FI108611B - Menetelmä mikropartikkelien valmistamiseksi - Google Patents
Menetelmä mikropartikkelien valmistamiseksi Download PDFInfo
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- FI108611B FI108611B FI903429A FI903429A FI108611B FI 108611 B FI108611 B FI 108611B FI 903429 A FI903429 A FI 903429A FI 903429 A FI903429 A FI 903429A FI 108611 B FI108611 B FI 108611B
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- water
- drug
- microparticles
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- polymer
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Classifications
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- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
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- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/095—Oxytocins; Vasopressins; Related peptides
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/23—Calcitonins
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
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- A—HUMAN NECESSITIES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A61K9/1647—Polyesters, e.g. poly(lactide-co-glycolide)
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- A—HUMAN NECESSITIES
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Diabetes (AREA)
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- Immunology (AREA)
- Zoology (AREA)
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- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Obesity (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI991120A FI106926B (fi) | 1989-07-07 | 1999-05-17 | Menetelmä pitkäaikaisesti vapautuvan koostumuksen muodostamiseksi |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37702389A | 1989-07-07 | 1989-07-07 | |
| US37702389 | 1989-07-07 | ||
| US41134789A | 1989-09-22 | 1989-09-22 | |
| US41134789 | 1989-09-22 |
Publications (2)
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|---|---|
| FI903429A0 FI903429A0 (fi) | 1990-07-06 |
| FI108611B true FI108611B (fi) | 2002-02-28 |
Family
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Family Applications (3)
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| FI903429A FI108611B (fi) | 1989-07-07 | 1990-07-06 | Menetelmä mikropartikkelien valmistamiseksi |
| FI20000059A FI109543B (fi) | 1989-07-07 | 2000-01-12 | Menetelmä terapeuttisesti käyttökelpoisen oktreotidipamoaatin valmistamiseksi |
| FI20000060A FI109334B (fi) | 1989-07-07 | 2000-01-12 | Menetelmä pitkäaikaisesti vapautuvan koostumuksen muodostamiseksi |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI20000059A FI109543B (fi) | 1989-07-07 | 2000-01-12 | Menetelmä terapeuttisesti käyttökelpoisen oktreotidipamoaatin valmistamiseksi |
| FI20000060A FI109334B (fi) | 1989-07-07 | 2000-01-12 | Menetelmä pitkäaikaisesti vapautuvan koostumuksen muodostamiseksi |
Country Status (27)
| Country | Link |
|---|---|
| JP (5) | JPH0832624B2 (enExample) |
| KR (2) | KR100303681B1 (enExample) |
| AT (1) | AT406225B (enExample) |
| AU (2) | AU641407B2 (enExample) |
| BE (1) | BE1004486A3 (enExample) |
| CA (1) | CA2020477C (enExample) |
| CH (1) | CH685230A5 (enExample) |
| CY (1) | CY1965A (enExample) |
| DE (2) | DE4042752B4 (enExample) |
| DK (1) | DK175849B1 (enExample) |
| FI (3) | FI108611B (enExample) |
| FR (1) | FR2649319A1 (enExample) |
| GB (2) | GB2234896B (enExample) |
| GR (1) | GR1001121B (enExample) |
| HK (2) | HK97695A (enExample) |
| HU (2) | HU221294B1 (enExample) |
| IE (2) | IE64216B1 (enExample) |
| IL (3) | IL131880A (enExample) |
| IT (1) | IT1241460B (enExample) |
| LU (1) | LU87764A1 (enExample) |
| MY (1) | MY106722A (enExample) |
| NL (1) | NL195027C (enExample) |
| NO (2) | NO302928B1 (enExample) |
| NZ (1) | NZ234384A (enExample) |
| PT (1) | PT94628B (enExample) |
| SE (1) | SE512992C2 (enExample) |
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Families Citing this family (45)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4990336A (en) * | 1989-02-08 | 1991-02-05 | Biosearch, Inc. | Sustained release dosage form |
| YU48420B (sh) * | 1991-03-25 | 1998-07-10 | Hoechst Aktiengesellschaft | Postupak za dobijanje biološki razgradljivih mikročestica sa dugotrajnim delovanjem |
| CH683149A5 (fr) * | 1991-07-22 | 1994-01-31 | Debio Rech Pharma Sa | Procédé pour la préparation de microsphères en matériau polymère biodégradable. |
| US6013853A (en) * | 1992-02-14 | 2000-01-11 | The University Of Texas System | Continuous release polymeric implant carrier |
| US5876452A (en) * | 1992-02-14 | 1999-03-02 | Board Of Regents, University Of Texas System | Biodegradable implant |
| DE4218510A1 (de) * | 1992-06-02 | 1993-12-09 | Pharmatech Gmbh | Verfahren zur Herstellung biologisch abbaubarer Polyester |
| AU4198793A (en) † | 1992-07-24 | 1994-01-27 | Takeda Chemical Industries Ltd. | Microparticle preparation and production thereof |
| JP2944419B2 (ja) * | 1993-05-10 | 1999-09-06 | ノバルティス アクチエンゲゼルシャフト | 持続性遊離組成物中の薬理学的活性成分の安定 |
| US5603960A (en) * | 1993-05-25 | 1997-02-18 | O'hagan; Derek T. | Preparation of microparticles and method of immunization |
| GB9310781D0 (en) * | 1993-05-25 | 1993-07-14 | Davis Stanley S | Preparation of microparticles |
| ATE288270T1 (de) | 1993-11-19 | 2005-02-15 | Janssen Pharmaceutica Nv | Mikroverkapselte 1,2-benzazole |
| US6270795B1 (en) | 1995-11-09 | 2001-08-07 | Microbiological Research Authority | Method of making microencapsulated DNA for vaccination and gene therapy |
| EP0965336A1 (en) | 1995-11-09 | 1999-12-22 | Microbiological Research Authority | Microencapsulated DNA for gene therapy |
| DE19545257A1 (de) | 1995-11-24 | 1997-06-19 | Schering Ag | Verfahren zur Herstellung von morphologisch einheitlichen Mikrokapseln sowie nach diesem Verfahren hergestellte Mikrokapseln |
| US5817343A (en) * | 1996-05-14 | 1998-10-06 | Alkermes, Inc. | Method for fabricating polymer-based controlled-release devices |
| US5968895A (en) * | 1996-12-11 | 1999-10-19 | Praecis Pharmaceuticals, Inc. | Pharmaceutical formulations for sustained drug delivery |
| US6126919A (en) | 1997-02-07 | 2000-10-03 | 3M Innovative Properties Company | Biocompatible compounds for pharmaceutical drug delivery systems |
| GB9810236D0 (en) | 1998-05-13 | 1998-07-08 | Microbiological Res Authority | Improvements relating to encapsulation of bioactive agents |
| US6632457B1 (en) * | 1998-08-14 | 2003-10-14 | Incept Llc | Composite hydrogel drug delivery systems |
| US7107268B1 (en) | 1998-11-12 | 2006-09-12 | Printable Technologies, Inc. | Centralized system and method for managing enterprise operations |
| US6226656B1 (en) | 1998-11-12 | 2001-05-01 | Sourcefinder, Inc. | System and method for creating, generating and processing user-defined generic specs |
| US6204308B1 (en) | 1999-03-01 | 2001-03-20 | Novartis Ag | Organic compounds |
| EP1044683A1 (en) * | 1999-04-15 | 2000-10-18 | Debio Recherche Pharmaceutique S.A. | One-step dispersion method for the microencapsulation of water soluble substances |
| US6461631B1 (en) * | 1999-11-16 | 2002-10-08 | Atrix Laboratories, Inc. | Biodegradable polymer composition |
| KR100392501B1 (ko) * | 2000-06-28 | 2003-07-22 | 동국제약 주식회사 | 다중 에멀젼법에 의한 서방출성 미립구의 제조방법 |
| US6824822B2 (en) * | 2001-08-31 | 2004-11-30 | Alkermes Controlled Therapeutics Inc. Ii | Residual solvent extraction method and microparticles produced thereby |
| AU2002232824A1 (en) | 2000-12-21 | 2002-07-01 | Inhale Therapeutic Systems, Inc. | Induced phase transition method for the production of microparticles containing hydrophobic active agents |
| US20040097419A1 (en) * | 2002-11-19 | 2004-05-20 | Holger Petersen | Organic compounds |
| AR044852A1 (es) * | 2003-06-24 | 2005-10-05 | Novartis Ag | Una composicion farmaceutica para la administracion parenteral que comprende un analogo de somatostatina |
| EP1660039B1 (en) * | 2003-07-18 | 2016-09-28 | Oakwood Laboratories L.L.C. | Prevention of molecular weight reduction of the polymer, impurity formation and gelling in polymer compositions |
| MY158342A (en) | 2003-11-14 | 2016-09-30 | Novartis Ag | Pharmaceutical composition |
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| GB | Transfer or assigment of application |
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Owner name: NOVARTIS AG |