IT1301968B1 - Derivati di eritromicina ad attivita' antibiotica - Google Patents
Derivati di eritromicina ad attivita' antibioticaInfo
- Publication number
- IT1301968B1 IT1301968B1 IT1998MI001776A ITMI981776A IT1301968B1 IT 1301968 B1 IT1301968 B1 IT 1301968B1 IT 1998MI001776 A IT1998MI001776 A IT 1998MI001776A IT MI981776 A ITMI981776 A IT MI981776A IT 1301968 B1 IT1301968 B1 IT 1301968B1
- Authority
- IT
- Italy
- Prior art keywords
- erythromycin derivatives
- antibiotic activity
- erythromycin
- derivatives
- preparing
- Prior art date
Links
- ULGZDMOVFRHVEP-RWJQBGPGSA-N Erythromycin Chemical class O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)C(=O)[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 ULGZDMOVFRHVEP-RWJQBGPGSA-N 0.000 title abstract 3
- 230000003115 biocidal effect Effects 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Priority Applications (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
| US09/744,244 US6468979B1 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
| ES99938386T ES2215396T3 (es) | 1998-07-30 | 1999-07-27 | Derivados de eritromicina con actividad antibiotica. |
| PCT/EP1999/005485 WO2000006606A2 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
| DE69915487T DE69915487T2 (de) | 1998-07-30 | 1999-07-27 | Erythromycin-derivate mit antibiotischer wirkung |
| EP99938386A EP1100762B1 (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
| AU52901/99A AU5290199A (en) | 1998-07-30 | 1999-07-27 | Erythromycin derivatives with antibiotic activity |
| AT99938386T ATE261425T1 (de) | 1998-07-30 | 1999-07-27 | Erythromycin-derivate mit antibiotischer wirkung |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITMI981776A0 ITMI981776A0 (it) | 1998-07-30 |
| ITMI981776A1 ITMI981776A1 (it) | 2000-01-30 |
| IT1301968B1 true IT1301968B1 (it) | 2000-07-20 |
Family
ID=11380563
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT1998MI001776A IT1301968B1 (it) | 1998-07-30 | 1998-07-30 | Derivati di eritromicina ad attivita' antibiotica |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US6468979B1 (it) |
| EP (1) | EP1100762B1 (it) |
| AT (1) | ATE261425T1 (it) |
| AU (1) | AU5290199A (it) |
| DE (1) | DE69915487T2 (it) |
| ES (1) | ES2215396T3 (it) |
| IT (1) | IT1301968B1 (it) |
| WO (1) | WO2000006606A2 (it) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6947844B2 (en) * | 2000-08-09 | 2005-09-20 | Yale University | Modulators of ribosomal function and identification thereof |
| US6638908B1 (en) * | 2000-08-09 | 2003-10-28 | Yale University | Crystals of the large ribosomal subunit |
| US6952650B2 (en) | 2001-08-03 | 2005-10-04 | Yale University | Modulators of ribosomal function and identification thereof |
| IL151012A0 (en) * | 2001-08-03 | 2003-02-12 | Ribosomes Structure And Protei | Ribosomes structure and protein synthesis inhibitors |
| AR043050A1 (es) * | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
| CA2517970A1 (en) * | 2003-03-05 | 2004-09-16 | Rib-X Pharmaceuticals, Inc. | Bifunctional heterocyclic compounds and methods of making and using the same |
| KR20060015602A (ko) | 2003-05-31 | 2006-02-17 | 마이크로메트 에이지 | EpCAM 에 대한 이중 특이성 항체를 포함하는약학조성물 |
| US20070149463A1 (en) * | 2003-10-30 | 2007-06-28 | Oyelere Adegboyega K | Bifunctional macrolide heterocyclic compounds and methods of making and using the same |
| US20070270357A1 (en) * | 2003-11-18 | 2007-11-22 | Farmer Jay J | Bifunctional Macrolide Heterocyclic Compounds and Methods of Making and Using the Same |
| JP5383037B2 (ja) | 2004-02-27 | 2014-01-08 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | 大環状化合物およびそれらを製造し使用する方法 |
| EP1928893A2 (en) | 2005-08-24 | 2008-06-11 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
| JP5953308B2 (ja) | 2010-10-22 | 2016-07-20 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | 殺害虫剤としての新規ヘテロ環式化合物 |
| US10537558B2 (en) | 2015-06-01 | 2020-01-21 | Bantam Pharmaceutical, Llc | Substituted pyrazole and pyrrole compounds and methods for using them for inhibition of initiation of translation and treatment of diseases and disorders relating thereto |
| CN110603254B (zh) | 2016-11-30 | 2024-04-12 | 班塔姆制药有限责任公司 | 被取代的吡唑化合物以及使用其治疗过度增生性疾病的方法 |
| JP2020513403A (ja) | 2016-11-30 | 2020-05-14 | バンタム、ファーマシューティカル、リミテッド、ライアビリティー、カンパニーBantam Pharmaceutical, Llc | 置換ピラゾールおよびピロール化合物の使用する方法ならびに過剰増殖性疾患の治療のための方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1276901B1 (it) * | 1994-12-13 | 1997-11-03 | Zambon Spa | Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica |
-
1998
- 1998-07-30 IT IT1998MI001776A patent/IT1301968B1/it active IP Right Grant
-
1999
- 1999-07-27 ES ES99938386T patent/ES2215396T3/es not_active Expired - Lifetime
- 1999-07-27 EP EP99938386A patent/EP1100762B1/en not_active Expired - Lifetime
- 1999-07-27 AT AT99938386T patent/ATE261425T1/de not_active IP Right Cessation
- 1999-07-27 AU AU52901/99A patent/AU5290199A/en not_active Abandoned
- 1999-07-27 DE DE69915487T patent/DE69915487T2/de not_active Expired - Fee Related
- 1999-07-27 US US09/744,244 patent/US6468979B1/en not_active Expired - Fee Related
- 1999-07-27 WO PCT/EP1999/005485 patent/WO2000006606A2/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| ATE261425T1 (de) | 2004-03-15 |
| AU5290199A (en) | 2000-02-21 |
| DE69915487T2 (de) | 2005-02-17 |
| DE69915487D1 (de) | 2004-04-15 |
| ITMI981776A0 (it) | 1998-07-30 |
| WO2000006606A3 (en) | 2000-05-04 |
| ES2215396T3 (es) | 2004-10-01 |
| EP1100762B1 (en) | 2004-03-10 |
| US6468979B1 (en) | 2002-10-22 |
| WO2000006606A2 (en) | 2000-02-10 |
| ITMI981776A1 (it) | 2000-01-30 |
| EP1100762A2 (en) | 2001-05-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted |