IT1301968B1 - Derivati di eritromicina ad attivita' antibiotica - Google Patents

Derivati di eritromicina ad attivita' antibiotica

Info

Publication number
IT1301968B1
IT1301968B1 IT1998MI001776A ITMI981776A IT1301968B1 IT 1301968 B1 IT1301968 B1 IT 1301968B1 IT 1998MI001776 A IT1998MI001776 A IT 1998MI001776A IT MI981776 A ITMI981776 A IT MI981776A IT 1301968 B1 IT1301968 B1 IT 1301968B1
Authority
IT
Italy
Prior art keywords
erythromycin derivatives
antibiotic activity
erythromycin
derivatives
preparing
Prior art date
Application number
IT1998MI001776A
Other languages
English (en)
Inventor
Franco Pellacini
Daniela Botta
Enrico Albini
Domenico Ungheri
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of ITMI981776A0 publication Critical patent/ITMI981776A0/it
Priority to IT1998MI001776A priority Critical patent/IT1301968B1/it
Priority to DE69915487T priority patent/DE69915487T2/de
Priority to ES99938386T priority patent/ES2215396T3/es
Priority to PCT/EP1999/005485 priority patent/WO2000006606A2/en
Priority to US09/744,244 priority patent/US6468979B1/en
Priority to EP99938386A priority patent/EP1100762B1/en
Priority to AU52901/99A priority patent/AU5290199A/en
Priority to AT99938386T priority patent/ATE261425T1/de
Publication of ITMI981776A1 publication Critical patent/ITMI981776A1/it
Application granted granted Critical
Publication of IT1301968B1 publication Critical patent/IT1301968B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IT1998MI001776A 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica IT1301968B1 (it)

Priority Applications (8)

Application Number Priority Date Filing Date Title
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica
US09/744,244 US6468979B1 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
ES99938386T ES2215396T3 (es) 1998-07-30 1999-07-27 Derivados de eritromicina con actividad antibiotica.
PCT/EP1999/005485 WO2000006606A2 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
DE69915487T DE69915487T2 (de) 1998-07-30 1999-07-27 Erythromycin-derivate mit antibiotischer wirkung
EP99938386A EP1100762B1 (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
AU52901/99A AU5290199A (en) 1998-07-30 1999-07-27 Erythromycin derivatives with antibiotic activity
AT99938386T ATE261425T1 (de) 1998-07-30 1999-07-27 Erythromycin-derivate mit antibiotischer wirkung

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica

Publications (3)

Publication Number Publication Date
ITMI981776A0 ITMI981776A0 (it) 1998-07-30
ITMI981776A1 ITMI981776A1 (it) 2000-01-30
IT1301968B1 true IT1301968B1 (it) 2000-07-20

Family

ID=11380563

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1998MI001776A IT1301968B1 (it) 1998-07-30 1998-07-30 Derivati di eritromicina ad attivita' antibiotica

Country Status (8)

Country Link
US (1) US6468979B1 (it)
EP (1) EP1100762B1 (it)
AT (1) ATE261425T1 (it)
AU (1) AU5290199A (it)
DE (1) DE69915487T2 (it)
ES (1) ES2215396T3 (it)
IT (1) IT1301968B1 (it)
WO (1) WO2000006606A2 (it)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6947844B2 (en) * 2000-08-09 2005-09-20 Yale University Modulators of ribosomal function and identification thereof
US6638908B1 (en) * 2000-08-09 2003-10-28 Yale University Crystals of the large ribosomal subunit
US6952650B2 (en) 2001-08-03 2005-10-04 Yale University Modulators of ribosomal function and identification thereof
IL151012A0 (en) * 2001-08-03 2003-02-12 Ribosomes Structure And Protei Ribosomes structure and protein synthesis inhibitors
AR043050A1 (es) * 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
CA2517970A1 (en) * 2003-03-05 2004-09-16 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using the same
KR20060015602A (ko) 2003-05-31 2006-02-17 마이크로메트 에이지 EpCAM 에 대한 이중 특이성 항체를 포함하는약학조성물
US20070149463A1 (en) * 2003-10-30 2007-06-28 Oyelere Adegboyega K Bifunctional macrolide heterocyclic compounds and methods of making and using the same
US20070270357A1 (en) * 2003-11-18 2007-11-22 Farmer Jay J Bifunctional Macrolide Heterocyclic Compounds and Methods of Making and Using the Same
JP5383037B2 (ja) 2004-02-27 2014-01-08 リブ−エックス ファーマシューティカルズ,インコーポレイテッド 大環状化合物およびそれらを製造し使用する方法
EP1928893A2 (en) 2005-08-24 2008-06-11 Rib-X Pharmaceuticals, Inc. Triazole compounds and methods of making and using the same
JP5953308B2 (ja) 2010-10-22 2016-07-20 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH 殺害虫剤としての新規ヘテロ環式化合物
US10537558B2 (en) 2015-06-01 2020-01-21 Bantam Pharmaceutical, Llc Substituted pyrazole and pyrrole compounds and methods for using them for inhibition of initiation of translation and treatment of diseases and disorders relating thereto
CN110603254B (zh) 2016-11-30 2024-04-12 班塔姆制药有限责任公司 被取代的吡唑化合物以及使用其治疗过度增生性疾病的方法
JP2020513403A (ja) 2016-11-30 2020-05-14 バンタム、ファーマシューティカル、リミテッド、ライアビリティー、カンパニーBantam Pharmaceutical, Llc 置換ピラゾールおよびピロール化合物の使用する方法ならびに過剰増殖性疾患の治療のための方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1276901B1 (it) * 1994-12-13 1997-11-03 Zambon Spa Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica

Also Published As

Publication number Publication date
ATE261425T1 (de) 2004-03-15
AU5290199A (en) 2000-02-21
DE69915487T2 (de) 2005-02-17
DE69915487D1 (de) 2004-04-15
ITMI981776A0 (it) 1998-07-30
WO2000006606A3 (en) 2000-05-04
ES2215396T3 (es) 2004-10-01
EP1100762B1 (en) 2004-03-10
US6468979B1 (en) 2002-10-22
WO2000006606A2 (en) 2000-02-10
ITMI981776A1 (it) 2000-01-30
EP1100762A2 (en) 2001-05-23

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Legal Events

Date Code Title Description
0001 Granted