DK2081955T3 - Metastinderivater og anvendelse deraf - Google Patents

Metastinderivater og anvendelse deraf Download PDF

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Publication number
DK2081955T3
DK2081955T3 DK07830903.6T DK07830903T DK2081955T3 DK 2081955 T3 DK2081955 T3 DK 2081955T3 DK 07830903 T DK07830903 T DK 07830903T DK 2081955 T3 DK2081955 T3 DK 2081955T3
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Prior art keywords
metastin derivatives
metastin
derivatives
Prior art date
Application number
DK07830903.6T
Other languages
English (en)
Inventor
Taiji Asami
Naoki Nishizawa
Original Assignee
Takeda Pharmaceutical
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Publication of DK2081955T3 publication Critical patent/DK2081955T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4702—Regulators; Modulating activity
    • C07K14/4703—Inhibitors; Suppressors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • A61K38/1709—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • A—HUMAN NECESSITIES
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DK07830903.6T 2006-10-25 2007-10-24 Metastinderivater og anvendelse deraf DK2081955T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2006290536 2006-10-25
JP2007021387 2007-01-31
JP2007221911 2007-08-28
PCT/JP2007/071169 WO2008050897A1 (en) 2006-10-25 2007-10-24 Metastin derivatives and use thereof

Publications (1)

Publication Number Publication Date
DK2081955T3 true DK2081955T3 (da) 2015-06-15

Family

ID=38925530

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07830903.6T DK2081955T3 (da) 2006-10-25 2007-10-24 Metastinderivater og anvendelse deraf

Country Status (34)

Country Link
US (2) US7786083B2 (da)
EP (1) EP2081955B1 (da)
JP (2) JP2010507565A (da)
KR (1) KR101424306B1 (da)
AR (1) AR063367A1 (da)
AU (1) AU2007309969B2 (da)
BR (1) BRPI0717441B8 (da)
CA (1) CA2667537C (da)
CL (1) CL2007003053A1 (da)
CR (1) CR10799A (da)
CY (1) CY1116627T1 (da)
DK (1) DK2081955T3 (da)
EC (1) ECSP099279A (da)
ES (1) ES2539430T3 (da)
GE (1) GEP20125568B (da)
HK (1) HK1130500A1 (da)
HR (1) HRP20150819T1 (da)
HU (1) HUE025291T2 (da)
IL (1) IL198046A (da)
JO (1) JO3048B1 (da)
MA (1) MA30887B1 (da)
ME (1) ME00786B (da)
MX (1) MX2009004148A (da)
MY (1) MY145975A (da)
NO (1) NO341584B1 (da)
NZ (1) NZ576375A (da)
PE (1) PE20081469A1 (da)
PL (1) PL2081955T3 (da)
PT (1) PT2081955E (da)
RS (1) RS54083B1 (da)
SI (1) SI2081955T1 (da)
TN (1) TN2009000140A1 (da)
TW (1) TWI404726B (da)
WO (1) WO2008050897A1 (da)

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WO2004063221A1 (ja) * 2002-12-26 2004-07-29 Takeda Pharmaceutical Company Limited メタスチン誘導体およびその用途
SG153865A1 (en) * 2004-06-25 2009-07-29 Takeda Pharmaceutical Metastin derivatives and use thereof
US20090093615A1 (en) * 2005-12-22 2009-04-09 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US20090099334A1 (en) * 2005-12-22 2009-04-16 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
US8404643B2 (en) * 2005-12-22 2013-03-26 Takeda Pharmaceutical Company Limited Metastin derivatives and use thereof
TWI386417B (zh) 2005-12-22 2013-02-21 Takeda Pharmaceutical 轉移抑素衍生物及其用途
JP5279021B2 (ja) * 2006-04-26 2013-09-04 国立大学法人京都大学 Ｇｐｒ５４アゴニスト活性を有する新規化合物
TWI404726B (zh) 2006-10-25 2013-08-11 Takeda Pharmaceutical 腫瘤轉移抑制素衍生物及其用途
US8110639B2 (en) * 2006-11-17 2012-02-07 Solvay Advanced Polymers, L.L.C. Transparent and flame retardant polysulfone compositions
EP2277900A4 (en) * 2008-04-24 2011-08-03 Takeda Pharmaceutical METASTIN DERIVATIVE AND USE THEREOF
WO2009139298A1 (ja) * 2008-04-30 2009-11-19 国立大学法人京都大学 メタスチン誘導体およびその用途
ES2617657T3 (es) 2008-07-30 2017-06-19 Takeda Pharmaceutical Company Limited Derivado de metastina y uso del mismo
US8716228B2 (en) 2009-05-27 2014-05-06 Yeda Research And Development Co. Ltd. GPR54 agonists or antagonists for treatment of diseases presenting behavioral abnormalities
KR20130097088A (ko) * 2010-06-25 2013-09-02 다케다 야쿠힌 고교 가부시키가이샤 서방성 제제
US9127038B2 (en) 2011-08-04 2015-09-08 Merck Sharp & Dohme Corp. Kisspeptide-pentasaccharide conjugates
AU2014280593B2 (en) * 2013-06-12 2018-11-08 Merck Patent Gmbh Hydroxy-ethylene derivatives for the treatment of arthrosis
WO2015112703A1 (en) * 2014-01-22 2015-07-30 The Johns Hopkins University Compositions and methods for treating diabetes
JP6253146B2 (ja) * 2014-02-04 2017-12-27 国立大学法人山口大学 新規なペプチド誘導体及びこれを含有する医薬
EP3253774B1 (en) * 2015-02-08 2018-11-21 Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. Peptides for the treatment of malignant proliferative diseases
US11427615B2 (en) 2017-07-05 2022-08-30 Xdcexplorer (Shanghai) Co., Ltd. Peptide compound and application thereof, and composition containing peptide compound
TWI795462B (zh) * 2017-11-17 2023-03-11 日商鹽野義製藥股份有限公司 光安定性及溶出性優異的醫藥製劑

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IL198046A0 (en) 2011-08-01
JO3048B1 (ar) 2016-09-05
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PT2081955E (pt) 2015-07-10
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AR063367A1 (es) 2009-01-21
CL2007003053A1 (es) 2008-08-08
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IL198046A (en) 2014-06-30
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CA2667537C (en) 2017-01-17
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