EE05007B1 - 9a-N-(N'-arlkarbamol)- ja 9a-N-(N'-arltiokarbamol)-9-desokso-9a-asa-9a-homoertromtsiini Ahalogeenderivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja kasutamine - Google Patents

9a-N-(N'-arlkarbamol)- ja 9a-N-(N'-arltiokarbamol)-9-desokso-9a-asa-9a-homoertromtsiini Ahalogeenderivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja kasutamine

Info

Publication number
EE05007B1
EE05007B1 EEP200100582A EEP200100582A EE05007B1 EE 05007 B1 EE05007 B1 EE 05007B1 EE P200100582 A EEP200100582 A EE P200100582A EE P200100582 A EEP200100582 A EE P200100582A EE 05007 B1 EE05007 B1 EE 05007B1
Authority
EE
Estonia
Prior art keywords
preparation
meaning
arylthiocarbamoyl
deoxo
arylcarbamoyl
Prior art date
Application number
EEP200100582A
Other languages
English (en)
Estonian (et)
Inventor
Maru�ic- I�tuk Zorica
Kujundzic Nedjelko
Kobrehel Gabrijela
Mutak Stjepan
Mar�ic Nata�a
Original Assignee
PLIVA, farmaceutska industrija, dionicko dru�tvo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by PLIVA, farmaceutska industrija, dionicko dru�tvo filed Critical PLIVA, farmaceutska industrija, dionicko dru�tvo
Publication of EE200100582A publication Critical patent/EE200100582A/xx
Publication of EE05007B1 publication Critical patent/EE05007B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
EEP200100582A 1999-05-03 2000-05-02 9a-N-(N'-arlkarbamol)- ja 9a-N-(N'-arltiokarbamol)-9-desokso-9a-asa-9a-homoertromtsiini Ahalogeenderivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja kasutamine EE05007B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HR990130A HRP990130B1 (en) 1999-05-03 1999-05-03 HALOGEN DERIVATIVES 9a-N-(N'-ARYLCARBAMOYL)- AND 9a-N-(N'-ARYLTHIOCARBAMOYL)-9-DEOXO-9a-AZA-9a OF HOMOERYTHROMYCIN A
PCT/HR2000/000013 WO2000066603A1 (en) 1999-05-03 2000-05-02 Halo derivatives of 9-deoxo-9a-aza-9a-homerythromycin a

Publications (2)

Publication Number Publication Date
EE200100582A EE200100582A (et) 2003-02-17
EE05007B1 true EE05007B1 (et) 2008-04-15

Family

ID=10946916

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100582A EE05007B1 (et) 1999-05-03 2000-05-02 9a-N-(N'-arlkarbamol)- ja 9a-N-(N'-arltiokarbamol)-9-desokso-9a-asa-9a-homoertromtsiini Ahalogeenderivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja kasutamine

Country Status (33)

Country Link
US (1) US6872707B1 (is)
EP (1) EP1175429B1 (is)
JP (1) JP2002543213A (is)
KR (1) KR100714740B1 (is)
CN (1) CN1140535C (is)
AT (1) ATE244258T1 (is)
AU (1) AU767681B2 (is)
BG (1) BG106173A (is)
BR (1) BR0010231A (is)
CA (1) CA2372977A1 (is)
CZ (1) CZ20013913A3 (is)
DE (1) DE60003671T2 (is)
DK (1) DK1175429T3 (is)
EA (1) EA005214B1 (is)
EE (1) EE05007B1 (is)
ES (1) ES2202107T3 (is)
GE (1) GEP20032928B (is)
HK (1) HK1045522B (is)
HR (1) HRP990130B1 (is)
HU (1) HUP0201146A3 (is)
IL (2) IL145986A0 (is)
IS (1) IS6115A (is)
MX (1) MXPA01011038A (is)
NO (1) NO320138B1 (is)
NZ (1) NZ515278A (is)
PL (1) PL351402A1 (is)
PT (1) PT1175429E (is)
SI (1) SI1175429T1 (is)
SK (1) SK284513B6 (is)
TR (1) TR200103143T2 (is)
UA (1) UA71962C2 (is)
WO (1) WO2000066603A1 (is)
ZA (1) ZA200108484B (is)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010146B1 (en) * 2001-02-28 2005-10-31 Pliva D.D. 9a-N-(N'-(PHENYLSULFONYL)CARBAMOYL) DERIVATIVES OF 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMYCIN A AND OF 5-O-DESOSAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHRONOLIDE A
HRP20020885B1 (en) 2002-11-11 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. SUBSTITUTED 9a-N-{N'-[4-(SULFONYL)PHENYLCARBAMOYL]}DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHROMYCIN A AND 5-O-DESOZAMINYL-9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERITHRONOLIDE A
HRP20020886A2 (en) * 2002-11-11 2005-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. SUBSTITUTED 9a-N-[N'-(BENZENSULFONYL)CARBAMOYL-γ-AMINOPROPYL) AND 9a-N(N' -(?-CYANOETHIL)-N' -(b
HRP20020991A2 (en) * 2002-12-12 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. N"-Substituted 9a-N-(N'-carbamoyl-Gamma-aminopropyl), 9a-N-(N'? -thiocarbamoyl-Gamma-aminopropyl), 9a-N-(N'-((Beta-cyanoethyl)-N'-carbamoyl-Gamma? -aminopropyl) and 9a-N-(N'-(Beta-cyanoethyl)-N'-thiocarbamoyl-Gamma? -aminopropyl) derivatives of 9-de
HRP20030381B1 (en) * 2003-05-14 2007-05-31 GlaxoSmithKline istra�iva�ki centar Zagreb d.o.o. 3-DECLADINOZYL 9a-N-CARBAMOYL AND 9a-N-THIOCARBAMOYL DERIVATIVES 9-DEOXO-9-DIHYDRO-9a-AZA-9a-HOMOERYTHROMICYNE A
ES2326002T3 (es) * 2005-01-14 2009-09-28 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. 9a-carbamoil y tiocarbamoil azalidos con actividad antipaludica.
WO2009039177A1 (en) * 2007-09-17 2009-03-26 Enanta Pharmaceuticals, Inc. 6, 11-bicycloides: bridged biaryl macrolide derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU43116B (en) * 1979-04-02 1989-04-30 Pliva Pharm & Chem Works Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
EP0553353A1 (en) * 1990-10-15 1993-08-04 Taisho Pharmaceutical Co. Ltd 2'-modified erythromycin or derivative thereof
HRP931480B1 (en) * 1993-12-08 1997-08-31 Sour Pliva 9a-N-(N'-CARBAMONYL) and 9a-N-(N'-THIOCARBAMONYL) DERIVATES OF 9-DEOXO-9a-HOMOERYTHROMYCIN A

Also Published As

Publication number Publication date
EA200101170A1 (ru) 2002-04-25
PT1175429E (pt) 2003-11-28
EE200100582A (et) 2003-02-17
SI1175429T1 (en) 2003-12-31
HRP990130B1 (en) 2004-06-30
BG106173A (bg) 2002-07-31
CN1140535C (zh) 2004-03-03
KR100714740B1 (ko) 2007-05-07
NO20015346L (no) 2001-11-01
JP2002543213A (ja) 2002-12-17
DE60003671D1 (de) 2003-08-07
HK1045522B (zh) 2004-08-20
NO320138B1 (no) 2005-10-31
CN1351606A (zh) 2002-05-29
US6872707B1 (en) 2005-03-29
SK15702001A3 (sk) 2002-04-04
NZ515278A (en) 2003-06-30
HUP0201146A3 (en) 2003-03-28
HK1045522A1 (en) 2002-11-29
AU4135000A (en) 2000-11-17
IL145986A (en) 2006-10-31
IS6115A (is) 2001-10-19
GEP20032928B (en) 2003-03-25
UA71962C2 (en) 2005-01-17
TR200103143T2 (tr) 2002-04-22
AU767681B2 (en) 2003-11-20
KR20020007397A (ko) 2002-01-26
SK284513B6 (sk) 2005-05-05
ZA200108484B (en) 2003-03-26
EP1175429B1 (en) 2003-07-02
NO20015346D0 (no) 2001-11-01
CA2372977A1 (en) 2000-11-09
DE60003671T2 (de) 2004-06-17
ES2202107T3 (es) 2004-04-01
IL145986A0 (en) 2002-07-25
CZ20013913A3 (cs) 2002-04-17
WO2000066603A1 (en) 2000-11-09
PL351402A1 (en) 2003-04-07
BR0010231A (pt) 2002-02-19
EA005214B1 (ru) 2004-12-30
HRP990130A2 (en) 2001-10-31
HUP0201146A2 (hu) 2002-07-29
EP1175429A1 (en) 2002-01-30
ATE244258T1 (de) 2003-07-15
MXPA01011038A (es) 2002-07-22
DK1175429T3 (da) 2003-10-20

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Legal Events

Date Code Title Description
GB1A Change in the ownership or in the address of the owner
GB1A Change in the ownership or in the address of the owner
KB4A Valid patent at the end of a year

Effective date: 20081231

MM4A Lapsed by not paying the annual fees

Effective date: 20090502