DK2402325T3 - Hydroxylerede cyclopenta[d]pyrimidiner som AKT-proteinkinaseinhibitorer - Google Patents

Hydroxylerede cyclopenta[d]pyrimidiner som AKT-proteinkinaseinhibitorer Download PDF

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Publication number
DK2402325T3
DK2402325T3 DK11166125.2T DK11166125T DK2402325T3 DK 2402325 T3 DK2402325 T3 DK 2402325T3 DK 11166125 T DK11166125 T DK 11166125T DK 2402325 T3 DK2402325 T3 DK 2402325T3
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alkyl
cancer
mmol
compound
optionally substituted
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DK11166125.2T
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Danish (da)
English (en)
Inventor
Ian S Mitchell
James F Blake
Rui Xu
Nicholas C Kallan
Dengming Xiao
Keith Lee Spencer
Josef R Bencsik
Jun Liang
Brian Safina
Birong Zhang
Christine Chabot
Steven Do
Eli W Wallace
Anna L Banka
Stephen T Schlachter
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Array Biopharma Inc
Genentech Inc
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Application filed by Array Biopharma Inc, Genentech Inc filed Critical Array Biopharma Inc
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Publication of DK2402325T3 publication Critical patent/DK2402325T3/en

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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DK11166125.2T 2006-07-06 2007-07-05 Hydroxylerede cyclopenta[d]pyrimidiner som AKT-proteinkinaseinhibitorer DK2402325T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81871806P 2006-07-06 2006-07-06
EP07799337A EP2049501B1 (en) 2006-07-06 2007-07-05 Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors

Publications (1)

Publication Number Publication Date
DK2402325T3 true DK2402325T3 (en) 2015-12-07

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ID=38686743

Family Applications (2)

Application Number Title Priority Date Filing Date
DK07799337.6T DK2049501T3 (da) 2006-07-06 2007-07-05 Hydroxyleret og methoxyleret cyclopenta [D]-pyrimidiner som AKT-proteinkinase-inhibitorer
DK11166125.2T DK2402325T3 (en) 2006-07-06 2007-07-05 Hydroxylerede cyclopenta[d]pyrimidiner som AKT-proteinkinaseinhibitorer

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DK07799337.6T DK2049501T3 (da) 2006-07-06 2007-07-05 Hydroxyleret og methoxyleret cyclopenta [D]-pyrimidiner som AKT-proteinkinase-inhibitorer

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EP (4) EP2966065A3 (OSRAM)
JP (4) JP5266216B2 (OSRAM)
KR (5) KR101578877B1 (OSRAM)
CN (2) CN101578273B (OSRAM)
AR (3) AR061842A1 (OSRAM)
AT (1) ATE524447T1 (OSRAM)
AU (1) AU2007269060B2 (OSRAM)
BR (3) BR122013028012B8 (OSRAM)
CA (2) CA2656622C (OSRAM)
CL (1) CL2007001993A1 (OSRAM)
CO (1) CO6150161A2 (OSRAM)
CR (1) CR10600A (OSRAM)
CY (1) CY1112117T1 (OSRAM)
DK (2) DK2049501T3 (OSRAM)
ES (3) ES2554228T3 (OSRAM)
HR (1) HRP20110908T1 (OSRAM)
HU (1) HUE026237T2 (OSRAM)
IL (2) IL196028A (OSRAM)
IN (1) IN2014KN02886A (OSRAM)
MA (1) MA31655B1 (OSRAM)
MX (4) MX377920B (OSRAM)
MY (1) MY147364A (OSRAM)
NO (1) NO342346B1 (OSRAM)
NZ (3) NZ597647A (OSRAM)
PL (2) PL2402325T3 (OSRAM)
PT (1) PT2049501E (OSRAM)
RS (1) RS52212B (OSRAM)
RU (2) RU2478632C2 (OSRAM)
SG (4) SG185980A1 (OSRAM)
SI (2) SI2049501T1 (OSRAM)
TW (2) TW201332994A (OSRAM)
UA (1) UA95641C2 (OSRAM)
WO (1) WO2008006040A1 (OSRAM)
ZA (1) ZA200900070B (OSRAM)

Families Citing this family (52)

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US8063050B2 (en) 2006-07-06 2011-11-22 Array Biopharma Inc. Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors
UA95641C2 (xx) * 2006-07-06 2011-08-25 Эррей Биофарма Инк. Гідроксильовані піримідильні циклопентани як інгібітори акт протеїнкінази$гидроксилированные пиримидильные циклопентаны как ингибиторы акт протеинкиназы
ES2372955T3 (es) 2006-07-06 2012-01-30 Array Biopharma, Inc. Ciclopenta[d]pirimidinas como inhibidores de la proteína cinasa akt.
JP5231411B2 (ja) * 2006-07-06 2013-07-10 アレイ バイオファーマ、インコーポレイテッド Ａｋｔプロテインキナーゼ阻害剤としてのジヒドロチエノピリミジン
ATE493418T1 (de) 2006-07-06 2011-01-15 Array Biopharma Inc Dihydrofuropyrimidine als akt- proteinkinaseinhibitoren
WO2008115511A1 (en) 2007-03-20 2008-09-25 Peak Biosciences, Inc. Method for therapeutic administration of radionucleosides
NZ582692A (en) 2007-07-05 2012-05-25 Array Biopharma Inc Pyrimidyl cyclopentanes as akt protein kinase inhibitors
US9409886B2 (en) 2007-07-05 2016-08-09 Array Biopharma Inc. Pyrimidyl cyclopentanes as AKT protein kinase inhibitors
US8846683B2 (en) 2007-07-05 2014-09-30 Array Biopharma, Inc. Pyrimidyl cyclopentanes as Akt protein kinase inhibitors
US8377937B2 (en) 2007-07-05 2013-02-19 Array Biopharma Inc. Pyrimidyl cyclopentanes as AKT protein kinase inhibitors
CA2711692A1 (en) * 2008-01-09 2009-07-16 Array Biopharma Inc. Hydroxylated pyrimidyl cyclopentane as akt protein kinase inhibitor
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