DK169538B1 - Aminoalkoholer og syreadditionssalte deraf, fremgangsmåde til deres fremstilling og lægemidler med indhold af sådanne - Google Patents

Aminoalkoholer og syreadditionssalte deraf, fremgangsmåde til deres fremstilling og lægemidler med indhold af sådanne Download PDF

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Publication number
DK169538B1
DK169538B1 DK040687A DK40687A DK169538B1 DK 169538 B1 DK169538 B1 DK 169538B1 DK 040687 A DK040687 A DK 040687A DK 40687 A DK40687 A DK 40687A DK 169538 B1 DK169538 B1 DK 169538B1
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DK
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Prior art keywords
formula
compounds
alkyl
compound
methyl
Prior art date
Application number
DK040687A
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Danish (da)
English (en)
Other versions
DK40687A (da
DK40687D0 (da
Inventor
Gilbert Aubard
Jacques Bure
Pierre Alain Calvet
Claude Gouret
Genevieve Agnes Grouhel
Jean-Louis Junien
Original Assignee
Jouveinal Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jouveinal Sa filed Critical Jouveinal Sa
Publication of DK40687D0 publication Critical patent/DK40687D0/da
Publication of DK40687A publication Critical patent/DK40687A/da
Application granted granted Critical
Publication of DK169538B1 publication Critical patent/DK169538B1/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
    • C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/092—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Heat Treatment Of Sheet Steel (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DK040687A 1986-01-30 1987-01-26 Aminoalkoholer og syreadditionssalte deraf, fremgangsmåde til deres fremstilling og lægemidler med indhold af sådanne DK169538B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8601295 1986-01-30
FR8601295A FR2593499B1 (fr) 1986-01-30 1986-01-30 Aminoalcools, leur procede de preparation et leurs applications, notamment en therapeutique

Publications (3)

Publication Number Publication Date
DK40687D0 DK40687D0 (da) 1987-01-26
DK40687A DK40687A (da) 1987-07-31
DK169538B1 true DK169538B1 (da) 1994-11-28

Family

ID=9331637

Family Applications (1)

Application Number Title Priority Date Filing Date
DK040687A DK169538B1 (da) 1986-01-30 1987-01-26 Aminoalkoholer og syreadditionssalte deraf, fremgangsmåde til deres fremstilling og lægemidler med indhold af sådanne

Country Status (17)

Country Link
US (1) US4994617A (el)
EP (1) EP0237366B1 (el)
JP (1) JPH089580B2 (el)
KR (1) KR950006891B1 (el)
AT (1) ATE42540T1 (el)
AU (1) AU590664B2 (el)
BR (1) BR1100977A (el)
CA (1) CA1294961C (el)
DE (1) DE3760117D1 (el)
DK (1) DK169538B1 (el)
ES (1) ES2008109B3 (el)
FI (1) FI87068C (el)
FR (1) FR2593499B1 (el)
GR (1) GR3000026T3 (el)
IE (1) IE59448B1 (el)
NZ (1) NZ218988A (el)
PT (1) PT84223B (el)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4939133A (en) * 1985-10-01 1990-07-03 Warner-Lambert Company N-substituted-2-hydroxy-α-oxo-benzeneacetamides and pharmaceutical compositions having activity as modulators of the arachidonic acid cascade
US5482947A (en) * 1990-11-19 1996-01-09 Talley; John J. Retroviral protease inhibitors
FR2690916B1 (fr) * 1992-05-05 1994-06-17 Jouveinal Inst Rech Nouveaux enantiomeres derives du (s)-amino-2-(dichloro-3,4-benzyl)-2-propanol-1.
US5472970A (en) * 1992-05-05 1995-12-05 Institut De Recherche Jouveinal S.A. Allylaminoesters and their application in therapeutics
FR2690917B1 (fr) * 1992-05-05 1994-06-17 Jouveinal Inst Rech Aminoesters, leur procede de preparation et leur application en therapeutique.
US5367094A (en) * 1993-06-04 1994-11-22 Yukong, Ltd. Convenient process for the preparation of chiral or racemic phenylalaninols and their N-blocked derivatives
FR2761686B1 (fr) * 1997-04-07 1999-05-14 Sipsy Sa Nouveau procede de preparation du (+/-)3-(3,4- dichlorophenyl)-2-dimethylamino-2-methyl-propan-1-ol ou cericlamine (inn)
US7216702B2 (en) * 2003-02-28 2007-05-15 Yates Petroleum Corporation Methods of evaluating undersaturated coalbed methane reservoirs
AU2004305563C1 (en) 2003-12-11 2011-07-07 Sunovion Pharmaceuticals Inc. Combination of a sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression
US7467260B2 (en) * 2004-10-08 2008-12-16 International Business Machines Corporation Method and apparatus to purge remote node cache lines to support hot node replace in a computing system
CZ301920B6 (cs) * 2009-06-16 2010-07-28 Zentiva, K. S. Zpusob výroby (S)-4-methylamino-3-(3,4-dichlorfenyl)butan-1-olu

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3132179A (en) * 1959-08-27 1964-05-05 Sterling Drug Inc Ethers of alpha-hydroxymethyl-beta-monocarbocyclic aryl ethyl amines and their preparation
US3193581A (en) * 1961-03-01 1965-07-06 Yamanouchi Pharma Co Ltd Process of preparing 1-phenyl-2-aminopropane
US3573304A (en) * 1968-12-03 1971-03-30 Delalande Sa 1-dimethylamino - 3 - methyl-2(pyridyl or pyridazinyl) pentane and the corresponding non-toxic acid addition salts thereof
US3706764A (en) * 1969-04-16 1972-12-19 Yoshitomi Pharmaceutical Phenethylaminomethyl-chromanones and- thiochromanones
US3896166A (en) * 1970-05-06 1975-07-22 Hoffmann La Roche Formyl-substituted tyrosine
NL7112938A (el) * 1970-09-30 1972-04-05
ES399820A1 (es) * 1971-02-17 1975-07-01 Sandoz Ag Procedimiento para la obtencion de derivados de amino pro- panol.
GB1346401A (en) * 1971-05-12 1974-02-13 Lepetit Spa Cardioactive arylaminobutanols
US4058642A (en) * 1973-10-11 1977-11-15 Boehringer Ingelheim Gmbh 2-Amino-3-(3'-hydroxy-phenyl)-propanols and salts thereof
GB1434826A (en) * 1973-11-14 1976-05-05 Gallardo Antonio Sa Esters and carbamates of aminoalkanols
US4536601A (en) * 1982-09-28 1985-08-20 Dainippon Pharmaceutical Co., Ltd. Optically active N-substituted phenylalaninols and use thereof

Also Published As

Publication number Publication date
BR1100977A (pt) 1999-10-13
DK40687A (da) 1987-07-31
ATE42540T1 (de) 1989-05-15
EP0237366A1 (fr) 1987-09-16
US4994617A (en) 1991-02-19
JPH089580B2 (ja) 1996-01-31
GR3000026T3 (en) 1990-01-19
FI870418A (fi) 1987-07-31
KR870007101A (ko) 1987-08-14
EP0237366B1 (fr) 1989-04-26
ES2008109B3 (es) 1989-07-16
JPS62190150A (ja) 1987-08-20
AU6795987A (en) 1987-08-06
NZ218988A (en) 1990-02-26
AU590664B2 (en) 1989-11-09
FI87068C (fi) 1992-11-25
FI870418A0 (fi) 1987-01-30
CA1294961C (en) 1992-01-28
FR2593499B1 (fr) 1988-08-12
PT84223B (pt) 1989-05-31
KR950006891B1 (ko) 1995-06-26
FI87068B (fi) 1992-08-14
FR2593499A1 (fr) 1987-07-31
IE59448B1 (en) 1994-02-23
DK40687D0 (da) 1987-01-26
DE3760117D1 (en) 1989-06-01
PT84223A (fr) 1987-02-01
IE870062L (en) 1987-07-30

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B1 Patent granted (law 1993)
PBP Patent lapsed

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