MX2020005518A - Mezclas no racemicas y usos de las mismas. - Google Patents

Mezclas no racemicas y usos de las mismas.

Info

Publication number
MX2020005518A
MX2020005518A MX2020005518A MX2020005518A MX2020005518A MX 2020005518 A MX2020005518 A MX 2020005518A MX 2020005518 A MX2020005518 A MX 2020005518A MX 2020005518 A MX2020005518 A MX 2020005518A MX 2020005518 A MX2020005518 A MX 2020005518A
Authority
MX
Mexico
Prior art keywords
amisulpride
disorders
compositions
treatment
amount
Prior art date
Application number
MX2020005518A
Other languages
English (en)
Inventor
Seth Cabot Hopkins
Kenneth Stephen Koblan
John R Snoonian
Harold Scott Wilkinson
Original Assignee
Sunovion Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sunovion Pharmaceuticals Inc filed Critical Sunovion Pharmaceuticals Inc
Publication of MX2020005518A publication Critical patent/MX2020005518A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)

Abstract

Se proporcionan composiciones que comprenden mezclas desiguales de (R)-amisulprida y (S)-amisulprida, o sales farmacéuticamente aceptables de las mismas, donde la cantidad de (R)-amisulprida es mayor que la cantidad de (S)- amisulprida, composiciones y medicamentos que comprenden las mismas usadas para el tratamiento de varias enfermedades y trastornos, y métodos para usarlas para el tratamiento de varias enfermedades y trastornos, que incluyen, de modo no limitante, regímenes de dosis. Además, se proporcionan varias formulaciones de las mismas, incluyendo, pero no limitado a, formulaciones que emplean substancias polimorfas de amisulprida enantiomérica.
MX2020005518A 2017-12-05 2018-12-04 Mezclas no racemicas y usos de las mismas. MX2020005518A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762594883P 2017-12-05 2017-12-05
US201862650613P 2018-03-30 2018-03-30
US201862716804P 2018-08-09 2018-08-09
PCT/US2018/063859 WO2019113079A1 (en) 2017-12-05 2018-12-04 Nonracemic mixtures and uses thereof

Publications (1)

Publication Number Publication Date
MX2020005518A true MX2020005518A (es) 2020-11-06

Family

ID=66657756

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020005518A MX2020005518A (es) 2017-12-05 2018-12-04 Mezclas no racemicas y usos de las mismas.

Country Status (12)

Country Link
US (6) US10369134B2 (es)
EP (1) EP3720434A4 (es)
JP (2) JP7268026B2 (es)
KR (1) KR20200110648A (es)
CN (1) CN112118838A (es)
AU (1) AU2018379992B2 (es)
BR (1) BR112020011189A2 (es)
CA (1) CA3084953A1 (es)
MX (1) MX2020005518A (es)
PH (1) PH12020500543A1 (es)
SG (1) SG11202005016SA (es)
WO (1) WO2019113079A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11377421B2 (en) 2016-11-28 2022-07-05 Lb Pharmaceuticals Inc. Psychotropic agents and uses thereof
BR112019010127A2 (pt) 2016-11-28 2019-08-20 Lb Pharmaceuticals Inc agentes psicotrópicos e usos dos mesmos
CN110944630A (zh) * 2017-05-18 2020-03-31 Lb制药公司 精神药剂及其用途
CN112236138B (zh) 2017-12-05 2024-05-31 赛诺维信制药公司 晶体形式及其制备方法
AU2018379992B2 (en) 2017-12-05 2022-07-21 Sunovion Pharmaceuticals Inc. Nonracemic mixtures and uses thereof
WO2020247603A1 (en) * 2019-06-04 2020-12-10 Sunovion Pharmaceuticals Inc. Modified release formulations and uses thereof
CN114401717A (zh) * 2019-06-04 2022-04-26 赛诺维信制药公司 修饰释放配制品及其用途
JP2024520704A (ja) * 2021-04-01 2024-05-24 サノビオン ファーマシューティカルズ インク アミスルプリドの結晶形態を製造するための方法

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