DK175842B1 - Prostaglandinderivater til behandling af glaukom eller foröget okulært tryk - Google Patents

Prostaglandinderivater til behandling af glaukom eller foröget okulært tryk Download PDF

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Publication number
DK175842B1
DK175842B1 DK199001121A DK112190A DK175842B1 DK 175842 B1 DK175842 B1 DK 175842B1 DK 199001121 A DK199001121 A DK 199001121A DK 112190 A DK112190 A DK 112190A DK 175842 B1 DK175842 B1 DK 175842B1
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Prior art keywords
phenyl
trinor
prostaglandin derivative
groups
group
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DK199001121A
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Danish (da)
English (en)
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DK112190A (da
DK112190D0 (da
Inventor
Johan W Stjernschantz
Bahram Resul
Original Assignee
Pharmacia Ab
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26660291&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK175842(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from SE8803110A external-priority patent/SE8803110D0/xx
Application filed by Pharmacia Ab filed Critical Pharmacia Ab
Publication of DK112190A publication Critical patent/DK112190A/da
Publication of DK112190D0 publication Critical patent/DK112190D0/da
Priority to DK200401645A priority Critical patent/DK176053B1/da
Application granted granted Critical
Publication of DK175842B1 publication Critical patent/DK175842B1/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/557Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5578Eicosanoids, e.g. leukotrienes or prostaglandins having a pentalene ring system, e.g. carbacyclin, iloprost
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK199001121A 1988-09-06 1990-05-04 Prostaglandinderivater til behandling af glaukom eller foröget okulært tryk DK175842B1 (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK200401645A DK176053B1 (da) 1988-09-06 2004-10-27 Prostaglandinderivater til behandling af glaukom eller foröget okulært tryk

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
SE8803110 1988-09-06
SE8803110A SE8803110D0 (sv) 1988-09-06 1988-09-06 Prostaglandinderivat for behandling av glaukom eller okuler hypertension
SE8803855 1988-10-28
SE8803855 1988-10-28
SE8900475 1989-02-13
PCT/SE1989/000475 WO1990002553A1 (en) 1988-09-06 1989-09-06 Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension

Publications (3)

Publication Number Publication Date
DK112190A DK112190A (da) 1990-05-04
DK112190D0 DK112190D0 (da) 1990-05-04
DK175842B1 true DK175842B1 (da) 2005-03-29

Family

ID=26660291

Family Applications (1)

Application Number Title Priority Date Filing Date
DK199001121A DK175842B1 (da) 1988-09-06 1990-05-04 Prostaglandinderivater til behandling af glaukom eller foröget okulært tryk

Country Status (13)

Country Link
US (6) US5422368A (es)
EP (6) EP0569046B1 (es)
JP (3) JP2721414B2 (es)
AT (3) ATE227576T1 (es)
DE (5) DE68929563D1 (es)
DK (1) DK175842B1 (es)
ES (5) ES2186670T3 (es)
FI (1) FI92690C (es)
HK (2) HK1048106A1 (es)
HU (1) HU211593A9 (es)
LU (1) LU91541I2 (es)
NL (1) NL970039I2 (es)
WO (1) WO1990002553A1 (es)

Families Citing this family (253)

* Cited by examiner, † Cited by third party
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EP1225168A2 (en) 2002-07-24
JPH1081624A (ja) 1998-03-31
EP1224935A3 (en) 2003-03-26
EP0569046B1 (en) 2002-11-13
EP1348437A3 (en) 2003-11-19
US5849791A (en) 1998-12-15
ES2213504T1 (es) 2004-09-01
NL970039I2 (nl) 1998-04-01
DE68929563D1 (de) 2009-03-05
EP0364417B9 (en) 2004-10-06
ES2317964T5 (es) 2015-02-20
US6030999A (en) 2000-02-29
EP1225168B8 (en) 2015-03-18
ATE101342T1 (de) 1994-02-15
ES2062102T5 (es) 2004-12-01
US5422368A (en) 1995-06-06
EP1225168B1 (en) 2009-01-14
EP0364417B1 (en) 1994-02-09
EP1224934A2 (en) 2002-07-24
US5627208A (en) 1997-05-06
JP2721414B2 (ja) 1998-03-04
EP1225168A3 (en) 2003-03-26
DE68929435T2 (de) 2003-07-17
NL970039I1 (nl) 1998-02-02
FI902258A0 (fi) 1990-05-04
ATE420857T1 (de) 2009-01-15
AU4189889A (en) 1990-04-02
AU625096B2 (en) 1992-07-02
DE68913000T2 (de) 1994-06-16
LU91541I2 (fr) 2009-05-11
US5578618A (en) 1996-11-26

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