FI64590C - Analogifoerfarande foer framstaellning av terapeutiskt aktiva indoler - Google Patents

Analogifoerfarande foer framstaellning av terapeutiskt aktiva indoler Download PDF

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Publication number
FI64590C
FI64590C FI753669A FI753669A FI64590C FI 64590 C FI64590 C FI 64590C FI 753669 A FI753669 A FI 753669A FI 753669 A FI753669 A FI 753669A FI 64590 C FI64590 C FI 64590C
Authority
FI
Finland
Prior art keywords
formula
compound
iii
methyl
group
Prior art date
Application number
FI753669A
Other languages
English (en)
Finnish (fi)
Other versions
FI753669A (no
FI64590B (fi
Inventor
Michael Zelesko
David Mccomsey
Original Assignee
Mcneilab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mcneilab Inc filed Critical Mcneilab Inc
Publication of FI753669A publication Critical patent/FI753669A/fi
Application granted granted Critical
Publication of FI64590B publication Critical patent/FI64590B/fi
Publication of FI64590C publication Critical patent/FI64590C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms
FI753669A 1974-12-30 1975-12-29 Analogifoerfarande foer framstaellning av terapeutiskt aktiva indoler FI64590C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US53761274A 1974-12-30 1974-12-30
US53761274 1974-12-30
US63179875A 1975-11-13 1975-11-13
US63179875 1975-11-13

Publications (3)

Publication Number Publication Date
FI753669A FI753669A (no) 1976-07-01
FI64590B FI64590B (fi) 1983-08-31
FI64590C true FI64590C (fi) 1983-12-12

Family

ID=27065555

Family Applications (1)

Application Number Title Priority Date Filing Date
FI753669A FI64590C (fi) 1974-12-30 1975-12-29 Analogifoerfarande foer framstaellning av terapeutiskt aktiva indoler

Country Status (27)

Country Link
JP (1) JPS51131872A (no)
AR (1) AR219052A1 (no)
AT (1) AT356648B (no)
AU (1) AU505215B2 (no)
CA (1) CA1065874A (no)
CH (1) CH622516A5 (no)
DD (1) DD125781A5 (no)
DE (1) DE2559211A1 (no)
DK (1) DK580175A (no)
ES (1) ES443935A1 (no)
FI (1) FI64590C (no)
FR (2) FR2296413A1 (no)
GB (1) GB1527510A (no)
HU (2) HU174948B (no)
IE (1) IE42390B1 (no)
IL (1) IL48756A (no)
IN (1) IN142735B (no)
IT (1) IT1052654B (no)
NL (1) NL7515100A (no)
NO (1) NO145383C (no)
NZ (1) NZ179580A (no)
PH (1) PH12328A (no)
PL (1) PL99353B1 (no)
RO (1) RO69196A (no)
SE (1) SE422210B (no)
SU (1) SU667132A3 (no)
YU (1) YU332275A (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1595056A (en) * 1976-10-12 1981-08-05 Wellcome Found Pharmaceutical combination
FR2540109B1 (fr) * 1983-01-28 1985-08-30 Logeais Labor Jacques Imino-2 pyrrolidines, leur procede de preparation et leurs applications en therapeutique
US4558048A (en) * 1984-04-06 1985-12-10 Pfizer Inc. Method of treating diarrhoea using indole compounds
WO2001023350A1 (en) * 1999-09-28 2001-04-05 Nihon Nohyaku Co., Ltd. Thioalkylamine derivatives and process for the preparation thereof
UA79504C2 (en) * 2002-11-07 2007-06-25 Organon Nv Indols for treating diseases associated with androgen receptors
US7795280B2 (en) 2002-11-07 2010-09-14 N.V. Organon Indoles useful in the treatment of androgen-receptor related diseases
TW200602317A (en) 2004-04-23 2006-01-16 Akzo Nobel Nv Novel androgens
WO2007020653A1 (en) * 2005-08-12 2007-02-22 Suven Life Sciences Limited Thioether derivatives as functional 5-ht6 ligands

Also Published As

Publication number Publication date
NL7515100A (nl) 1976-07-02
NZ179580A (en) 1978-04-03
FR2296413B1 (no) 1980-06-27
IE42390L (en) 1976-06-30
JPS51131872A (en) 1976-11-16
GB1527510A (en) 1978-10-04
DK580175A (da) 1976-07-01
PL99353B1 (pl) 1978-07-31
ATA986075A (de) 1979-10-15
HU174948B (hu) 1980-04-28
DD125781A5 (no) 1977-05-18
AT356648B (de) 1980-05-12
IL48756A (en) 1979-03-12
SE422210B (sv) 1982-02-22
SU667132A3 (ru) 1979-06-05
AR219052A1 (es) 1980-07-31
ES443935A1 (es) 1977-08-16
HU174949B (hu) 1980-04-28
AU8791675A (en) 1977-07-07
NO754313L (no) 1976-07-01
NO145383C (no) 1982-03-10
NO145383B (no) 1981-11-30
SE7514458L (sv) 1976-07-31
IN142735B (no) 1977-08-20
PH12328A (en) 1979-01-16
RO69196A (ro) 1980-08-15
IE42390B1 (en) 1980-07-30
FR2315921A1 (fr) 1977-01-28
AU505215B2 (en) 1979-11-15
DE2559211A1 (de) 1976-07-08
FR2296413A1 (fr) 1976-07-30
YU332275A (en) 1983-02-28
FI753669A (no) 1976-07-01
FI64590B (fi) 1983-08-31
CA1065874A (en) 1979-11-06
FR2315921B1 (no) 1979-09-28
IT1052654B (it) 1981-07-20
IL48756A0 (en) 1976-02-29
CH622516A5 (en) 1981-04-15

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MM Patent lapsed

Owner name: MCNEIL LABORATORIES INC.