DK2081955T3 - Metastinderivater og anvendelse deraf - Google Patents
Metastinderivater og anvendelse deraf Download PDFInfo
- Publication number
- DK2081955T3 DK2081955T3 DK07830903.6T DK07830903T DK2081955T3 DK 2081955 T3 DK2081955 T3 DK 2081955T3 DK 07830903 T DK07830903 T DK 07830903T DK 2081955 T3 DK2081955 T3 DK 2081955T3
- Authority
- DK
- Denmark
- Prior art keywords
- metastin derivatives
- metastin
- derivatives
- Prior art date
Links
- KAHDONZOCXSKII-NJVVDGNHSA-N kisspeptin Chemical class C([C@@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CCC(N)=O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C=CC=CC=1)C(N)=O)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H]1N(CCC1)C(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H]1N(CCC1)C(=O)[C@H]1N(CCC1)C(=O)[C@H]1N(CCC1)C(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)CN)[C@@H](C)O)C1=CN=CN1 KAHDONZOCXSKII-NJVVDGNHSA-N 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
- C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
- C07K14/4702—Regulators; Modulating activity
- C07K14/4703—Inhibitors; Suppressors
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
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- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
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- Biomedical Technology (AREA)
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- Reproductive Health (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Zoology (AREA)
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- Physical Education & Sports Medicine (AREA)
- Molecular Biology (AREA)
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- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
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- Pain & Pain Management (AREA)
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- Obesity (AREA)
- Pregnancy & Childbirth (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2006290536 | 2006-10-25 | ||
| JP2007021387 | 2007-01-31 | ||
| JP2007221911 | 2007-08-28 | ||
| PCT/JP2007/071169 WO2008050897A1 (en) | 2006-10-25 | 2007-10-24 | Metastin derivatives and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK2081955T3 true DK2081955T3 (da) | 2015-06-15 |
Family
ID=38925530
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK07830903.6T DK2081955T3 (da) | 2006-10-25 | 2007-10-24 | Metastinderivater og anvendelse deraf |
Country Status (33)
| Country | Link |
|---|---|
| US (2) | US8765909B2 (OSRAM) |
| EP (1) | EP2081955B1 (OSRAM) |
| JP (2) | JP2010507565A (OSRAM) |
| KR (1) | KR101424306B1 (OSRAM) |
| AR (1) | AR063367A1 (OSRAM) |
| AU (1) | AU2007309969B2 (OSRAM) |
| BR (1) | BRPI0717441B8 (OSRAM) |
| CA (1) | CA2667537C (OSRAM) |
| CL (1) | CL2007003053A1 (OSRAM) |
| CR (1) | CR10799A (OSRAM) |
| CY (1) | CY1116627T1 (OSRAM) |
| DK (1) | DK2081955T3 (OSRAM) |
| EC (1) | ECSP099279A (OSRAM) |
| ES (1) | ES2539430T3 (OSRAM) |
| GE (1) | GEP20125568B (OSRAM) |
| HR (1) | HRP20150819T1 (OSRAM) |
| HU (1) | HUE025291T2 (OSRAM) |
| IL (1) | IL198046A (OSRAM) |
| JO (1) | JO3048B1 (OSRAM) |
| MA (1) | MA30887B1 (OSRAM) |
| ME (1) | ME00786B (OSRAM) |
| MX (1) | MX2009004148A (OSRAM) |
| MY (1) | MY145975A (OSRAM) |
| NO (1) | NO341584B1 (OSRAM) |
| NZ (1) | NZ576375A (OSRAM) |
| PE (1) | PE20081469A1 (OSRAM) |
| PL (1) | PL2081955T3 (OSRAM) |
| PT (1) | PT2081955E (OSRAM) |
| RS (1) | RS54083B1 (OSRAM) |
| SI (1) | SI2081955T1 (OSRAM) |
| TN (1) | TN2009000140A1 (OSRAM) |
| TW (1) | TWI404726B (OSRAM) |
| WO (1) | WO2008050897A1 (OSRAM) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2004063221A1 (ja) | 2002-12-26 | 2004-07-29 | Takeda Pharmaceutical Company Limited | メタスチン誘導体およびその用途 |
| PE20091567A1 (es) * | 2004-06-25 | 2009-11-03 | Takeda Pharmaceutical | Derivados de metastina en el tratamiento del cancer |
| US20090093615A1 (en) * | 2005-12-22 | 2009-04-09 | Takeda Pharmaceutical Company Limited | Metastin derivatives and use thereof |
| US20090099334A1 (en) * | 2005-12-22 | 2009-04-16 | Takeda Pharmaceutical Company Limited | Metastin derivatives and use thereof |
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