CH622516A5 - Process for the preparation of substituted indoles, and their use - Google Patents

Process for the preparation of substituted indoles, and their use Download PDF

Info

Publication number
CH622516A5
CH622516A5 CH1679775A CH1679775A CH622516A5 CH 622516 A5 CH622516 A5 CH 622516A5 CH 1679775 A CH1679775 A CH 1679775A CH 1679775 A CH1679775 A CH 1679775A CH 622516 A5 CH622516 A5 CH 622516A5
Authority
CH
Switzerland
Prior art keywords
formula
compounds
radical
prepared
same meaning
Prior art date
Application number
CH1679775A
Other languages
German (de)
English (en)
Inventor
Michael Zelesko
David Mccomsey
Original Assignee
Mcneilab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mcneilab Inc filed Critical Mcneilab Inc
Publication of CH622516A5 publication Critical patent/CH622516A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24Oxygen or sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
CH1679775A 1974-12-30 1975-12-24 Process for the preparation of substituted indoles, and their use CH622516A5 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53761274A 1974-12-30 1974-12-30
US63179875A 1975-11-13 1975-11-13

Publications (1)

Publication Number Publication Date
CH622516A5 true CH622516A5 (en) 1981-04-15

Family

ID=27065555

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1679775A CH622516A5 (en) 1974-12-30 1975-12-24 Process for the preparation of substituted indoles, and their use

Country Status (27)

Country Link
JP (1) JPS51131872A (no)
AR (1) AR219052A1 (no)
AT (1) AT356648B (no)
AU (1) AU505215B2 (no)
CA (1) CA1065874A (no)
CH (1) CH622516A5 (no)
DD (1) DD125781A5 (no)
DE (1) DE2559211A1 (no)
DK (1) DK580175A (no)
ES (1) ES443935A1 (no)
FI (1) FI64590C (no)
FR (2) FR2296413A1 (no)
GB (1) GB1527510A (no)
HU (2) HU174948B (no)
IE (1) IE42390B1 (no)
IL (1) IL48756A (no)
IN (1) IN142735B (no)
IT (1) IT1052654B (no)
NL (1) NL7515100A (no)
NO (1) NO145383C (no)
NZ (1) NZ179580A (no)
PH (1) PH12328A (no)
PL (1) PL99353B1 (no)
RO (1) RO69196A (no)
SE (1) SE422210B (no)
SU (1) SU667132A3 (no)
YU (1) YU332275A (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1595056A (en) * 1976-10-12 1981-08-05 Wellcome Found Pharmaceutical combination
FR2540109B1 (fr) * 1983-01-28 1985-08-30 Logeais Labor Jacques Imino-2 pyrrolidines, leur procede de preparation et leurs applications en therapeutique
US4558048A (en) * 1984-04-06 1985-12-10 Pfizer Inc. Method of treating diarrhoea using indole compounds
WO2001023350A1 (en) * 1999-09-28 2001-04-05 Nihon Nohyaku Co., Ltd. Thioalkylamine derivatives and process for the preparation thereof
UA79504C2 (en) * 2002-11-07 2007-06-25 Organon Nv Indols for treating diseases associated with androgen receptors
US7795280B2 (en) 2002-11-07 2010-09-14 N.V. Organon Indoles useful in the treatment of androgen-receptor related diseases
TW200602317A (en) 2004-04-23 2006-01-16 Akzo Nobel Nv Novel androgens
WO2007020653A1 (en) * 2005-08-12 2007-02-22 Suven Life Sciences Limited Thioether derivatives as functional 5-ht6 ligands

Also Published As

Publication number Publication date
NL7515100A (nl) 1976-07-02
NZ179580A (en) 1978-04-03
FR2296413B1 (no) 1980-06-27
IE42390L (en) 1976-06-30
JPS51131872A (en) 1976-11-16
GB1527510A (en) 1978-10-04
DK580175A (da) 1976-07-01
PL99353B1 (pl) 1978-07-31
ATA986075A (de) 1979-10-15
FI64590C (fi) 1983-12-12
HU174948B (hu) 1980-04-28
DD125781A5 (no) 1977-05-18
AT356648B (de) 1980-05-12
IL48756A (en) 1979-03-12
SE422210B (sv) 1982-02-22
SU667132A3 (ru) 1979-06-05
AR219052A1 (es) 1980-07-31
ES443935A1 (es) 1977-08-16
HU174949B (hu) 1980-04-28
AU8791675A (en) 1977-07-07
NO754313L (no) 1976-07-01
NO145383C (no) 1982-03-10
NO145383B (no) 1981-11-30
SE7514458L (sv) 1976-07-31
IN142735B (no) 1977-08-20
PH12328A (en) 1979-01-16
RO69196A (ro) 1980-08-15
IE42390B1 (en) 1980-07-30
FR2315921A1 (fr) 1977-01-28
AU505215B2 (en) 1979-11-15
DE2559211A1 (de) 1976-07-08
FR2296413A1 (fr) 1976-07-30
YU332275A (en) 1983-02-28
FI753669A (no) 1976-07-01
FI64590B (fi) 1983-08-31
CA1065874A (en) 1979-11-06
FR2315921B1 (no) 1979-09-28
IT1052654B (it) 1981-07-20
IL48756A0 (en) 1976-02-29

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Legal Events

Date Code Title Description
PL Patent ceased