ECSP045140A - Formulaciones farmacéuticas derivadas del platino - Google Patents

Formulaciones farmacéuticas derivadas del platino

Info

Publication number
ECSP045140A
ECSP045140A EC2004005140A ECSP045140A ECSP045140A EC SP045140 A ECSP045140 A EC SP045140A EC 2004005140 A EC2004005140 A EC 2004005140A EC SP045140 A ECSP045140 A EC SP045140A EC SP045140 A ECSP045140 A EC SP045140A
Authority
EC
Ecuador
Prior art keywords
platinum
pharmaceutical formulations
formulations derived
derived
formulas
Prior art date
Application number
EC2004005140A
Other languages
English (en)
Inventor
Sara Lauria
Alessandro Martini
Cristina Ciocca
Original Assignee
Pharmacia Italia Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21744006&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP045140(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacia Italia Spa filed Critical Pharmacia Italia Spa
Publication of ECSP045140A publication Critical patent/ECSP045140A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12Carboxylic acids; Salts or anhydrides thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/555Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/04Antineoplastic agents specific for metastasis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente invención está dirigida a nuevas fórmulas estables de oxaliplatino, en las cuales el ácido láctico y/o una sal farmacéuticamente aceptable funciona como un medio novedoso para preparar una unidad de dosis con una estabilidad mejorada. También está dentro del alcance de esta invención un método para elaborar tales formulaciones listas para ser administradas y su uso en una terapia contra tumores.
EC2004005140A 2001-12-06 2004-06-04 Formulaciones farmacéuticas derivadas del platino ECSP045140A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10/010,122 US6476068B1 (en) 2001-12-06 2001-12-06 Platinum derivative pharmaceutical formulations

Publications (1)

Publication Number Publication Date
ECSP045140A true ECSP045140A (es) 2004-08-27

Family

ID=21744006

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2004005140A ECSP045140A (es) 2001-12-06 2004-06-04 Formulaciones farmacéuticas derivadas del platino

Country Status (41)

Country Link
US (3) US6476068B1 (es)
EP (1) EP1453517B1 (es)
JP (1) JP2005515202A (es)
KR (1) KR100941210B1 (es)
CN (1) CN100540006C (es)
AP (1) AP1760A (es)
AR (1) AR037629A1 (es)
AT (1) ATE317260T1 (es)
AU (1) AU2002352105B2 (es)
BR (1) BR0214757A (es)
CA (1) CA2468916C (es)
CO (1) CO5580776A2 (es)
CR (1) CR7362A (es)
CY (1) CY1105608T1 (es)
DE (1) DE60209145T2 (es)
DK (1) DK1453517T3 (es)
EA (1) EA008090B1 (es)
EC (1) ECSP045140A (es)
ES (1) ES2258661T3 (es)
GE (1) GEP20063895B (es)
HR (1) HRP20040514A2 (es)
HU (1) HUP0402217A3 (es)
IL (2) IL162348A0 (es)
IS (1) IS2580B (es)
MA (1) MA27153A1 (es)
ME (1) MEP10408A (es)
MX (1) MXPA04005423A (es)
MY (1) MY134422A (es)
NO (1) NO330159B1 (es)
NZ (1) NZ533383A (es)
OA (1) OA12739A (es)
PL (1) PL206755B1 (es)
PT (1) PT1453517E (es)
RO (1) RO121509B1 (es)
RS (1) RS50360B (es)
SI (1) SI21493A (es)
TN (1) TNSN04104A1 (es)
TW (1) TW200409640A (es)
UA (1) UA77728C2 (es)
WO (1) WO2003047587A1 (es)
ZA (1) ZA200404525B (es)

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US20040022842A1 (en) * 2002-06-03 2004-02-05 Mebiopharm Co., Ltd. Liposome preparations containing oxaliplatin
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EP2762475A1 (en) * 2003-11-07 2014-08-06 Novartis Vaccines and Diagnostics, Inc. Pharmaceutically acceptable salts of quinolinone compounds and their medical use
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US7795205B2 (en) * 2004-04-12 2010-09-14 Canyon Pharmaceuticals, Inc. Methods for effecting regression of tumor mass and size in a metastasized pancreatic tumor
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US20060063720A1 (en) * 2004-09-22 2006-03-23 Edgar Schridde Oxaliplatin solution concentrate
US20060063833A1 (en) * 2004-09-22 2006-03-23 Edgar Schridde Ready-to-use oxaliplatin solutions
DE102004052877B4 (de) * 2004-11-02 2008-06-19 Ebewe Pharma Ges.M.B.H. Nfg.Kg Stabile wässrige Formulierungen eines Platin-Derivats
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DE102004063764A1 (de) * 2004-12-29 2006-07-13 Hexal Ag Kunststoff-Flasche für Oxaliplatin
JP2006248978A (ja) 2005-03-10 2006-09-21 Mebiopharm Co Ltd 新規なリポソーム製剤
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US9023834B2 (en) * 2008-11-13 2015-05-05 Taigen Biotechnology Co., Ltd. Lyophilization formulation
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CN102274171A (zh) * 2011-08-04 2011-12-14 上海希迪制药有限公司 一种奥沙利铂注射剂
EP2874606B1 (en) 2012-07-18 2019-03-06 Onyx Therapeutics, Inc. Liposomal compositions of epoxyketone-based proteasome inhibitors
JP5929607B2 (ja) * 2012-08-06 2016-06-08 ニプロ株式会社 オキサリプラチン製剤
CN102885765B (zh) * 2012-10-25 2013-11-06 哈药集团生物工程有限公司 一种盐酸伊立替康注射液及其制备方法
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KR101683635B1 (ko) 2014-12-29 2016-12-09 가천대학교 산학협력단 락테이트 금속염을 포함하는 암 치료용 약학 조성물
JP6869899B2 (ja) * 2015-02-13 2021-05-12 サン・ファーマシューティカル・インダストリーズ・リミテッド 静脈内注入剤形
KR102293907B1 (ko) 2015-06-30 2021-08-26 한미약품 주식회사 이리노테칸 함유 경구용 고형제제 및 그 제조방법
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Also Published As

Publication number Publication date
CR7362A (es) 2009-02-12
MEP10408A (en) 2011-02-10
CN100540006C (zh) 2009-09-16
JP2005515202A (ja) 2005-05-26
KR100941210B1 (ko) 2010-02-10
IL162348A0 (en) 2005-11-20
US20030109515A1 (en) 2003-06-12
HUP0402217A3 (en) 2005-11-28
EP1453517A1 (en) 2004-09-08
HRP20040514A2 (en) 2004-10-31
UA77728C2 (en) 2007-01-15
NZ533383A (en) 2007-02-23
ZA200404525B (en) 2005-08-15
ES2258661T3 (es) 2006-09-01
DE60209145T2 (de) 2006-10-26
AR037629A1 (es) 2004-11-17
RS50360B (sr) 2009-11-10
AP2004003055A0 (en) 2004-06-30
MA27153A1 (fr) 2005-01-03
RO121509B1 (ro) 2007-10-30
SI21493A (sl) 2004-12-31
GEP20063895B (en) 2006-08-10
BR0214757A (pt) 2004-09-14
TNSN04104A1 (fr) 2006-06-01
YU59704A (sh) 2006-08-17
HUP0402217A2 (hu) 2005-01-28
NO330159B1 (no) 2011-02-28
HK1072002A1 (zh) 2005-08-12
MY134422A (en) 2007-12-31
IL162348A (en) 2010-11-30
CY1105608T1 (el) 2010-12-22
DK1453517T3 (da) 2006-06-19
EP1453517B1 (en) 2006-02-08
CA2468916C (en) 2009-01-20
US6476068B1 (en) 2002-11-05
CN1612737A (zh) 2005-05-04
KR20050058278A (ko) 2005-06-16
MXPA04005423A (es) 2004-10-11
NO20042842L (no) 2004-07-05
DE60209145D1 (de) 2006-04-20
PL206755B1 (pl) 2010-09-30
EA008090B1 (ru) 2007-02-27
TW200409640A (en) 2004-06-16
CA2468916A1 (en) 2003-06-12
ATE317260T1 (de) 2006-02-15
AP1760A (en) 2007-07-18
IS2580B (is) 2010-02-15
CO5580776A2 (es) 2005-11-30
IS7298A (is) 2004-06-03
PT1453517E (pt) 2006-06-30
OA12739A (en) 2006-06-30
AU2002352105B2 (en) 2009-12-03
US6673805B2 (en) 2004-01-06
US20030109514A1 (en) 2003-06-12
EA200400777A1 (ru) 2004-12-30
AU2002352105A1 (en) 2003-06-17
PL370254A1 (en) 2005-05-16
WO2003047587A1 (en) 2003-06-12

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