FI970578A0 - Uusia kinoloni- tai naftyridonikarboksyylihappojohdannaisia tai niiden suola - Google Patents

Uusia kinoloni- tai naftyridonikarboksyylihappojohdannaisia tai niiden suola

Info

Publication number
FI970578A0
FI970578A0 FI970578A FI970578A FI970578A0 FI 970578 A0 FI970578 A0 FI 970578A0 FI 970578 A FI970578 A FI 970578A FI 970578 A FI970578 A FI 970578A FI 970578 A0 FI970578 A0 FI 970578A0
Authority
FI
Finland
Prior art keywords
group
substituted
hydrogen atom
lower alkyl
salts
Prior art date
Application number
FI970578A
Other languages
English (en)
Swedish (sv)
Other versions
FI113652B (fi
FI970578A (fi
Inventor
Yozo Todo
Kazuya Hayashi
Masahiro Takahata
Yasuo Watanabe
Hirokazu Narita
Original Assignee
Toyoma Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyoma Chemical Co Ltd filed Critical Toyoma Chemical Co Ltd
Publication of FI970578A0 publication Critical patent/FI970578A0/fi
Publication of FI970578A publication Critical patent/FI970578A/fi
Application granted granted Critical
Publication of FI113652B publication Critical patent/FI113652B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/22Tin compounds
    • C07F7/2208Compounds having tin linked only to carbon, hydrogen and/or halogen
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI970578A 1994-08-12 1997-02-11 Uusia kinoloni- tai naftyridonikarboksyylihappojohdannaisia tai niiden suola FI113652B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP21208394 1994-08-12
JP21208394 1994-08-12
PCT/JP1995/001551 WO1996005192A1 (fr) 1994-08-12 1995-08-04 Derive du nouvel acide quinolone- ou naphthyridonecarboxylique ou son sel
JP9501551 1995-08-04

Publications (3)

Publication Number Publication Date
FI970578A0 true FI970578A0 (fi) 1997-02-11
FI970578A FI970578A (fi) 1997-04-10
FI113652B FI113652B (fi) 2004-05-31

Family

ID=16616594

Family Applications (1)

Application Number Title Priority Date Filing Date
FI970578A FI113652B (fi) 1994-08-12 1997-02-11 Uusia kinoloni- tai naftyridonikarboksyylihappojohdannaisia tai niiden suola

Country Status (17)

Country Link
US (1) US5935952A (fi)
EP (1) EP0775702B1 (fi)
KR (1) KR100371723B1 (fi)
CN (1) CN1070191C (fi)
AT (1) ATE245638T1 (fi)
AU (1) AU692583B2 (fi)
CA (1) CA2196271C (fi)
DE (1) DE69531350T2 (fi)
DK (1) DK0775702T3 (fi)
ES (1) ES2203644T3 (fi)
FI (1) FI113652B (fi)
HU (1) HU228062B1 (fi)
IL (1) IL114875A (fi)
NO (1) NO312032B1 (fi)
NZ (1) NZ290946A (fi)
WO (1) WO1996005192A1 (fi)
ZA (1) ZA956713B (fi)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69622569T2 (de) * 1995-08-21 2003-01-16 Takeda Chemical Industries Ltd Quinoneverbindung, seine herstellung und anwendung.
CA2242242C (en) * 1996-02-09 2001-08-07 Toyama Chemical Co., Ltd. Quinolonecarboxylic acid derivatives or salts thereof
WO1999007682A1 (fr) * 1997-08-08 1999-02-18 Toyama Chemical Co., Ltd. Derives d'acide quinolonecarboxylique ou sels de ces derives
AU735186B2 (en) 1997-09-15 2001-07-05 Warner Chilcott Company, Llc Antimicrobial quinolones, their compositions and uses
CN1515555A (zh) * 1997-10-27 2004-07-28 ��ɽ��ѧ��ҵ��ʽ���� 制备7-溴喹诺酮羧酸衍生物或其盐的方法
JP4549461B2 (ja) * 1998-08-31 2010-09-22 富山化学工業株式会社 7−ブロモ−キノロンカルボン酸誘導体の製造法
WO2000046223A1 (fr) * 1999-02-05 2000-08-10 Toyama Chemical Co., Ltd. Derives tricycliques d'acide quinolonecarboxylique ou sels de ces derives
AU7948900A (en) 1999-10-19 2001-04-30 Sato Pharmaceutical Co., Ltd. 4-oxoquinolizine antimicrobials having 2-pyridone skeletons as the partial structure
ATE364036T1 (de) 2000-03-07 2007-06-15 Ranbaxy Lab Ltd Eintopfsynthese von 3-cyclopropylamino-2- 2,4- dibromo-3-(difluoromethoxy)benzoylö-2-propensäu e alkylester als nützliches zwischenprodukt für antibakterielle quinolon-arzneistoffe
JP2005232000A (ja) * 2000-03-10 2005-09-02 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体又はその塩
US6525049B2 (en) 2000-07-05 2003-02-25 Pharmacia & Upjohn Company Pyrroloquinolones as antiviral agents
US6861071B2 (en) * 2000-08-08 2005-03-01 Daiichi Pharmaceutical Co., Ltd. Highly absorptive solid preparation
WO2002048143A2 (en) 2000-12-14 2002-06-20 The Procter & Gamble Company Antimicrobial 2-pyridones, their compositions and uses
AU3089102A (en) 2000-12-14 2002-06-24 Procter & Gamble Antimicrobial quinolones
EP1614680B1 (en) 2001-04-19 2011-12-21 Eisai R&D Management Co., Ltd. Process for preparing 2-iminopyrrolidine derivatives
CN100337630C (zh) * 2002-03-12 2007-09-19 布里斯托尔-迈尔斯斯奎布公司 可口的口服悬浮液及其制备方法
CN100439336C (zh) * 2003-02-19 2008-12-03 卫材R&D管理有限公司 制备环状苯甲脒衍生物的方法
KR101084521B1 (ko) 2006-03-28 2011-11-18 워너 칠콧 컴퍼니 엘엘씨 퀴놀론 중간체를 제조하기 위한 커플링 방법
MX2008012328A (es) 2006-03-28 2008-10-09 Procter & Gamble Sales de malato, y polimorfos de acido (3s,5s)-7-[3-amino-5-metil- piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinc arboxilico.
JP2008031090A (ja) * 2006-07-28 2008-02-14 Toyota Central Res & Dev Lab Inc 有機スズ化合物及びその製造方法、並びに芳香族化合物誘導体の製造方法
CN101298418B (zh) * 2008-06-13 2010-12-15 江苏康鹏农化有限公司 3-氧代-3-(2,4-二卤代-3-二氟甲氧基苯基)丙酸乙酯的制备方法
CN102212056A (zh) * 2010-04-09 2011-10-12 山东轩竹医药科技有限公司 新的双环喹诺酮类化合物
SG10201505811QA (en) 2011-08-31 2015-09-29 Otsuka Pharma Co Ltd Quinolone compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3248507A1 (de) * 1982-12-29 1984-07-05 Bayer Ag, 5090 Leverkusen Mikrobizide mittel auf chinoloncarbonsaeure basis
ZA859283B (en) * 1984-12-06 1987-07-29 Pfizer Substituted dihydroquinolone carboxylic acids and anti-bacterial compositions containing them
DE3816119A1 (de) * 1988-05-11 1989-11-23 Bayer Ag 7-substituierte chinolon- und naphthyridoncarbonsaeure-derivate
JPH0262875A (ja) * 1988-05-23 1990-03-02 Wakunaga Pharmaceut Co Ltd 新規イソインドリン誘導体
US4945160A (en) * 1988-11-22 1990-07-31 Warner-Lambert Company Preparation of certain 7-substituted quinolones

Also Published As

Publication number Publication date
ZA956713B (en) 1996-03-28
NO970622L (no) 1997-04-10
CA2196271C (en) 2007-01-09
IL114875A0 (en) 1995-12-08
DK0775702T3 (da) 2003-08-18
HUT77314A (hu) 1998-03-30
HU228062B1 (en) 2012-09-28
FI113652B (fi) 2004-05-31
DE69531350D1 (de) 2003-08-28
EP0775702A4 (en) 1997-11-05
CN1070191C (zh) 2001-08-29
US5935952A (en) 1999-08-10
KR970704728A (ko) 1997-09-06
NO970622D0 (no) 1997-02-11
AU3190695A (en) 1996-03-07
NZ290946A (en) 1997-12-19
DE69531350T2 (de) 2004-05-27
ATE245638T1 (de) 2003-08-15
CN1158611A (zh) 1997-09-03
ES2203644T3 (es) 2004-04-16
AU692583B2 (en) 1998-06-11
FI970578A (fi) 1997-04-10
EP0775702A1 (en) 1997-05-28
WO1996005192A1 (fr) 1996-02-22
CA2196271A1 (en) 1996-02-22
NO312032B1 (no) 2002-03-04
EP0775702B1 (en) 2003-07-23
IL114875A (en) 1999-12-22
KR100371723B1 (ko) 2003-03-15

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