BRPI0717441B8 - composto, medicamento, e, uso do derivado de metastina - Google Patents

composto, medicamento, e, uso do derivado de metastina

Info

Publication number
BRPI0717441B8
BRPI0717441B8 BRPI0717441A BRPI0717441A BRPI0717441B8 BR PI0717441 B8 BRPI0717441 B8 BR PI0717441B8 BR PI0717441 A BRPI0717441 A BR PI0717441A BR PI0717441 A BRPI0717441 A BR PI0717441A BR PI0717441 B8 BRPI0717441 B8 BR PI0717441B8
Authority
BR
Brazil
Prior art keywords
suppressing activity
metastin
activity
hormone secretion
present
Prior art date
Application number
BRPI0717441A
Other languages
English (en)
Portuguese (pt)
Inventor
Nishizawa Naoki
Asami Taiji
Original Assignee
Takeda Pharmaceuticals Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceuticals Co filed Critical Takeda Pharmaceuticals Co
Publication of BRPI0717441A2 publication Critical patent/BRPI0717441A2/pt
Publication of BRPI0717441B1 publication Critical patent/BRPI0717441B1/pt
Publication of BRPI0717441B8 publication Critical patent/BRPI0717441B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4702—Regulators; Modulating activity
    • C07K14/4703—Inhibitors; Suppressors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • A61K38/1709—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Reproductive Health (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Molecular Biology (AREA)
  • Toxicology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Pregnancy & Childbirth (AREA)
BRPI0717441A 2006-10-25 2007-10-24 composto, medicamento, e, uso do derivado de metastina BRPI0717441B8 (pt)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2006290536 2006-10-25
JP2006-290536 2006-10-25
JP2007021387 2007-01-31
JP2007-021387 2007-01-31
JP2007-221911 2007-08-28
JP2007221911 2007-08-28
PCT/JP2007/071169 WO2008050897A1 (en) 2006-10-25 2007-10-24 Metastin derivatives and use thereof

Publications (3)

Publication Number Publication Date
BRPI0717441A2 BRPI0717441A2 (pt) 2013-11-19
BRPI0717441B1 BRPI0717441B1 (pt) 2019-07-02
BRPI0717441B8 true BRPI0717441B8 (pt) 2021-05-25

Family

ID=38925530

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0717441A BRPI0717441B8 (pt) 2006-10-25 2007-10-24 composto, medicamento, e, uso do derivado de metastina

Country Status (33)

Country Link
US (2) US8765909B2 (OSRAM)
EP (1) EP2081955B1 (OSRAM)
JP (2) JP2010507565A (OSRAM)
KR (1) KR101424306B1 (OSRAM)
AR (1) AR063367A1 (OSRAM)
AU (1) AU2007309969B2 (OSRAM)
BR (1) BRPI0717441B8 (OSRAM)
CA (1) CA2667537C (OSRAM)
CL (1) CL2007003053A1 (OSRAM)
CR (1) CR10799A (OSRAM)
CY (1) CY1116627T1 (OSRAM)
DK (1) DK2081955T3 (OSRAM)
EC (1) ECSP099279A (OSRAM)
ES (1) ES2539430T3 (OSRAM)
GE (1) GEP20125568B (OSRAM)
HR (1) HRP20150819T1 (OSRAM)
HU (1) HUE025291T2 (OSRAM)
IL (1) IL198046A (OSRAM)
JO (1) JO3048B1 (OSRAM)
MA (1) MA30887B1 (OSRAM)
ME (1) ME00786B (OSRAM)
MX (1) MX2009004148A (OSRAM)
MY (1) MY145975A (OSRAM)
NO (1) NO341584B1 (OSRAM)
NZ (1) NZ576375A (OSRAM)
PE (1) PE20081469A1 (OSRAM)
PL (1) PL2081955T3 (OSRAM)
PT (1) PT2081955E (OSRAM)
RS (1) RS54083B1 (OSRAM)
SI (1) SI2081955T1 (OSRAM)
TN (1) TN2009000140A1 (OSRAM)
TW (1) TWI404726B (OSRAM)
WO (1) WO2008050897A1 (OSRAM)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004063221A1 (ja) 2002-12-26 2004-07-29 Takeda Pharmaceutical Company Limited メタスチン誘導体およびその用途
PE20091567A1 (es) * 2004-06-25 2009-11-03 Takeda Pharmaceutical Derivados de metastina en el tratamiento del cancer
US20090093615A1 (en) * 2005-12-22 2009-04-09 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US20090099334A1 (en) * 2005-12-22 2009-04-16 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US8404643B2 (en) 2005-12-22 2013-03-26 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
TWI386417B (zh) 2005-12-22 2013-02-21 Takeda Pharmaceutical 轉移抑素衍生物及其用途
WO2007125619A1 (ja) * 2006-04-26 2007-11-08 Kyoto University Ｇｐｒ５４アゴニスト活性を有する新規化合物
TWI404726B (zh) 2006-10-25 2013-08-11 Takeda Pharmaceutical 腫瘤轉移抑制素衍生物及其用途
US8110639B2 (en) * 2006-11-17 2012-02-07 Solvay Advanced Polymers, L.L.C. Transparent and flame retardant polysulfone compositions
US20110118172A1 (en) * 2008-04-24 2011-05-19 Takeda Pharmaceutical Company Limited Metastin derivative and use thereof
EP2275433B1 (en) * 2008-04-30 2017-06-07 Kyoto University Metastin derivative and use thereof
ES2617657T3 (es) 2008-07-30 2017-06-19 Takeda Pharmaceutical Company Limited Derivado de metastina y uso del mismo
WO2010137022A1 (en) * 2009-05-27 2010-12-02 Yeda Research And Development Co. Ltd Gpr54 agonists or antagonists for treatment of diseases presenting behavioral abnormalities
KR20130097088A (ko) * 2010-06-25 2013-09-02 다케다 야쿠힌 고교 가부시키가이샤 서방성 제제
EP2755690B1 (en) 2011-08-04 2020-04-01 Merck Sharp & Dohme B.V. Kisspeptide-pentasaccharide conjugates
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PT2081955E (pt) 2015-07-10
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CA2667537C (en) 2017-01-17
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US7786083B2 (en) 2010-08-31
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