Number Title Priority Date Filing Date
FR0013782A Expired - Fee Related FR2800277B1 (fr) 1998-03-06 2000-10-25 Compositions pharmaceutiques comprenant une substance active difficilement soluble et un milieu vehiculeur
FR0403163A Expired - Fee Related FR2853546B1 (fr) 1998-03-06 2004-03-26 Nouvelle composition pharmaceutique contenant la cyclosporine a
FR0600097A Withdrawn FR2881956A1 (fr) 1998-03-06 2006-01-05 Nouvelle composition pharmaceutique contenant la cycloporine a

Country Status (30)

Country Link
EP (2) EP1354582A3 (fr)
JP (2) JP2002505271A (fr)
KR (1) KR100443306B1 (fr)
CN (1) CN1195495C (fr)
AR (1) AR015729A1 (fr)
AT (1) ATE277599T1 (fr)
AU (1) AU749217B2 (fr)
BE (3) BE1012400A5 (fr)
BR (1) BR9908597A (fr)
CA (1) CA2322845C (fr)
CO (1) CO4930289A1 (fr)
CZ (1) CZ301967B6 (fr)
DE (2) DE19983012T1 (fr)
ES (1) ES2228014T3 (fr)
FR (4) FR2775596B1 (fr)
GB (1) GB2350791B (fr)
HK (2) HK1034038A1 (fr)
HU (1) HUP0101080A3 (fr)
ID (1) ID25908A (fr)
IL (2) IL138248A0 (fr)
IT (1) IT1313550B1 (fr)
MY (1) MY129274A (fr)
NO (1) NO331800B1 (fr)
NZ (1) NZ506644A (fr)
PE (1) PE20000324A1 (fr)
PT (1) PT1059913E (fr)
SK (1) SK285139B6 (fr)
TR (1) TR200002586T2 (fr)
TW (3) TWI236912B (fr)
WO (1) WO1999044584A1 (fr)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1236813C (zh) * 1998-12-11 2006-01-18 药品处理公司 水难溶性药物的自乳化组合物
DE69939335D1 (de) * 1998-12-30 2008-09-25 Dexcel Ltd Dispergierbares konzentrat zur verabreichung von cyclosporin
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
US6294192B1 (en) * 1999-02-26 2001-09-25 Lipocine, Inc. Triglyceride-free compositions and methods for improved delivery of hydrophobic therapeutic agents
US20070032853A1 (en) 2002-03-27 2007-02-08 Hossainy Syed F 40-O-(2-hydroxy)ethyl-rapamycin coated stent
GB2362573A (en) * 2000-05-25 2001-11-28 Cipla Ltd Cyclosporin formulation
WO2001032143A1 (fr) * 1999-11-02 2001-05-10 Cipla Ltd. Composition pharmaceutique pour administer des substances actives sur le plan pharmaceutique insolubles dans l'eau et procede de preparation afferent
AU1043201A (en) * 1999-11-02 2001-05-14 Cipla Limited Cyclosporin formulation
GB0008785D0 (en) * 2000-04-10 2000-05-31 Novartis Ag Organic compounds
DE10024451A1 (de) * 2000-05-18 2001-11-29 Asta Medica Ag Pharmazeutische Darreichungsform für Peptide, Verfahren zu deren Herstellung und Verwendung
WO2003002095A1 (fr) * 2001-06-28 2003-01-09 Chugai Seiyaku Kabushiki Kaisha Preparation d'une micro-emulsion de type huile-eau
US6960563B2 (en) 2001-08-31 2005-11-01 Morton Grove Pharmaceuticals, Inc. Spontaneous emulsions containing cyclosporine
GB2391471B (en) * 2002-08-02 2005-05-04 Satishchandra Punambhai Patel Pharmaceutical compositions
KR20040047056A (ko) * 2002-11-29 2004-06-05 한미약품 주식회사 비페닐디메틸디카복실레이트의 경구용 마이크로에멀젼조성물
US8802116B2 (en) 2003-02-27 2014-08-12 Novasel Australia Pty. Ltd. Poloxamer emulsion preparations
KR20040084240A (ko) * 2003-03-27 2004-10-06 (주) 코스메디 고형지질나노입자, 이를 함유하는 활성성분 전달용약학조성물 및 이의 제조방법
US20050118344A1 (en) 2003-12-01 2005-06-02 Pacetti Stephen D. Temperature controlled crimping
WO2006050123A1 (fr) * 2004-10-29 2006-05-11 Novartis Ag Compositions pharmaceutiques a dispersion spontanee
CN101141953A (zh) * 2005-03-21 2008-03-12 伊瓦克斯制药有限公司 结晶抑制剂及其在明胶胶囊中的用途
CN101032620B (zh) * 2007-03-08 2010-05-19 上海凯昭医药科技有限公司 一种环孢素自乳化制剂及其制备方法
US20090130198A1 (en) * 2007-11-21 2009-05-21 Innopharmax Inc. Pharmaceutical composition with enhanced bioavailability
US8282977B2 (en) 2008-03-20 2012-10-09 Virun, Inc. Compositions containing non-polar compounds
BRPI0909185A2 (pt) 2008-03-20 2015-08-25 Virun Inc Derivado de vitamina e e seus usos
US11304960B2 (en) 2009-01-08 2022-04-19 Chandrashekar Giliyar Steroidal compositions
JP5567909B2 (ja) * 2010-06-17 2014-08-06 東洋カプセル株式会社 タクロリムス含有カプセル剤
US8741373B2 (en) 2010-06-21 2014-06-03 Virun, Inc. Compositions containing non-polar compounds
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US9358241B2 (en) 2010-11-30 2016-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US9034858B2 (en) 2010-11-30 2015-05-19 Lipocine Inc. High-strength testosterone undecanoate compositions
US20120148675A1 (en) 2010-12-10 2012-06-14 Basawaraj Chickmath Testosterone undecanoate compositions
JO3337B1 (ar) 2010-12-13 2019-03-13 Debiopharm Sa تركيبات صيدلية تشمل أليسبوريفير
JP5717034B2 (ja) * 2012-08-27 2015-05-13 丸和バイオケミカル株式会社 マクロライド系化合物を含有する土壌線虫防除用薬剤
KR101458466B1 (ko) * 2013-06-24 2014-11-07 한국화학연구원 면역억제제가 봉입된 마이셀을 함유하는 경구제
WO2016033556A1 (fr) 2014-08-28 2016-03-03 Lipocine Inc. Esters de (17-β)-hydroxy-4-androstène-3-one biodisponibles à l'état solide
WO2016033549A2 (fr) 2014-08-28 2016-03-03 Lipocine Inc. Compositions de (17-ss)-3-oxoandrost-4-èn-17-yl tridécanoate et leurs procédés de préparation et d'utilisation
WO2017048807A1 (fr) 2015-09-17 2017-03-23 Jrx Biotechnology, Inc. Approches pour améliorer l'hydratation ou l'humidification de la peau
CA3078723A1 (fr) 2016-11-28 2018-05-31 Nachiappan Chidambaram Traitement oral a base d'undecanoate de testosterone
CN113194927B (zh) * 2018-11-26 2023-10-27 海必恩制药公司 环孢菌素类似物的药物制剂
WO2024014959A2 (fr) * 2022-07-15 2024-01-18 Seranovo Holding B.V. Formulations générant des micelles avec une hydrophobicité améliorée
WO2024014958A2 (fr) * 2022-07-15 2024-01-18 Seranovo Holding B.V. Plate-forme de formulation de lides

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8903804D0 (en) * 1989-02-20 1989-04-05 Sandoz Ltd Improvements in or relating to organic compounds
US5639724A (en) * 1984-07-24 1997-06-17 Sandoz Ltd. Cyclosporin galenic forms
JP2632010B2 (ja) * 1988-01-29 1997-07-16 三共株式会社 シクロスポリン製剤
KR0148748B1 (ko) * 1988-09-16 1998-08-17 장 크라메르, 한스 루돌프 하우스 사이클로스포린을 함유하는 약학조성물
GB9113872D0 (en) * 1991-06-27 1991-08-14 Sandoz Ag Improvements in or relating to organic compounds
DK0589843T3 (da) * 1992-09-25 2002-04-02 Novartis Ag Cyclosporinholdige farmaceutiske præparater
GB2278780B (en) * 1993-05-27 1998-10-14 Sandoz Ltd Macrolide formulations
DE4322826A1 (de) * 1993-07-08 1995-01-12 Galenik Labor Freiburg Gmbh Pharmazeutisches Präparat
EP0694308A4 (fr) * 1994-02-17 1997-09-10 Shiseido Co Ltd Composition d'emulsion a base de cyclosporine
JP3131112B2 (ja) * 1994-02-17 2001-01-31 株式会社資生堂 シクロスポリン含有乳化組成物
CN100335063C (zh) * 1994-10-26 2007-09-05 诺瓦蒂斯有限公司 药物组合物
MY129435A (en) * 1994-10-26 2007-04-30 Novartis Ag Pharmaceutical microemulsion preconcentrates
HU215966B (hu) * 1994-11-21 1999-07-28 BIOGAL Gyógyszergyár Rt. Orálisan alkalmazható, ciklosporint tartalmazó, összetett emulzió-előkoncentrátum
KR970064620A (ko) * 1996-03-05 1997-10-13 임성기 사이클로스포린-함유 외용약제 조성물
KR980008239A (ko) * 1996-07-26 1998-04-30 김충환 사이클로스포린-함유 약학적 조성물
US6063762A (en) * 1997-12-05 2000-05-16 Chong Kun Dang Corp. Cyclosporin-containing microemulsion preconcentrate composition
WO1999029316A1 (fr) * 1997-12-10 1999-06-17 Severson, Mary, L. Compositions pharmaceutiques contenant une huile d'acide gras omega-3

Also Published As

Publication number Publication date
GB2350791A (en) 2000-12-13
JP2004189753A (ja) 2004-07-08
BE1012400A5 (fr) 2000-10-03
KR20010041657A (ko) 2001-05-25
ITMI990452A1 (it) 2000-09-05
FR2800277A1 (fr) 2001-05-04
SK285139B6 (sk) 2006-07-07
NO20004299D0 (no) 2000-08-29
KR100443306B1 (ko) 2004-08-09
EP1059913B1 (fr) 2004-09-29
EP1059913A1 (fr) 2000-12-20
PE20000324A1 (es) 2000-04-13
TWI248368B (en) 2006-02-01
HK1034038A1 (en) 2001-10-12
HUP0101080A2 (hu) 2001-08-28
CA2322845A1 (fr) 1999-09-10
FR2881956A1 (fr) 2006-08-18
CN1195495C (zh) 2005-04-06
ES2228014T3 (es) 2005-04-01
TW200422057A (en) 2004-11-01
ATE277599T1 (de) 2004-10-15
AU2836199A (en) 1999-09-20
GB2350791B (en) 2003-04-02
AR015729A1 (es) 2001-05-16
FR2853546B1 (fr) 2006-04-07
CO4930289A1 (es) 2000-06-27
NO331800B1 (no) 2012-04-02
SK13192000A3 (sk) 2001-02-12
PT1059913E (pt) 2005-01-31
IL138248A0 (en) 2001-10-31
CZ301967B6 (cs) 2010-08-18
FR2853546A1 (fr) 2004-10-15
WO1999044584A1 (fr) 1999-09-10
CZ20003222A3 (cs) 2000-12-13
AU749217B2 (en) 2002-06-20
DE69920668T2 (de) 2005-10-06
HK1033277A1 (en) 2001-08-24
MY129274A (en) 2007-03-30
GB0021495D0 (en) 2000-10-18
NZ506644A (en) 2004-02-27
CN1292684A (zh) 2001-04-25
BE1013423A5 (fr) 2002-01-15
DE19983012T1 (de) 2001-02-01
BE1013648A5 (fr) 2002-05-07
CA2322845C (fr) 2009-12-08
IL138248A (en) 2006-06-11
JP2002505271A (ja) 2002-02-19
NO20004299L (no) 2000-08-29
ID25908A (id) 2000-11-09
IT1313550B1 (it) 2002-09-09
TWI257870B (en) 2006-07-11
DE69920668D1 (de) 2004-11-04
HUP0101080A3 (en) 2001-12-28
EP1354582A3 (fr) 2004-06-09
TWI236912B (en) 2005-08-01
TR200002586T2 (tr) 2000-11-21
EP1354582A2 (fr) 2003-10-22
FR2775596A1 (fr) 1999-09-10
FR2800277B1 (fr) 2004-06-25
BR9908597A (pt) 2000-11-14

Similar Documents

Publication Publication Date Title
FR2775596B1 (fr) Nouvelles compositions pharmaceutiques
FI991485A (fi) Uusi farmaseuttinen koostumus
IS5046A (is) Lyfjasamsetningar
ID27415A (id) Komposisi farmaseutik
NO20015175D0 (no) Farmasöytisk sammensetning
NO20005913D0 (no) Legemiddelsammensetning
PT1242087E (pt) Composicoes farmaceuticas
NO20012915D0 (no) Ny farmasöytisk formulering
FR2795324B1 (fr) Compositions pharmaceutiques stabilisees
ID29262A (id) Komposisi farmasi
ID27201A (id) Komposisi farmasi
ITMI982222A0 (it) Composizioni farmaceutiche orali contenenti buprenorfina
FR2802423B1 (fr) Compositions pharmaceutiques
IS2515B (is) Lyfjasamsetningar
FR2779145B1 (fr) Nouvelles compositions pharmaceutiques
ID30032A (id) Formulasi farmasi
FI4488U1 (fi) Farmaseuttinen koostumus
EE200000330A (et) Farmatseutilised kompositsioonid
PT1227817E (pt) Composicao farmaceutica aquosa contendo ciclesonida
EE200100281A (et) Analgeetiline ravimkoostis
MA26604A1 (fr) Compositions pharmaceutiques.
NO994436D0 (no) Farmasöytiske sammensetninger
SE9800052D0 (sv) Pharmaceutical compositions
SE9800330D0 (sv) Pharmaceutical compositions
FI981567A0 (fi) Farmaseuttiset koostumukset

Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20121130