FR05C0045I2 - - Google Patents

Info

Publication number
FR05C0045I2
FR05C0045I2 FR05C0045C FR05C0045C FR05C0045I2 FR 05C0045 I2 FR05C0045 I2 FR 05C0045I2 FR 05C0045 C FR05C0045 C FR 05C0045C FR 05C0045 C FR05C0045 C FR 05C0045C FR 05C0045 I2 FR05C0045 I2 FR 05C0045I2
Authority
FR
France
Prior art keywords
pct
date sep
sec
pub
antiobiotic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
FR05C0045C
Other languages
English (en)
French (fr)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Pharmacia and Upjohn Co
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia and Upjohn Co, Upjohn Co filed Critical Pharmacia and Upjohn Co
Publication of FR05C0045I1 publication Critical patent/FR05C0045I1/fr
Application granted granted Critical
Publication of FR05C0045I2 publication Critical patent/FR05C0045I2/fr
Active legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FR05C0045C 1993-03-12 2005-11-17 Active FR05C0045I2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3329193A 1993-03-12 1993-03-12
PCT/US1994/001862 WO1994020505A1 (en) 1993-03-12 1994-03-07 Crystalline ceftiofur free acid

Publications (2)

Publication Number Publication Date
FR05C0045I1 FR05C0045I1 (pt) 2006-01-06
FR05C0045I2 true FR05C0045I2 (pt) 2007-08-03

Family

ID=21869579

Family Applications (1)

Application Number Title Priority Date Filing Date
FR05C0045C Active FR05C0045I2 (pt) 1993-03-12 2005-11-17

Country Status (31)

Country Link
US (1) US5721359A (pt)
EP (1) EP0690864B1 (pt)
JP (1) JP3852946B2 (pt)
KR (1) KR100296810B1 (pt)
CN (1) CN1055090C (pt)
AT (1) ATE202109T1 (pt)
AU (1) AU694419B2 (pt)
BR (1) BR1101034A (pt)
CA (1) CA2155322C (pt)
CZ (1) CZ289332B6 (pt)
DE (2) DE122005000055I2 (pt)
DK (1) DK0690864T3 (pt)
ES (1) ES2157254T3 (pt)
FI (1) FI120307B (pt)
FR (1) FR05C0045I2 (pt)
GR (1) GR3036514T3 (pt)
HU (1) HU222244B1 (pt)
IL (1) IL108910A (pt)
LU (1) LU91206I2 (pt)
LV (1) LV12889B (pt)
NL (1) NL300208I2 (pt)
NO (2) NO313199B1 (pt)
NZ (1) NZ263002A (pt)
PL (1) PL184611B1 (pt)
PT (1) PT690864E (pt)
RU (1) RU2136685C1 (pt)
SI (1) SI0690864T1 (pt)
SK (1) SK283674B6 (pt)
TW (1) TW267170B (pt)
WO (1) WO1994020505A1 (pt)
ZA (1) ZA941586B (pt)

Families Citing this family (70)

* Cited by examiner, † Cited by third party
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US5736151A (en) * 1996-12-09 1998-04-07 Pharmacia & Upjohn Company Antibiotic oil suspensions
US6074657A (en) * 1997-03-20 2000-06-13 Pharmacia & Upjohn Company Administration of an injectable antibiotic in the ear of an animal
JP4738713B2 (ja) * 2000-09-12 2011-08-03 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 修飾された担体を含む医薬組成物
US7829100B2 (en) * 2000-09-12 2010-11-09 Teagarden Dirk L Pharmaceutical composition having modified carrier
KR100423895B1 (ko) * 2001-02-19 2004-03-24 주식회사 엘지생명과학 셉티오퍼 하이드로클로라이드의 현탁제 조성물
EP1406880A1 (en) * 2001-07-10 2004-04-14 PHARMACIA & UPJOHN COMPANY Crystalline thiazine oxazolidinones
EP3168218B1 (en) * 2001-08-15 2018-11-14 Pharmacia & Upjohn Company LLC A crystal comprising an l-malic acid salt of n-[2-(diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide for use as a medicament
KR20040097187A (ko) † 2002-03-21 2004-11-17 파마시아 앤드 업존 캄파니 동물의 귀로의 주사가능한 항생제의 투여 방법
US20040022815A1 (en) * 2002-08-05 2004-02-05 Orchid Health Care Novel pharmaceutical composition of ceftiofur
KR20040015622A (ko) * 2002-08-13 2004-02-19 대한뉴팜(주) 세프티오푸르나트륨을 활성성분으로 함유하는 현탁주사액조성물
US20040115822A1 (en) * 2002-09-12 2004-06-17 Schapaugh Randal Lee Methods of measuring the dissolution rate of an analyte in a non-aqueous liquid composition
US7659061B2 (en) * 2002-11-19 2010-02-09 Pharmacia & Upjohn Company Pharmaceutical compositions having a modified vehicle
US20040115837A1 (en) * 2002-11-27 2004-06-17 Schapaugh Randal Lee Methods of measuring the dissolution rate of an analyte in a non-aqueous liquid composition
US7842791B2 (en) * 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
ATE440101T1 (de) * 2003-03-27 2009-09-15 Basilea Pharmaceutica Ag Cephalosporin in kristalliner form
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US7815939B2 (en) 2005-07-20 2010-10-19 Astellas Pharma Inc. Coated fine particles containing drug for intrabuccally fast disintegrating dosage forms
EP1934231A4 (en) * 2005-10-12 2011-10-26 Orchid Chemicals & Pharm Ltd CRYSTALLINE SODIUM SALT OF ANTIBIOTICS BASED ON CEPHALOSPORINE
US8470809B2 (en) * 2005-10-12 2013-06-25 Orchid Chemicals & Pharmaceuticals Limited Crystalline sodium salt of cephalosporin antibiotic
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US9943614B2 (en) 2008-06-17 2018-04-17 Brigham Young University Cationic steroid antimicrobial diagnostic, detection, screening and imaging methods
WO2010020871A2 (en) * 2008-08-22 2010-02-25 Orchid Chemicals & Pharmaceuticals Limited Crystalline sodium salt of cephalosporin antibiotic
AU2009316708B2 (en) * 2008-11-19 2014-07-17 Boehringer Ingelheim Animal Health USA Inc. Formulations comprising ceftiofur and ketoprofen or ceftiofur and benzyl alcohol
PE20120003A1 (es) * 2009-01-30 2012-02-12 Glaxosmithkline Llc Hidrocloruro de n-{(1s)-2-amino-1-[(3-fluorofenil)metil)etil}-5-cloro-4-(4-cloro-1-metil-1h-pirazol-5-il)-2-tiofenocarboxamida cristalino
TW201039825A (en) 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
RU2012136148A (ru) 2010-02-18 2014-03-27 Астразенека Аб Новая кристаллическая форма производного циклопропилбензамида
AU2011218490B9 (en) * 2010-02-18 2014-12-18 Astrazeneca Ab Solid forms comprising a cyclopropyl amide derivative
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CN104053458B (zh) 2011-07-20 2016-07-20 布莱阿姆青年大学 包含洗脱塞拉集宁化合物的水凝胶材料
JP6038154B2 (ja) 2011-09-13 2016-12-07 ブリガム・ヤング・ユニバーシティＢｒｉｇｈａｍ Ｙｏｕｎｇ Ｕｎｉｖｅｒｓｉｔｙ 骨疾患および破断骨治療のための組成物
KR101966293B1 (ko) 2011-09-13 2019-04-08 브라이엄 영 유니버시티 손상조직 치유용 제품
US9694019B2 (en) 2011-09-13 2017-07-04 Brigham Young University Compositions and methods for treating bone diseases and broken bones
US9603859B2 (en) 2011-09-13 2017-03-28 Brigham Young University Methods and products for increasing the rate of healing of tissue wounds
MX2014007496A (es) 2011-12-21 2015-02-17 Univ Brigham Young Composiciones para el cuidado oral.
CN102584855B (zh) * 2012-02-16 2014-06-25 青岛科技大学 一种改进的头孢噻呋的制备方法
US9533063B1 (en) 2012-03-01 2017-01-03 Brigham Young University Aerosols incorporating ceragenin compounds and methods of use thereof
CA2872399C (en) 2012-05-02 2021-01-12 Brigham Young University Ceragenin particulate materials and methods for making same
BR112015008804A2 (pt) 2012-10-17 2017-07-04 Univ Brigham Young tratamento e prevenção de mastite
WO2014087972A1 (ja) * 2012-12-03 2014-06-12 株式会社カネカ 還元型補酵素ｑ10誘導体およびその製造方法
CA2897150C (en) 2013-01-07 2021-07-13 Brigham Young University Methods for reducing cellular proliferation and treating certain diseases
US11524015B2 (en) 2013-03-15 2022-12-13 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
WO2014151411A1 (en) 2013-03-15 2014-09-25 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
US10568893B2 (en) 2013-03-15 2020-02-25 Brigham Young University Methods for treating inflammation, autoimmune disorders and pain
RU2546675C2 (ru) * 2013-04-11 2015-04-10 Федеральное казённое предприятие "Государственный научно-исследовательский институт химических продуктов" (ФКП "ГосНИИХП") Способ определения степени кристалличности составов на основе дифениламина
US9387215B2 (en) 2013-04-22 2016-07-12 Brigham Young University Animal feed including cationic cholesterol additive and related methods
KR102177643B1 (ko) * 2013-09-05 2020-11-11 미쓰비시 타나베 파마 코퍼레이션 신규한 결정성 아릴알킬아민 화합물 및 그의 제조 방법
US11690855B2 (en) 2013-10-17 2023-07-04 Brigham Young University Methods for treating lung infections and inflammation
US20150203527A1 (en) 2014-01-23 2015-07-23 Brigham Young University Cationic steroidal antimicrobials
CA2844321C (en) 2014-02-27 2021-03-16 Brigham Young University Cationic steroidal antimicrobial compounds
US9867836B2 (en) 2014-03-13 2018-01-16 Brigham Young University Lavage and/or infusion using CSA compounds for increasing fertility in a mammal
US10220045B2 (en) 2014-03-13 2019-03-05 Brigham Young University Compositions and methods for forming stabilized compositions with reduced CSA agglomeration
US9931350B2 (en) 2014-03-14 2018-04-03 Brigham Young University Anti-infective and osteogenic compositions and methods of use
US9686966B2 (en) 2014-04-30 2017-06-27 Brigham Young University Methods and apparatus for cleaning or disinfecting a water delivery system
US10238665B2 (en) 2014-06-26 2019-03-26 Brigham Young University Methods for treating fungal infections
US10441595B2 (en) 2014-06-26 2019-10-15 Brigham Young University Methods for treating fungal infections
US10227376B2 (en) 2014-08-22 2019-03-12 Brigham Young University Radiolabeled cationic steroid antimicrobials and diagnostic methods
US10155788B2 (en) 2014-10-07 2018-12-18 Brigham Young University Cationic steroidal antimicrobial prodrug compositions and uses thereof
KR102331856B1 (ko) * 2014-10-21 2021-11-29 다케다 야쿠힌 고교 가부시키가이샤 결정 형태의 5-클로로-n4-[2-(디메틸포스포릴)페닐]-n2-｛2-메톡시-4-[4-(4-메틸피페라진-1-일)피페리딘-1-일]피리미딘-2,4-디아민
US9527883B2 (en) 2015-04-22 2016-12-27 Brigham Young University Methods for the synthesis of ceragenins
WO2016172543A1 (en) 2015-04-22 2016-10-27 Savage Paul B Methods for the synthesis of ceragenins
KR101753842B1 (ko) * 2015-05-12 2017-07-04 한국화학연구원 불화퀴놀론계 항생제를 담지한 서방형 제제 및 이의 제조방법
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CN106543203B (zh) * 2015-09-18 2019-07-02 瑞普（天津）生物药业有限公司 一种长效头孢噻呋自由酸晶体的制备方法
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KR101898282B1 (ko) * 2016-05-24 2018-09-13 주식회사 고려비엔피 항생제의 서방형 수의학적 조성물 및 이의 제조방법
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Also Published As

Publication number Publication date
FI120307B (fi) 2009-09-15
ES2157254T3 (es) 2001-08-16
SI0690864T1 (en) 2001-10-31
PL310556A1 (en) 1995-12-27
LV12889B (lv) 2002-12-20
NZ263002A (en) 1996-12-20
SK111495A3 (en) 1995-12-06
CA2155322A1 (en) 1994-09-15
SK283674B6 (sk) 2003-11-04
CZ289332B6 (cs) 2002-01-16
EP0690864A1 (en) 1996-01-10
DE69427469D1 (en) 2001-07-19
FR05C0045I1 (pt) 2006-01-06
HU9501960D0 (en) 1995-09-28
FI954250A0 (fi) 1995-09-11
AU694419B2 (en) 1998-07-23
IL108910A (en) 1999-10-28
JP3852946B2 (ja) 2006-12-06
DE122005000055I1 (de) 2006-02-23
NO953564L (no) 1995-11-07
EP0690864B1 (en) 2001-06-13
CZ9502290A3 (cs) 2001-08-15
NO2005025I2 (no) 2010-11-22
HU222244B1 (hu) 2003-05-28
DE122005000055I2 (de) 2008-06-05
GR3036514T3 (en) 2001-12-31
CN1055090C (zh) 2000-08-02
KR100296810B1 (ko) 2001-10-24
NO953564D0 (no) 1995-09-11
NL300208I1 (nl) 2006-02-01
FI954250A (fi) 1995-09-11
PT690864E (pt) 2001-11-30
ATE202109T1 (de) 2001-06-15
IL108910A0 (en) 1994-06-24
ZA941586B (en) 1995-09-07
PL184611B1 (pl) 2002-11-29
DE69427469T2 (de) 2001-10-31
JPH08507519A (ja) 1996-08-13
BR1101034A (pt) 2002-04-30
CA2155322C (en) 2000-02-29
RU2136685C1 (ru) 1999-09-10
NO2005025I1 (no) 2005-12-05
NL300208I2 (nl) 2006-05-01
CN1119016A (zh) 1996-03-20
AU6351094A (en) 1994-09-26
US5721359A (en) 1998-02-24
LU91206I2 (fr) 2006-05-30
DK0690864T3 (da) 2001-09-17
WO1994020505A1 (en) 1994-09-15
HUT73781A (en) 1996-09-30
NO313199B1 (no) 2002-08-26
TW267170B (pt) 1996-01-01

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