DK141622B - Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. - Google Patents
Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. Download PDFInfo
- Publication number
- DK141622B DK141622B DK439776AA DK439776A DK141622B DK 141622 B DK141622 B DK 141622B DK 439776A A DK439776A A DK 439776AA DK 439776 A DK439776 A DK 439776A DK 141622 B DK141622 B DK 141622B
- Authority
- DK
- Denmark
- Prior art keywords
- compound
- group
- general formula
- carbon atoms
- dihydroxyphenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
- C07C213/04—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reaction of ammonia or amines with olefin oxides or halohydrins
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
- C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
- C07D265/32—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings with oxygen atoms directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Immunology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE7510988 | 1975-10-01 | ||
| SE7510988A SE7510988L (sv) | 1975-10-01 | 1975-10-01 | Nya farmaceutiskt aktiva foreningar |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK439776A DK439776A (cs) | 1977-04-02 |
| DK141622B true DK141622B (da) | 1980-05-12 |
Family
ID=20325688
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK439776AA DK141622B (da) | 1975-10-01 | 1976-09-30 | Analogifremgangsmåde til fremstilling af racemiske eller optisk aktive 1-(3,5-dihydroxyfenyl)-2-aminoætanolderivater eller syreadditionssalte deraf. |
Country Status (19)
| Country | Link |
|---|---|
| JP (1) | JPS5242840A (cs) |
| AT (1) | AT347427B (cs) |
| AU (1) | AU503212B2 (cs) |
| BE (1) | BE846837A (cs) |
| CS (2) | CS199643B2 (cs) |
| DD (1) | DD126278A5 (cs) |
| DE (1) | DE2640972A1 (cs) |
| DK (1) | DK141622B (cs) |
| ES (1) | ES451979A1 (cs) |
| FI (1) | FI762660A (cs) |
| FR (1) | FR2326183A1 (cs) |
| GB (1) | GB1542317A (cs) |
| LU (1) | LU75916A1 (cs) |
| NL (1) | NL7610845A (cs) |
| NO (1) | NO763345L (cs) |
| NZ (1) | NZ182165A (cs) |
| SE (1) | SE7510988L (cs) |
| SU (2) | SU638252A3 (cs) |
| ZA (1) | ZA765331B (cs) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4419364A (en) | 1980-07-09 | 1983-12-06 | Aktiebolaget Draco | Bronchospasmolytic carbamate derivatives |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0103830A3 (de) * | 1982-09-22 | 1985-07-31 | Bayer Ag | Wachstumsfördernde Phenylethylamin-Derivate |
| PL2332921T3 (pl) | 2003-06-17 | 2016-08-31 | Arena Pharm Inc | Chlorowodorek 8-chloro-1-metylo-2,3,4,5-tetrahydro-1H-3-benzazepiny |
| EP2471779A1 (en) | 2006-04-03 | 2012-07-04 | Arena Pharmaceuticals, Inc. | Process for the resolution of a mixture of (R)- and (S)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine |
| ES2522587T3 (es) | 2006-12-05 | 2014-11-17 | Arena Pharmaceuticals, Inc. | Procesos para preparar (R)-8-cloro-1-metil-2,3,4,5-tetrahidro-1H-3-benzacepina e intermedios de la misma |
| WO2009111004A1 (en) | 2008-03-04 | 2009-09-11 | Arena Pharmaceuticals, Inc. | Processes for the preparation of intermediates related to the 5-ht2c agonist (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine |
| US8952197B2 (en) | 2009-06-18 | 2015-02-10 | Arena Pharmaceuticals, Inc. | Processes for the preparation of 5-HT2C receptor agonists |
| KR20130112848A (ko) | 2010-06-02 | 2013-10-14 | 아레나 파마슈티칼스, 인크. | 5-ｈｔ2ｃ 수용체 아고니스트의 제조 방법 |
| CN103347523A (zh) | 2010-09-01 | 2013-10-09 | 艾尼纳制药公司 | 向具有肾损伤的个体给药氯卡色林 |
| CA2808909A1 (en) | 2010-09-01 | 2012-03-08 | Arena Pharmaceuticals, Inc. | Salts of lorcaserin with optically active acids |
| KR20180118801A (ko) | 2010-09-01 | 2018-10-31 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 체중 관리에 유용한 5-ｈｔ2ｃ 작동제의 변형-방출 투여 형태 |
| WO2012030957A2 (en) | 2010-09-01 | 2012-03-08 | Arena Pharmaceuticals, Inc. | Non-hygroscopic salts of 5-ht2c agonists |
| BR112015007779A2 (pt) | 2012-10-09 | 2017-07-04 | Arena Pharm Inc | célula de fluxo de permeabilidade e sistema de condutância hidráulica |
-
1975
- 1975-10-01 SE SE7510988A patent/SE7510988L/xx unknown
-
1976
- 1976-09-07 ZA ZA765331A patent/ZA765331B/xx unknown
- 1976-09-11 DE DE19762640972 patent/DE2640972A1/de not_active Withdrawn
- 1976-09-15 AT AT682376A patent/AT347427B/de not_active IP Right Cessation
- 1976-09-16 FI FI762660A patent/FI762660A/fi not_active Application Discontinuation
- 1976-09-22 SU SU762402852A patent/SU638252A3/ru active
- 1976-09-27 NZ NZ182165A patent/NZ182165A/xx unknown
- 1976-09-27 AU AU18122/76A patent/AU503212B2/en not_active Expired
- 1976-09-28 DD DD195022A patent/DD126278A5/xx unknown
- 1976-09-30 GB GB7640684A patent/GB1542317A/en not_active Expired
- 1976-09-30 ES ES451979A patent/ES451979A1/es not_active Expired
- 1976-09-30 NL NL7610845A patent/NL7610845A/xx not_active Application Discontinuation
- 1976-09-30 DK DK439776AA patent/DK141622B/da unknown
- 1976-09-30 NO NO763345A patent/NO763345L/no unknown
- 1976-09-30 FR FR7629467A patent/FR2326183A1/fr not_active Withdrawn
- 1976-09-30 LU LU75916A patent/LU75916A1/xx unknown
- 1976-10-01 BE BE171148A patent/BE846837A/xx unknown
- 1976-10-01 CS CS766357A patent/CS199643B2/cs unknown
- 1976-10-01 JP JP51118924A patent/JPS5242840A/ja active Pending
- 1976-10-01 CS CS782253A patent/CS199644B2/cs unknown
-
1977
- 1977-10-13 SU SU772532454A patent/SU674669A3/ru active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4419364A (en) | 1980-07-09 | 1983-12-06 | Aktiebolaget Draco | Bronchospasmolytic carbamate derivatives |
Also Published As
| Publication number | Publication date |
|---|---|
| AT347427B (de) | 1978-12-27 |
| SU638252A3 (ru) | 1978-12-15 |
| ZA765331B (en) | 1977-08-31 |
| GB1542317A (en) | 1979-03-14 |
| NL7610845A (nl) | 1977-04-05 |
| NO763345L (cs) | 1977-04-04 |
| SU674669A3 (ru) | 1979-07-15 |
| BE846837A (fr) | 1977-04-01 |
| SE7510988L (sv) | 1977-04-02 |
| ES451979A1 (es) | 1978-01-01 |
| FR2326183A1 (fr) | 1977-04-29 |
| FI762660A (cs) | 1977-04-02 |
| NZ182165A (en) | 1978-07-10 |
| ATA682376A (de) | 1978-05-15 |
| CS199643B2 (en) | 1980-07-31 |
| AU503212B2 (en) | 1979-08-30 |
| DD126278A5 (cs) | 1977-07-06 |
| DK439776A (cs) | 1977-04-02 |
| AU1812276A (en) | 1978-04-06 |
| JPS5242840A (en) | 1977-04-04 |
| DE2640972A1 (de) | 1977-04-14 |
| LU75916A1 (cs) | 1978-05-16 |
| CS199644B2 (en) | 1980-07-31 |
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