FI890652A - Förfarande för framställning av terapeutiskt aktiva substituerade indolylpyrrolderivat - Google Patents

Förfarande för framställning av terapeutiskt aktiva substituerade indolylpyrrolderivat Download PDF

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Publication number
FI890652A
FI890652A FI890652A FI890652A FI890652A FI 890652 A FI890652 A FI 890652A FI 890652 A FI890652 A FI 890652A FI 890652 A FI890652 A FI 890652A FI 890652 A FI890652 A FI 890652A
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Finland
Prior art keywords
indolylpyrrole
derivatives
preparation
therapeutically active
active substituted
Prior art date
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FI890652A
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English (en)
Finnish (fi)
Other versions
FI96861C (sv
FI96861B (sv
FI890652A0 (sv
Inventor
Peter David Davis
Christopher Huw Hill
Geoffrey Lawton
Original Assignee
Hoffmann La Roche
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Priority claimed from GB888803048A external-priority patent/GB8803048D0/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of FI890652A0 publication Critical patent/FI890652A0/sv
Publication of FI890652A publication Critical patent/FI890652A/sv
Application granted granted Critical
Publication of FI96861B publication Critical patent/FI96861B/sv
Publication of FI96861C publication Critical patent/FI96861C/sv

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/044Pyrrole radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrrole Compounds (AREA)
FI890652A 1988-02-10 1989-02-10 Förfarande för framställning av terapeutiskt aktiva substituerade indolylpyrrolderivat FI96861C (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8803048 1988-02-10
GB888803048A GB8803048D0 (en) 1988-02-10 1988-02-10 Substituted pyrroles
GB8827565 1988-10-25
GB888827565A GB8827565D0 (en) 1988-02-10 1988-11-25 Substituted pyrroles

Publications (4)

Publication Number Publication Date
FI890652A0 FI890652A0 (sv) 1989-02-10
FI890652A true FI890652A (sv) 1989-08-11
FI96861B FI96861B (sv) 1996-05-31
FI96861C FI96861C (sv) 1996-09-10

Family

ID=26293462

Family Applications (1)

Application Number Title Priority Date Filing Date
FI890652A FI96861C (sv) 1988-02-10 1989-02-10 Förfarande för framställning av terapeutiskt aktiva substituerade indolylpyrrolderivat

Country Status (22)

Country Link
US (1) US5057614A (sv)
EP (1) EP0328026B1 (sv)
JP (1) JPH0730071B2 (sv)
AU (1) AU623630B2 (sv)
CA (1) CA1320194C (sv)
CZ (1) CZ280738B6 (sv)
DE (1) DE58904168D1 (sv)
DK (1) DK171891B1 (sv)
DZ (1) DZ1323A1 (sv)
ES (1) ES2054890T3 (sv)
FI (1) FI96861C (sv)
HU (1) HU201054B (sv)
IE (1) IE63489B1 (sv)
IL (1) IL89167A (sv)
IS (1) IS1941B (sv)
MC (1) MC2010A1 (sv)
NO (1) NO172540C (sv)
NZ (1) NZ227850A (sv)
PH (1) PH25185A (sv)
PT (1) PT89661B (sv)
SK (1) SK278989B6 (sv)
YU (1) YU47101B (sv)

Families Citing this family (132)

* Cited by examiner, † Cited by third party
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PH25185A (en) 1991-03-27
MC2010A1 (fr) 1990-02-16
FI96861C (sv) 1996-09-10
IE63489B1 (en) 1995-05-03
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PT89661B (pt) 1994-02-28
ES2054890T3 (es) 1994-08-16
YU28489A (en) 1991-06-30
NO890568D0 (no) 1989-02-09
FI96861B (sv) 1996-05-31
EP0328026A1 (de) 1989-08-16
IL89167A0 (en) 1989-09-10
EP0328026B1 (de) 1993-04-28
PT89661A (pt) 1989-10-04
CA1320194C (en) 1993-07-13
DZ1323A1 (fr) 2004-09-13
CZ75289A3 (en) 1995-12-13
AU623630B2 (en) 1992-05-21
SK278989B6 (sk) 1998-05-06
HUT49348A (en) 1989-09-28
IS1941B (is) 2004-07-30
HU201054B (en) 1990-09-28
IE890416L (en) 1989-08-10
NZ227850A (en) 1991-11-26
US5057614A (en) 1991-10-15
NO172540C (no) 1993-08-04
IL89167A (en) 1994-02-27
JPH01233281A (ja) 1989-09-19
JPH0730071B2 (ja) 1995-04-05
CZ280738B6 (cs) 1996-04-17
NO890568L (no) 1989-08-11
NO172540B (no) 1993-04-26
DK171891B1 (da) 1997-08-04
DK55889D0 (da) 1989-02-07
DE58904168D1 (de) 1993-06-03
IS3433A7 (is) 1989-08-11
AU2965889A (en) 1989-08-10
DK55889A (da) 1989-08-11
FI890652A0 (sv) 1989-02-10
YU47101B (sh) 1994-12-28

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