ECSP034831A - Derivados sustituidos de la 2-piridina ciclohexano-1,4-diamina - Google Patents

Derivados sustituidos de la 2-piridina ciclohexano-1,4-diamina

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Publication number
ECSP034831A
ECSP034831A EC2003004831A ECSP034831A ECSP034831A EC SP034831 A ECSP034831 A EC SP034831A EC 2003004831 A EC2003004831 A EC 2003004831A EC SP034831 A ECSP034831 A EC SP034831A EC SP034831 A ECSP034831 A EC SP034831A
Authority
EC
Ecuador
Prior art keywords
diamine
substituted derivatives
pyridine
cyclhexan
production
Prior art date
Application number
EC2003004831A
Other languages
English (en)
Inventor
Helmut Heinrich Buschmann
Bernd Sundermann
Corinna Maul
Barbara Heller
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of ECSP034831A publication Critical patent/ECSP034831A/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
    • C07C211/36—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing at least two amino groups bound to the carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/132—Amines having two or more amino groups, e.g. spermidine, putrescine
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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  • Neurology (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
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  • Nutrition Science (AREA)
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  • Dermatology (AREA)

Abstract

La presente invención se relaciona con los derivados sustituidos de 2-piridina ciclohexano-1,4-diamina, un proceso para su producción, medicamentos que contienen estos compuestos y el uso de derivados sustituidos de 2-piridina ciclohexano-1,4-diamina para la producción de medicamentos
EC2003004831A 2001-05-09 2003-11-07 Derivados sustituidos de la 2-piridina ciclohexano-1,4-diamina ECSP034831A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10123163A DE10123163A1 (de) 2001-05-09 2001-05-09 Substituierte Cyclohexan-1,4-diaminderivate

Publications (1)

Publication Number Publication Date
ECSP034831A true ECSP034831A (es) 2004-03-23

Family

ID=7684562

Family Applications (2)

Application Number Title Priority Date Filing Date
EC2003004830A ECSP034830A (es) 2001-05-09 2003-11-07 Derivados sustituidos de la ciclohexano-1,4- diamina
EC2003004831A ECSP034831A (es) 2001-05-09 2003-11-07 Derivados sustituidos de la 2-piridina ciclohexano-1,4-diamina

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EC2003004830A ECSP034830A (es) 2001-05-09 2003-11-07 Derivados sustituidos de la ciclohexano-1,4- diamina

Country Status (31)

Country Link
US (3) US6998409B2 (es)
EP (3) EP1392641B1 (es)
JP (3) JP2004533439A (es)
KR (2) KR20040002943A (es)
CN (2) CN1307158C (es)
AR (1) AR035883A1 (es)
AT (2) ATE359260T1 (es)
AU (3) AU2002312883B2 (es)
BR (2) BR0209580A (es)
CA (3) CA2446463C (es)
CO (2) CO5540300A2 (es)
CY (2) CY1106468T1 (es)
CZ (2) CZ20033005A3 (es)
DE (3) DE10123163A1 (es)
DK (2) DK1392641T3 (es)
EC (2) ECSP034830A (es)
ES (2) ES2291486T3 (es)
HK (2) HK1062911A1 (es)
HU (3) HU228253B1 (es)
IL (4) IL158784A0 (es)
MX (3) MXPA03010134A (es)
NO (2) NO326784B1 (es)
NZ (2) NZ529334A (es)
PE (1) PE20021094A1 (es)
PL (3) PL220595B1 (es)
PT (2) PT1392641E (es)
RU (2) RU2321579C2 (es)
SI (2) SI1385825T1 (es)
SK (2) SK286617B6 (es)
WO (3) WO2002090330A1 (es)
ZA (2) ZA200309522B (es)

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WO2004043902A1 (de) 2002-11-12 2004-05-27 Grünenthal GmbH 4-hydroxymethyl-1-aryl-cyclohexylamin-derivative
JP4206382B2 (ja) * 2002-11-19 2009-01-07 アキリオン ファーマシューティカルズ，インコーポレーテッド 置換されたアリールチオウレアおよび関連化合物；ウイルス複製のインヒビター
US7378409B2 (en) * 2003-08-21 2008-05-27 Bristol-Myers Squibb Company Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity
DE10360793A1 (de) * 2003-12-23 2005-07-28 Grünenthal GmbH Spirocyclische Cyclohexan-Derivate
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DE102004023501A1 (de) 2004-05-10 2005-12-01 Grünenthal GmbH Oxosubstituierte Cyclohexyl-1,4-diamin-Derivate
DE102004023635A1 (de) 2004-05-10 2006-04-13 Grünenthal GmbH Heteroarylsubstituierte Cyclohexyl-1,4-diamin-Derivate
DE102004023632A1 (de) 2004-05-10 2005-12-08 Grünenthal GmbH Substituierte Cyclohexylcarbonsäure-Derivate
DE102004023508A1 (de) * 2004-05-10 2005-12-08 Grünenthal GmbH Säurederivate substituierter Cyclohexyl-1,4-diamine
DE102004023506A1 (de) 2004-05-10 2005-12-01 Grünenthal GmbH Kettenverlängerte substituierte Cyclohexyl-1,4-diamin-Derivate
DE102004023507A1 (de) 2004-05-10 2005-12-01 Grünenthal GmbH Substituierte Cyclohexylessigsäure-Derivate
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DE102005061428A1 (de) 2005-12-22 2007-08-16 Grünenthal GmbH Substituierte Cyclohexylmethyl-Derivate
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DE102006035787A1 (de) 2006-07-28 2008-03-13 Tesa Ag Verfahren zum Stanzen von bei Raumtemperatur nicht tackigen hitzeaktivierbaren Klebmassen
US20080194557A1 (en) * 2007-01-18 2008-08-14 Joseph Barbosa Methods and compositions for the treatment of pain, inflammation and cancer
US8003692B2 (en) * 2007-06-15 2011-08-23 Board Of Regents, The University Of Texas System Methods and compositions to inhibit edema factor and adenylyl cyclase
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BR122013017393A2 (pt) 2008-03-27 2019-10-15 Grünenthal GmbH Compostos derivados substituídos de 4-aminociclohexano, medicamentos contendo pelo menos um composto e uso dos referidos compostos
CN102046591B (zh) 2008-03-27 2014-12-03 格吕伦塔尔有限公司 羟甲基环己胺
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DK2324013T6 (en) 2008-07-21 2014-12-15 Purdue Pharma Lp Substituted bridged piperidine compounds of quinoxalintype and uses thereof
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