DK0797579T3 - Erythromycin A-9-O-oxim-derivater udstyret med antibiotisk aktivitet - Google Patents

Erythromycin A-9-O-oxim-derivater udstyret med antibiotisk aktivitet

Info

Publication number
DK0797579T3
DK0797579T3 DK95941076T DK95941076T DK0797579T3 DK 0797579 T3 DK0797579 T3 DK 0797579T3 DK 95941076 T DK95941076 T DK 95941076T DK 95941076 T DK95941076 T DK 95941076T DK 0797579 T3 DK0797579 T3 DK 0797579T3
Authority
DK
Denmark
Prior art keywords
erythromycin
antibiotic activity
oxime derivatives
derivatives equipped
oxime
Prior art date
Application number
DK95941076T
Other languages
Danish (da)
English (en)
Inventor
Franco Pellacini
Enrico Albini
Daniela Botta
Stefano Romagnano
Giovanna Schioppacassi
Francesco Santangelo
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Application granted granted Critical
Publication of DK0797579T3 publication Critical patent/DK0797579T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK95941076T 1994-12-13 1995-12-07 Erythromycin A-9-O-oxim-derivater udstyret med antibiotisk aktivitet DK0797579T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT94MI002496A IT1276901B1 (it) 1994-12-13 1994-12-13 Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica
PCT/EP1995/004815 WO1996018633A1 (en) 1994-12-13 1995-12-07 Erythromycin a 9-0-oxime derivatives endowed with antibiotic activity

Publications (1)

Publication Number Publication Date
DK0797579T3 true DK0797579T3 (da) 2000-06-05

Family

ID=11369979

Family Applications (1)

Application Number Title Priority Date Filing Date
DK95941076T DK0797579T3 (da) 1994-12-13 1995-12-07 Erythromycin A-9-O-oxim-derivater udstyret med antibiotisk aktivitet

Country Status (35)

Country Link
US (1) US5847092A (fi)
EP (1) EP0797579B1 (fi)
JP (1) JPH10510520A (fi)
KR (1) KR100367559B1 (fi)
CN (1) CN1046535C (fi)
AP (1) AP739A (fi)
AT (1) ATE190620T1 (fi)
AU (1) AU690791B2 (fi)
BG (1) BG63261B1 (fi)
BR (1) BR9510015A (fi)
CA (1) CA2207029A1 (fi)
CZ (1) CZ289943B6 (fi)
DE (1) DE69515694T2 (fi)
DK (1) DK0797579T3 (fi)
EE (1) EE03401B1 (fi)
ES (1) ES2144154T3 (fi)
FI (1) FI972493A0 (fi)
GE (1) GEP20012391B (fi)
GR (1) GR3033622T3 (fi)
HU (1) HU220631B1 (fi)
IT (1) IT1276901B1 (fi)
LT (1) LT4276B (fi)
LV (1) LV11898B (fi)
MD (1) MD1788G2 (fi)
NO (1) NO309816B1 (fi)
NZ (1) NZ297446A (fi)
OA (1) OA10491A (fi)
PL (1) PL182053B1 (fi)
PT (1) PT797579E (fi)
RO (1) RO116282B1 (fi)
RU (1) RU2152951C1 (fi)
SI (1) SI9520124A (fi)
TJ (1) TJ306B (fi)
UA (1) UA48958C2 (fi)
WO (1) WO1996018633A1 (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1290447B1 (it) 1997-03-28 1998-12-03 Zambon Spa Derivati 1,3-ossatiolanici ad attivita' antivirale
IT1301967B1 (it) * 1998-07-30 2000-07-20 Zambon Spa Derivato di eritromicina ad attivita' antibiotica
IT1301968B1 (it) * 1998-07-30 2000-07-20 Zambon Spa Derivati di eritromicina ad attivita' antibiotica
IT1306205B1 (it) * 1999-01-15 2001-05-30 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
US6947844B2 (en) 2000-08-09 2005-09-20 Yale University Modulators of ribosomal function and identification thereof
US6638908B1 (en) 2000-08-09 2003-10-28 Yale University Crystals of the large ribosomal subunit
IL151012A0 (en) 2001-08-03 2003-02-12 Ribosomes Structure And Protei Ribosomes structure and protein synthesis inhibitors
US6952650B2 (en) 2001-08-03 2005-10-04 Yale University Modulators of ribosomal function and identification thereof
ITMI20021726A1 (it) 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
JP5383037B2 (ja) 2004-02-27 2014-01-08 リブ−エックス ファーマシューティカルズ,インコーポレイテッド 大環状化合物およびそれらを製造し使用する方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2473525A1 (fr) * 1980-01-11 1981-07-17 Roussel Uclaf Nouvelles oximes derivees de l'erythromycine, leur procede de preparation et leur application comme medicaments
GB8521402D0 (en) 1985-08-28 1985-10-02 Beecham Group Plc Chemical compounds
US4740502A (en) * 1986-06-20 1988-04-26 Abbott Laboratories Semisynthetic erythromycin antibiotics
PT86800B (pt) 1987-02-24 1992-05-29 Beecham Group Plc Processo para a preparacao de derivados de eritromicina
US5302705A (en) * 1989-10-07 1994-04-12 Taisho Pharmaceutical Co., Ltd. 6-O-methylerythromycin a oxime derivatives
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin

Also Published As

Publication number Publication date
DE69515694D1 (de) 2000-04-20
AP9700989A0 (en) 1997-07-31
CN1046535C (zh) 1999-11-17
NO972702L (no) 1997-08-13
JPH10510520A (ja) 1998-10-13
PL320688A1 (en) 1997-10-27
LV11898B (en) 1998-03-20
MD1788F2 (en) 2001-11-30
MD1788G2 (ro) 2002-05-31
KR100367559B1 (ko) 2003-04-21
AU4260396A (en) 1996-07-03
HU220631B1 (hu) 2002-03-28
CN1169727A (zh) 1998-01-07
PT797579E (pt) 2000-08-31
US5847092A (en) 1998-12-08
RO116282B1 (ro) 2000-12-29
GR3033622T3 (en) 2000-10-31
WO1996018633A1 (en) 1996-06-20
CA2207029A1 (en) 1996-06-20
OA10491A (en) 2002-04-10
FI972493A (fi) 1997-06-12
TJ306B (en) 2001-08-06
MD970243A (en) 1999-05-31
BG101570A (en) 1998-02-27
MX9704253A (es) 1997-09-30
EE03401B1 (et) 2001-04-16
BG63261B1 (bg) 2001-07-31
BR9510015A (pt) 1997-10-28
PL182053B1 (pl) 2001-10-31
AP739A (en) 1999-03-24
CZ178697A3 (en) 1997-12-17
ITMI942496A0 (it) 1994-12-13
EP0797579B1 (en) 2000-03-15
ITMI942496A1 (it) 1996-06-13
LT4276B (lt) 1998-01-26
CZ289943B6 (cs) 2002-04-17
LV11898A (lv) 1997-12-20
IT1276901B1 (it) 1997-11-03
ATE190620T1 (de) 2000-04-15
ES2144154T3 (es) 2000-06-01
DE69515694T2 (de) 2000-10-26
NZ297446A (en) 1999-06-29
UA48958C2 (uk) 2002-09-16
GEP20012391B (en) 2001-03-25
EE9700124A (et) 1997-12-15
NO309816B1 (no) 2001-04-02
HUT77126A (hu) 1998-03-02
RU2152951C1 (ru) 2000-07-20
LT97116A (en) 1997-10-27
SI9520124A (sl) 1998-04-30
FI972493A0 (fi) 1997-06-12
EP0797579A1 (en) 1997-10-01
AU690791B2 (en) 1998-04-30
NO972702D0 (no) 1997-06-12

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