CY1106468T1 - Υποκατεστημενα παραγωγα κυκλοεξανο-1,4-διαμινης - Google Patents

Υποκατεστημενα παραγωγα κυκλοεξανο-1,4-διαμινης

Info

Publication number
CY1106468T1
CY1106468T1 CY20071100630T CY071100630T CY1106468T1 CY 1106468 T1 CY1106468 T1 CY 1106468T1 CY 20071100630 T CY20071100630 T CY 20071100630T CY 071100630 T CY071100630 T CY 071100630T CY 1106468 T1 CY1106468 T1 CY 1106468T1
Authority
CY
Cyprus
Prior art keywords
substituted cyclohexane
diamine derivatives
preparation
diamine
cyclohexane
Prior art date
Application number
CY20071100630T
Other languages
English (en)
Inventor
Bernd Sundermann
Hagen-Heinrich Hennies
Werner Englberger
Babette-Yvonne Kögel
Original Assignee
Grünenthal GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Grünenthal GmbH filed Critical Grünenthal GmbH
Publication of CY1106468T1 publication Critical patent/CY1106468T1/el

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
    • C07C211/36—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing at least two amino groups bound to the carbon skeleton
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/132—Amines having two or more amino groups, e.g. spermidine, putrescine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404—Indoles, e.g. pindolol
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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Abstract

Η εφεύρεση αφορά υποκατεστημένα παράγωγα κυκλοεξανο-1,4-διαμίνης, μεθόδους για την παρασκευή τους, φάρμακα που περιέχουν τις ενώσεις αυτές και τη χρησιμοποίηση υποκατεστημένων παραγώγων κυκλοεξανο-1,4-διαμίνης για την παρασκευή φαρμάκων.
CY20071100630T 2001-05-09 2007-05-10 Υποκατεστημενα παραγωγα κυκλοεξανο-1,4-διαμινης CY1106468T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10123163A DE10123163A1 (de) 2001-05-09 2001-05-09 Substituierte Cyclohexan-1,4-diaminderivate
PCT/EP2002/005051 WO2002090317A1 (de) 2001-05-09 2002-05-08 Substituierte cyclohexan-1,4-diaminderivate

Publications (1)

Publication Number Publication Date
CY1106468T1 true CY1106468T1 (el) 2012-01-25

Family

ID=7684562

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20071100630T CY1106468T1 (el) 2001-05-09 2007-05-10 Υποκατεστημενα παραγωγα κυκλοεξανο-1,4-διαμινης
CY20071101374T CY1108067T1 (el) 2001-05-09 2007-10-25 Υποκατεστημενα παραγωγα 2-πυριδινο-κυκλοεξανο-1,4-διαμινης

Family Applications After (1)

Application Number Title Priority Date Filing Date
CY20071101374T CY1108067T1 (el) 2001-05-09 2007-10-25 Υποκατεστημενα παραγωγα 2-πυριδινο-κυκλοεξανο-1,4-διαμινης

Country Status (31)

Country Link
US (3) US7276518B2 (el)
EP (3) EP1385825B1 (el)
JP (3) JP2004528374A (el)
KR (2) KR100895778B1 (el)
CN (2) CN1307158C (el)
AR (1) AR035883A1 (el)
AT (2) ATE370120T1 (el)
AU (3) AU2002312883B2 (el)
BR (2) BR0209579A (el)
CA (3) CA2446461C (el)
CO (2) CO5540300A2 (el)
CY (2) CY1106468T1 (el)
CZ (2) CZ20033005A3 (el)
DE (3) DE10123163A1 (el)
DK (2) DK1385825T3 (el)
EC (2) ECSP034830A (el)
ES (2) ES2284876T3 (el)
HK (2) HK1062911A1 (el)
HU (3) HU228253B1 (el)
IL (4) IL158784A0 (el)
MX (3) MXPA03010201A (el)
NO (2) NO328600B1 (el)
NZ (2) NZ529334A (el)
PE (1) PE20021094A1 (el)
PL (3) PL220595B1 (el)
PT (2) PT1385825E (el)
RU (2) RU2287523C2 (el)
SI (2) SI1385825T1 (el)
SK (2) SK286617B6 (el)
WO (3) WO2002090317A1 (el)
ZA (2) ZA200309521B (el)

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DE102004023501A1 (de) 2004-05-10 2005-12-01 Grünenthal GmbH Oxosubstituierte Cyclohexyl-1,4-diamin-Derivate
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CN104203914B (zh) 2011-10-20 2017-07-11 奥瑞泽恩基因组学股份有限公司 作为lsd1抑制剂的(杂)芳基环丙胺化合物
CN103958474B (zh) 2011-10-20 2017-03-08 奥莱松基因组股份有限公司 作为lsd1抑制剂的(杂)芳基环丙基胺化合物
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